JP5628796B2 - 性的不能の治療用のメラノコルチンレセプタ特異的ペプチド - Google Patents

性的不能の治療用のメラノコルチンレセプタ特異的ペプチド Download PDF

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JP5628796B2
JP5628796B2 JP2011512730A JP2011512730A JP5628796B2 JP 5628796 B2 JP5628796 B2 JP 5628796B2 JP 2011512730 A JP2011512730 A JP 2011512730A JP 2011512730 A JP2011512730 A JP 2011512730A JP 5628796 B2 JP5628796 B2 JP 5628796B2
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peptide
peptides
cyclic
cyclic peptide
acid
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JP2011522839A5 (https=
JP2011522839A (ja
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シー，イ−クン
シャルマ，シュッブ，ディー．
ヤン，ウェイ
チェン，シン
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Palatin Technologies Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/68—Melanocyte-stimulating hormone [MSH]
    • C07K14/685—Alpha-melanotropin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13—Cyclosporins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/02—Peptides of undefined number of amino acids; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Reproductive Health (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
JP2011512730A 2008-06-09 2009-06-08 性的不能の治療用のメラノコルチンレセプタ特異的ペプチド Expired - Fee Related JP5628796B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5991008P 2008-06-09 2008-06-09
US61/059,910 2008-06-09
PCT/US2009/046571 WO2009152079A1 (en) 2008-06-09 2009-06-08 Melanocortin receptor-specific peptides for treatment of sexual dysfunction

Publications (3)

Publication Number Publication Date
JP2011522839A JP2011522839A (ja) 2011-08-04
JP2011522839A5 JP2011522839A5 (https=) 2012-06-07
JP5628796B2 true JP5628796B2 (ja) 2014-11-19

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JP2011512730A Expired - Fee Related JP5628796B2 (ja) 2008-06-09 2009-06-08 性的不能の治療用のメラノコルチンレセプタ特異的ペプチド

Country Status (14)

Country Link
US (2) US8487073B2 (https=)
EP (1) EP2300036B1 (https=)
JP (1) JP5628796B2 (https=)
KR (1) KR101687037B1 (https=)
CN (1) CN102131514B (https=)
AU (1) AU2009257631B2 (https=)
BR (1) BRPI0909947A2 (https=)
CA (1) CA2727317C (https=)
EA (1) EA018630B1 (https=)
IL (1) IL209867A (https=)
MX (1) MX2010013436A (https=)
NZ (1) NZ590254A (https=)
WO (1) WO2009152079A1 (https=)
ZA (1) ZA201009165B (https=)

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Publication number Publication date
MX2010013436A (es) 2011-06-21
US20110065652A1 (en) 2011-03-17
IL209867A0 (en) 2011-02-28
CA2727317C (en) 2015-02-17
IL209867A (en) 2015-08-31
NZ590254A (en) 2012-07-27
KR101687037B1 (ko) 2016-12-15
EP2300036B1 (en) 2017-04-05
ZA201009165B (en) 2012-03-28
CN102131514B (zh) 2014-08-20
BRPI0909947A2 (pt) 2017-06-27
US8729224B2 (en) 2014-05-20
EA201001722A1 (ru) 2011-08-30
US8487073B2 (en) 2013-07-16
CA2727317A1 (en) 2009-12-17
WO2009152079A1 (en) 2009-12-17
EA018630B1 (ru) 2013-09-30
US20130288987A1 (en) 2013-10-31
CN102131514A (zh) 2011-07-20
EP2300036A1 (en) 2011-03-30
EP2300036A4 (en) 2012-01-18
KR20110040819A (ko) 2011-04-20
AU2009257631A1 (en) 2009-12-17
AU2009257631B2 (en) 2014-07-24
JP2011522839A (ja) 2011-08-04

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