KR102496504B1 - 남성 피임을 위한 비호르몬 조성물 및 방법 - Google Patents
남성 피임을 위한 비호르몬 조성물 및 방법 Download PDFInfo
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- KR102496504B1 KR102496504B1 KR1020207029031A KR20207029031A KR102496504B1 KR 102496504 B1 KR102496504 B1 KR 102496504B1 KR 1020207029031 A KR1020207029031 A KR 1020207029031A KR 20207029031 A KR20207029031 A KR 20207029031A KR 102496504 B1 KR102496504 B1 KR 102496504B1
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- silodosin
- alpha
- azoospermia
- contraception
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
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- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
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| PCT/EP2019/057267 WO2019180217A1 (en) | 2018-03-23 | 2019-03-22 | Non-hormonal compositions and methods for male contraception |
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| AU2023384256A1 (en) * | 2022-11-23 | 2025-03-20 | Pharmajor Incorporated | Modified-release silodosin compositions and use thereof in methods for male contraception |
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| US1091276A (en) | 1911-12-09 | 1914-03-24 | Basf Ag | Producing unsaturated terpene hydrocarbons. |
| US4210644A (en) | 1978-02-23 | 1980-07-01 | The Johns Hopkins University | Male contraception |
| DE4308406C1 (de) | 1993-03-12 | 1994-06-16 | Jenapharm Gmbh | Kombinationspräparat zur Kontrazeption |
| HUP0300128A3 (en) | 2000-02-15 | 2004-03-29 | Schering Ag | Male contraceptive composition comprising norethisterone and its use |
| FR2861990B1 (fr) * | 2003-11-10 | 2006-02-10 | Nouveaux Produits Pharma | Comprimes faiblement doses a reseau de polymeres |
| US20090186896A1 (en) * | 2005-09-29 | 2009-07-23 | Bayer Healthcare Ag | PDE Inhibitors and Combinations Thereof for the Treatment of Urological Disorders |
| CN101316934A (zh) * | 2005-09-29 | 2008-12-03 | 拜耳医药保健股份公司 | 用于治疗泌尿系统疾病的pde抑制剂及其组合 |
| MX2009003737A (es) * | 2006-10-05 | 2009-06-16 | Panacea Biotec Ltd | Composicion inyectable en deposito y su procedimiento de preparacion. |
| GB0700893D0 (en) | 2007-01-17 | 2007-02-21 | King S College London | Male contraceptive |
| US20080242717A1 (en) | 2007-02-28 | 2008-10-02 | Fumiyasu Sato | Methods for treating benign prostatic hyperplasia |
| US20120184591A1 (en) * | 2011-01-13 | 2012-07-19 | Watson Pharmaceuticals, Inc. | Methods for treating prostatitis |
| CN102283816B (zh) | 2011-08-05 | 2013-09-11 | 北京海步国际医药科技发展有限公司 | 西洛多辛缓释片剂及其制备方法 |
| WO2014118606A2 (en) * | 2013-01-29 | 2014-08-07 | Alembic Pharmaceuticals Limited | A novel process for the preparation of silodosin |
| JPWO2016051782A1 (ja) | 2014-09-30 | 2017-07-13 | キッセイ薬品工業株式会社 | 苦味を有する薬剤の苦味をマスキングした経口投与製剤 |
| US20170049834A1 (en) * | 2015-08-18 | 2017-02-23 | Golden Biotechnology Corporation | Benign prostatic hyperplasia add-on therapy |
| PL3750538T3 (pl) * | 2018-03-23 | 2024-11-25 | Pharmajor International | Niehormonalne sposoby męskiej antykoncepcji obejmujące (r) -sylodosynę |
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2020
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2023
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Non-Patent Citations (2)
| Title |
|---|
| Amrican Soc. of Andrology and Eur. Acad. of Andrology, Vol. 5(4), pp 640-663(2017년) |
| Urology, Vol. 80(2), pp 614~617(2012년) |
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