JP6294314B2 - ホスフィン配位パラジウムスルホナートパラダサイクル - Google Patents

ホスフィン配位パラジウムスルホナートパラダサイクル Download PDF

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JP6294314B2
JP6294314B2 JP2015516006A JP2015516006A JP6294314B2 JP 6294314 B2 JP6294314 B2 JP 6294314B2 JP 2015516006 A JP2015516006 A JP 2015516006A JP 2015516006 A JP2015516006 A JP 2015516006A JP 6294314 B2 JP6294314 B2 JP 6294314B2
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aryl
certain embodiments
precatalyst
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JP2015527300A (ja
JP2015527300A5 (enExample
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シー ブルーノ，ニコラス
シー ブルーノ，ニコラス
エル バックウォルド，スティーヴン
エル バックウォルド，スティーヴン
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Massachusetts Institute of Technology
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/006—Palladium compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B37/00—Reactions without formation or introduction of functional groups containing hetero atoms, involving either the formation of a carbon-to-carbon bond between two carbon atoms not directly linked already or the disconnection of two directly linked carbon atoms
    • C07B37/04—Substitution
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0086—Platinum compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
JP2015516006A 2012-06-08 2013-03-13 ホスフィン配位パラジウムスルホナートパラダサイクル Active JP6294314B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261657377P 2012-06-08 2012-06-08
US61/657,377 2012-06-08
PCT/US2013/030779 WO2013184198A1 (en) 2012-06-08 2013-03-13 Phosphine-ligated palladium sulfonate palladacycles

Related Child Applications (1)

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JP2017236262A Division JP2018061956A (ja) 2012-06-08 2017-12-08 ホスフィン配位パラジウムスルホナートパラダサイクル

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JP2015527300A JP2015527300A (ja) 2015-09-17
JP2015527300A5 JP2015527300A5 (enExample) 2016-05-12
JP6294314B2 true JP6294314B2 (ja) 2018-03-14

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JP2015516006A Active JP6294314B2 (ja) 2012-06-08 2013-03-13 ホスフィン配位パラジウムスルホナートパラダサイクル
JP2017236262A Withdrawn JP2018061956A (ja) 2012-06-08 2017-12-08 ホスフィン配位パラジウムスルホナートパラダサイクル

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US (2) US8889857B2 (enExample)
EP (1) EP2859005B1 (enExample)
JP (2) JP6294314B2 (enExample)
WO (1) WO2013184198A1 (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8563573B2 (en) 2007-11-02 2013-10-22 Vertex Pharmaceuticals Incorporated Azaindole derivatives as CFTR modulators
US8802868B2 (en) 2010-03-25 2014-08-12 Vertex Pharmaceuticals Incorporated Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxo1-5-yl)-N-(1-(2,3-dihydroxypropyl-6-fluoro-2-(1-hydroxy-2-methylpropan2-yl)-1H-Indol-5-yl)-Cyclopropanecarboxamide
KR20190061096A (ko) 2010-04-22 2019-06-04 버텍스 파마슈티칼스 인코포레이티드 시클로알킬카르복스아미도-인돌 화합물의 제조 방법
PL3925607T3 (pl) 2014-04-15 2023-10-30 Vertex Pharmaceuticals Incorporated Kompozycje farmaceutyczne do leczenia chorób, w których pośredniczy mukowiscydozowy przezbłonowy regulator przewodnictwa
WO2017094655A1 (ja) * 2015-12-02 2017-06-08 住友化学株式会社 芳香族化合物の製造方法およびパラジウム錯体
CN105618144B (zh) * 2016-03-10 2018-01-05 南京理工大学 一种用于吲哚二位芳基化的氟功能化介孔硅胶负载钯催化剂及其制备方法和应用
GB201604970D0 (en) 2016-03-23 2016-05-04 Syngenta Participations Ag Improvements in or relating to organic compounds
EP3454981B1 (en) 2016-05-10 2021-03-03 Promega Corporation Palladium catalysts with improved performance in biological environments
CN107537575B (zh) * 2016-06-24 2020-05-05 中国科学院大连化学物理研究所 一种咪唑盐有机聚合物催化剂及其制备方法和应用
CN107537562B (zh) * 2016-06-24 2020-06-19 中国科学院大连化学物理研究所 含膦-离子液体有机共聚物多相催化剂及其制备和应用
WO2018106338A1 (en) 2016-12-06 2018-06-14 Dow Global Technologies Llc Mono-ligated palladium catalysts, their synthesis and use in suzuki coupling
WO2018106337A1 (en) 2016-12-06 2018-06-14 Dow Global Technologies Llc Mono-ligated palladium catalyts, their synthesis and use in suzuki coupling
WO2018106336A1 (en) 2016-12-06 2018-06-14 Dow Global Technologies Llc Mono-ligated palladium catalyts, their synthesis and use in suzuki coupling
WO2020094440A1 (en) 2018-11-07 2020-05-14 Basf Se Process for the synthesis of aryl hydrazines
US11377420B2 (en) 2019-06-24 2022-07-05 Board Of Regents, The University Of Texas System Compositions and methods for making donor-acceptor azetines
EP4313997A1 (en) * 2021-03-25 2024-02-07 Sigma-Aldrich Co. LLC Novel ferrocene-based unsymmetrical ligands bearing bulky di(adamantly)phosphino motif and their metal catalysts
CN113019463B (zh) * 2021-05-25 2021-09-07 江苏欣诺科催化剂有限公司 钯复合催化剂及其制备方法和应用
CN114632552B (zh) * 2022-05-19 2022-08-02 苏州欣诺科生物科技有限公司 Buchwald预催化剂及其制备方法与应用
CN116813890A (zh) * 2023-06-02 2023-09-29 中国科学院大学 一种Suzuki-Miyaura催化聚合体系用于合成共轭聚合物的方法和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006010885A1 (en) * 2004-07-30 2006-02-02 Heriot-Watt University Palladacyles, their preparation and catalytic processes involving their use as catalyst, especially catalytic carbonylation processes
CA2708369C (en) * 2007-12-12 2017-04-04 Massachusetts Institute Of Technology Ligands for transition-metal-catalyzed cross-couplings, and methods of use thereof
WO2011008725A2 (en) 2009-07-13 2011-01-20 Massachusetts Institute Of Technology Metal-catalyzed carbon-fluorine bond formation

Also Published As

Publication number Publication date
EP2859005B1 (en) 2018-10-31
WO2013184198A1 (en) 2013-12-12
US8889857B2 (en) 2014-11-18
EP2859005A4 (en) 2016-02-17
JP2015527300A (ja) 2015-09-17
JP2018061956A (ja) 2018-04-19
EP2859005A1 (en) 2015-04-15
US8981086B2 (en) 2015-03-17
US20130331566A1 (en) 2013-12-12
US20150045570A1 (en) 2015-02-12

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