JP6789941B2 - Ｔｇｆ−ベータ阻害剤としての縮合イミダゾール誘導体 - Google Patents

Ｔｇｆ−ベータ阻害剤としての縮合イミダゾール誘導体 Download PDF

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JP6789941B2
JP6789941B2 JP2017527370A JP2017527370A JP6789941B2 JP 6789941 B2 JP6789941 B2 JP 6789941B2 JP 2017527370 A JP2017527370 A JP 2017527370A JP 2017527370 A JP2017527370 A JP 2017527370A JP 6789941 B2 JP6789941 B2 JP 6789941B2
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dihydro
pyrrolo
imidazol
imidazole
pyridine
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JP2018501209A5 (cg-RX-API-DMAC7.html
JP2018501209A (ja
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ラジンダー・シン
トッド・キンセラ
ジアシン・ユー
マリーナ・ジェルマン
イハブ・エス・ダーウィッシュ
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ライジェル ファーマシューティカルズ， インコーポレイテッド
ライジェル ファーマシューティカルズ， インコーポレイテッド
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    • C07—ORGANIC CHEMISTRY
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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JP2017527370A 2014-11-21 2015-11-16 Ｔｇｆ−ベータ阻害剤としての縮合イミダゾール誘導体 Expired - Fee Related JP6789941B2 (ja)

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US201462082959P 2014-11-21 2014-11-21
US62/082,959 2014-11-21
US201562141509P 2015-04-01 2015-04-01
US62/141,509 2015-04-01
PCT/US2015/060872 WO2016081364A1 (en) 2014-11-21 2015-11-16 Fused imidazole derivatives as tgf-beta inhibitors

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JP2018501209A JP2018501209A (ja) 2018-01-18
JP2018501209A5 JP2018501209A5 (cg-RX-API-DMAC7.html) 2018-12-27
JP6789941B2 true JP6789941B2 (ja) 2020-11-25

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