JP6925318B2 - ジシクロプラチンの製造方法 - Google Patents

ジシクロプラチンの製造方法 Download PDF

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Publication number
JP6925318B2
JP6925318B2 JP2018503718A JP2018503718A JP6925318B2 JP 6925318 B2 JP6925318 B2 JP 6925318B2 JP 2018503718 A JP2018503718 A JP 2018503718A JP 2018503718 A JP2018503718 A JP 2018503718A JP 6925318 B2 JP6925318 B2 JP 6925318B2
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carboplatin
dicycloplatin
range
combination step
xrpd
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Japanese (ja)
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JP2018510914A5 (OSRAM
JP2018510914A (ja
Inventor
シャオジョン リウ,
シャオジョン リウ,
ジールイ シー,
ジールイ シー,
イェ チャオ,
イェ チャオ,
リィァン チャン,
リィァン チャン,
Original Assignee
シン−ナット プロダクツ エンタープライズ エルエルシー
シン−ナット プロダクツ エンタープライズ エルエルシー
メドンケアー ファーマスーティカル カンパニー リミテッド
メドンケアー ファーマスーティカル カンパニー リミテッド
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Application filed by シン−ナット プロダクツ エンタープライズ エルエルシー, シン−ナット プロダクツ エンタープライズ エルエルシー, メドンケアー ファーマスーティカル カンパニー リミテッド, メドンケアー ファーマスーティカル カンパニー リミテッド filed Critical シン−ナット プロダクツ エンタープライズ エルエルシー
Publication of JP2018510914A publication Critical patent/JP2018510914A/ja
Publication of JP2018510914A5 publication Critical patent/JP2018510914A5/ja
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0086Platinum compounds
    • C07F15/0093Platinum compounds without a metal-carbon linkage
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/28Compounds containing heavy metals
    • A61K31/282Platinum compounds

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2018503718A 2015-04-10 2015-04-10 ジシクロプラチンの製造方法 Active JP6925318B2 (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2015/025334 WO2016164040A1 (en) 2015-04-10 2015-04-10 Process for the preparation of dicycloplatin

Publications (3)

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JP2018510914A JP2018510914A (ja) 2018-04-19
JP2018510914A5 JP2018510914A5 (OSRAM) 2018-06-07
JP6925318B2 true JP6925318B2 (ja) 2021-08-25

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ID=56895556

Family Applications (1)

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JP2018503718A Active JP6925318B2 (ja) 2015-04-10 2015-04-10 ジシクロプラチンの製造方法

Country Status (14)

Country Link
US (1) US9447130B1 (OSRAM)
EP (1) EP3280408B1 (OSRAM)
JP (1) JP6925318B2 (OSRAM)
KR (1) KR102432526B1 (OSRAM)
CN (1) CN106132408B (OSRAM)
AU (1) AU2015390714B2 (OSRAM)
CA (1) CA2981158C (OSRAM)
DK (1) DK3280408T3 (OSRAM)
ES (1) ES2765648T3 (OSRAM)
IL (1) IL254894B (OSRAM)
MX (1) MX2017012985A (OSRAM)
RU (1) RU2676269C1 (OSRAM)
WO (1) WO2016164040A1 (OSRAM)
ZA (1) ZA201706795B (OSRAM)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016205782A1 (en) 2015-06-19 2016-12-22 Syn-Nat Products Enterprise LLC Composition containing carboplatin and use
WO2016205785A1 (en) 2015-06-19 2016-12-22 Syn-Nat Products Enterprise LLC Pharmaceutical composition of carboplatin based co-crystals and use thereof
AU2016284816B2 (en) 2015-06-25 2021-10-07 Syn-Nat Products Enterprise LLC Pharmaceutical co-crystal composition and use thereof
CN106995467B (zh) * 2017-05-03 2019-06-21 江苏大红鹰恒顺药业有限公司 一种微波催化合成双环铂的方法
CN109053808B (zh) 2017-06-21 2020-12-29 宋勤华 一种高纯度双环铂针状晶体的工业化制备方法
MX2020005310A (es) * 2017-11-21 2020-10-08 Medoncare Pharmaceutical Co Ltd Producto de combinacion que comprende dicicloplatino y metodo de preparacion y uso del mismo.
WO2019153220A1 (zh) * 2018-02-09 2019-08-15 北京索普兴大医药研究有限公司 双环铂药物检测方法
WO2019161526A1 (zh) * 2018-02-22 2019-08-29 昆明贵研药业有限公司 一锅法制备双二羧酸二氨络铂(ii)衍生物的方法
WO2018171371A2 (zh) * 2018-02-22 2018-09-27 昆明贵研药业有限公司 一种双二羧酸二氨络铂(ii)衍生物的制备方法
CN112262123B (zh) * 2018-09-18 2023-12-15 昆明贵研药业有限公司 一种双二羧酸二氨络铂(ii)衍生物的纯化方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2106679C (en) * 1991-03-23 1996-01-09 Dae-Kee Kim Novel platinum (ii) complex and processes for preparing the same
US5455270A (en) * 1993-08-11 1995-10-03 Bristol-Myers Squibb Co. Stabilized solutions of platinum(II) antitumor agents
CN1121380C (zh) * 2000-03-03 2003-09-17 北京兴大豪斯科技有限公司 一种抗肿瘤的双二羧酸二氨络铂衍生物及其药物组合物
EP1473298B1 (en) * 2001-11-30 2009-05-13 Jingzun Wang Supermolecular carboplatinum derivatives, their preparation and pharmaceutical composition containing them as active ingredient and applications of the compositions
JP4992089B2 (ja) * 2005-03-18 2012-08-08 国立大学法人 東京大学 ジアミノシクロヘキサン白金(ii)とブロック共重合体との配位化合物及びそれを含有する抗がん剤
ATE430564T1 (de) * 2005-03-28 2009-05-15 Dabur Pharma Ltd Stabile pharmazeutische zusammensetzungen aus antitumoralen platin-(ii)-mitteln
JP2009525273A (ja) * 2006-01-30 2009-07-09 プラットコー テクノロジーズ (プロプライエタリー) リミテッド 白金(ii)錯体の調製
CA2691047A1 (en) * 2007-06-18 2008-12-24 Platco Technologies (Proprietary) Limited Platinum (iv) complexes

Also Published As

Publication number Publication date
EP3280408A1 (en) 2018-02-14
BR112017021590A2 (pt) 2018-07-03
IL254894A0 (en) 2017-12-31
ZA201706795B (en) 2019-02-27
US9447130B1 (en) 2016-09-20
KR20170134737A (ko) 2017-12-06
CN106132408B (zh) 2018-02-13
CA2981158A1 (en) 2016-10-13
DK3280408T3 (da) 2020-02-03
IL254894B (en) 2021-02-28
JP2018510914A (ja) 2018-04-19
CN106132408A (zh) 2016-11-16
AU2015390714B2 (en) 2021-02-04
AU2015390714A1 (en) 2017-10-26
EP3280408B1 (en) 2019-10-23
CA2981158C (en) 2022-05-24
US20160297842A1 (en) 2016-10-13
KR102432526B1 (ko) 2022-08-12
ES2765648T3 (es) 2020-06-10
RU2676269C1 (ru) 2018-12-27
WO2016164040A1 (en) 2016-10-13
MX2017012985A (es) 2018-05-22
EP3280408A4 (en) 2018-10-17

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