JP6020396B2 - アゾール誘導体を含有する医薬 - Google Patents
アゾール誘導体を含有する医薬 Download PDFInfo
- Publication number
- JP6020396B2 JP6020396B2 JP2013186829A JP2013186829A JP6020396B2 JP 6020396 B2 JP6020396 B2 JP 6020396B2 JP 2013186829 A JP2013186829 A JP 2013186829A JP 2013186829 A JP2013186829 A JP 2013186829A JP 6020396 B2 JP6020396 B2 JP 6020396B2
- Authority
- JP
- Japan
- Prior art keywords
- compound
- group
- methyl
- pyrrolidin
- difluoro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- XOZZPNYSQIRLEN-SFHVURJKSA-N CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1n[nH]c(COc(cc2OC)ccc2OC)n1)=O)(F)F)O Chemical compound CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1n[nH]c(COc(cc2OC)ccc2OC)n1)=O)(F)F)O XOZZPNYSQIRLEN-SFHVURJKSA-N 0.000 description 2
- AZEIEPKQCNOBBU-INIZCTEOSA-N CC(C)(C)OC(N(CCC1)[C@@H]1c1ncc(COc(cc2)cc(OC)c2OC)[s]1)=O Chemical compound CC(C)(C)OC(N(CCC1)[C@@H]1c1ncc(COc(cc2)cc(OC)c2OC)[s]1)=O AZEIEPKQCNOBBU-INIZCTEOSA-N 0.000 description 1
- BZTKSOGBWKDMTB-QHCPKHFHSA-N CC(C)(C)OC(N(CCC1)[C@@H]1c1nnc(CO[Si](C(C)(C)C)(c2ccccc2)c2ccccc2)[o]1)=O Chemical compound CC(C)(C)OC(N(CCC1)[C@@H]1c1nnc(CO[Si](C(C)(C)C)(c2ccccc2)c2ccccc2)[o]1)=O BZTKSOGBWKDMTB-QHCPKHFHSA-N 0.000 description 1
- BSVVLQXRQIHTSE-UHFFFAOYSA-N CC(C)(CC(C)(C)C1)CC1(C(C(C)=O)(F)F)O Chemical compound CC(C)(CC(C)(C)C1)CC1(C(C(C)=O)(F)F)O BSVVLQXRQIHTSE-UHFFFAOYSA-N 0.000 description 1
- CSZFOLMDHFDLLR-FQEVSTJZSA-N CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1n[o]c(COc2cnccc2)c1)=O)(F)F)O Chemical compound CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1n[o]c(COc2cnccc2)c1)=O)(F)F)O CSZFOLMDHFDLLR-FQEVSTJZSA-N 0.000 description 1
- IZQLJVNWGSKPHE-FQEVSTJZSA-N CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1ncc(COc(cc2OC)ccc2OC)[o]1)=O)(F)F)O Chemical compound CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1ncc(COc(cc2OC)ccc2OC)[o]1)=O)(F)F)O IZQLJVNWGSKPHE-FQEVSTJZSA-N 0.000 description 1
- UPOILGSZTBWGJW-FQEVSTJZSA-N CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1ncc(COc(cc2OC)ccc2OC)[s]1)=O)(F)F)O Chemical compound CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1ncc(COc(cc2OC)ccc2OC)[s]1)=O)(F)F)O UPOILGSZTBWGJW-FQEVSTJZSA-N 0.000 description 1
- BLKNOVDRFRHCTP-SFHVURJKSA-N CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1nnc(COc(cc2OC)ccc2OC)[s]1)=O)(F)F)O Chemical compound CC(C)(CC(C)(C)C1)CC1(C(C(N(CCC1)[C@@H]1c1nnc(COc(cc2OC)ccc2OC)[s]1)=O)(F)F)O BLKNOVDRFRHCTP-SFHVURJKSA-N 0.000 description 1
- WMVUDDPTEHKZKF-ZDUSSCGKSA-N COc(c(OC)c1)ccc1OCc1cnc([C@H]2NCCC2)[o]1 Chemical compound COc(c(OC)c1)ccc1OCc1cnc([C@H]2NCCC2)[o]1 WMVUDDPTEHKZKF-ZDUSSCGKSA-N 0.000 description 1
- PANWHYHNSGYWAG-UHFFFAOYSA-N CS(CC1CCCCC1)(=O)=O Chemical compound CS(CC1CCCCC1)(=O)=O PANWHYHNSGYWAG-UHFFFAOYSA-N 0.000 description 1
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2013186829A JP6020396B2 (ja) | 2012-09-12 | 2013-09-10 | アゾール誘導体を含有する医薬 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2012200100 | 2012-09-12 | ||
| JP2012200100 | 2012-09-12 | ||
| JP2013186829A JP6020396B2 (ja) | 2012-09-12 | 2013-09-10 | アゾール誘導体を含有する医薬 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2014074018A JP2014074018A (ja) | 2014-04-24 |
| JP2014074018A5 JP2014074018A5 (enExample) | 2014-12-25 |
| JP6020396B2 true JP6020396B2 (ja) | 2016-11-02 |
Family
ID=50748467
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013186829A Expired - Fee Related JP6020396B2 (ja) | 2012-09-12 | 2013-09-10 | アゾール誘導体を含有する医薬 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JP6020396B2 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2976327A1 (en) * | 2015-02-25 | 2016-09-01 | Taisho Pharmaceutical Co., Ltd. | Hair growth composition for cutaneous application |
| CN113248501B (zh) * | 2021-06-17 | 2021-10-08 | 南京韦尔优众医药有限公司 | Cly系列化合物及其制备方法和制备药物的用途 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5945441A (en) * | 1997-06-04 | 1999-08-31 | Gpi Nil Holdings, Inc. | Pyrrolidine carboxylate hair revitalizing agents |
| GB9804426D0 (en) * | 1998-03-02 | 1998-04-29 | Pfizer Ltd | Heterocycles |
| JP4240978B2 (ja) * | 2002-09-30 | 2009-03-18 | 大正製薬株式会社 | アリールオキシメチルオキサジアゾール誘導体 |
| JPWO2008075735A1 (ja) * | 2006-12-20 | 2010-04-15 | 大正製薬株式会社 | 脱毛症の予防又は治療剤 |
| TWI534142B (zh) * | 2011-03-15 | 2016-05-21 | 大正製藥股份有限公司 | Azole derivatives |
-
2013
- 2013-09-10 JP JP2013186829A patent/JP6020396B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP2014074018A (ja) | 2014-04-24 |
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