JP6994454B2 - ベンズアゾール化合物ならびに該化合物の作製方法および使用方法 - Google Patents

ベンズアゾール化合物ならびに該化合物の作製方法および使用方法 Download PDF

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JP6994454B2
JP6994454B2 JP2018505606A JP2018505606A JP6994454B2 JP 6994454 B2 JP6994454 B2 JP 6994454B2 JP 2018505606 A JP2018505606 A JP 2018505606A JP 2018505606 A JP2018505606 A JP 2018505606A JP 6994454 B2 JP6994454 B2 JP 6994454B2
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oxazole
carboxamide
thiazole
disease
benzo
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JP2018528181A5 (https=
JP2018528181A (ja
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ローズ イェン
ヤン チェン
ラジンダー シン
ヴァネッサ タイラー
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ライジェル ファーマシューティカルズ， インコーポレイテッド
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    • C—CHEMISTRY; METALLURGY
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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  • General Health & Medical Sciences (AREA)
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  • Diabetes (AREA)
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  • Dermatology (AREA)
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  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
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JP2018505606A 2015-08-04 2016-08-02 ベンズアゾール化合物ならびに該化合物の作製方法および使用方法 Expired - Fee Related JP6994454B2 (ja)

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JP2021201355A JP7339997B2 (ja) 2015-08-04 2021-12-13 ベンズアゾール化合物ならびに該化合物の作製方法および使用方法

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US201562200778P 2015-08-04 2015-08-04
US62/200,778 2015-08-04
PCT/US2016/045176 WO2017023941A1 (en) 2015-08-04 2016-08-02 Benzazole compounds and methods for making and using the compounds

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JP2018528181A JP2018528181A (ja) 2018-09-27
JP2018528181A5 JP2018528181A5 (https=) 2021-08-19
JP6994454B2 true JP6994454B2 (ja) 2022-01-14

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JP2021201355A Active JP7339997B2 (ja) 2015-08-04 2021-12-13 ベンズアゾール化合物ならびに該化合物の作製方法および使用方法

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EP (2) EP3719016A1 (https=)
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EA039043B1 (ru) * 2015-04-22 2021-11-25 Райджел Фармасьютикалз, Инк. Пиразольные соединения и способ получения и применения данных соединений
JP6994454B2 (ja) 2015-08-04 2022-01-14 ライジェル ファーマシューティカルズ， インコーポレイテッド ベンズアゾール化合物ならびに該化合物の作製方法および使用方法
TW202340194A (zh) 2017-02-16 2023-10-16 美商基利科學股份有限公司 吡咯并[1,2-b]嗒𠯤衍生物
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TWI842978B (zh) 2018-07-13 2024-05-21 美商基利科學股份有限公司 衍生物
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