JP5608653B2 - チュアブルな徐放性製剤 - Google Patents

チュアブルな徐放性製剤 Download PDF

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Publication number
JP5608653B2
JP5608653B2 JP2011526247A JP2011526247A JP5608653B2 JP 5608653 B2 JP5608653 B2 JP 5608653B2 JP 2011526247 A JP2011526247 A JP 2011526247A JP 2011526247 A JP2011526247 A JP 2011526247A JP 5608653 B2 JP5608653 B2 JP 5608653B2
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Japan
Prior art keywords
active ingredient
formulation
sustained release
certain embodiments
zein
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JP2011526247A
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English (en)
Japanese (ja)
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JP2012502061A5 (enExample
JP2012502061A (ja
Inventor
アンドリュー シャン チェン
パトリシア ディー. キギン
ハイ リャン チェン
ジュン ファン
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ファーナム・カンパニーズ・インコーポレーテッド
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1658—Proteins, e.g. albumin, gelatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1664—Compounds of unknown constitution, e.g. material from plants or animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2063—Proteins, e.g. gelatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2068—Compounds of unknown constitution, e.g. material from plants or animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Botany (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2011526247A 2008-09-04 2009-09-04 チュアブルな徐放性製剤 Expired - Fee Related JP5608653B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9436308P 2008-09-04 2008-09-04
US61/094,363 2008-09-04
PCT/US2009/056103 WO2010028290A1 (en) 2008-09-04 2009-09-04 Chewable sustained release formulations

Publications (3)

Publication Number Publication Date
JP2012502061A JP2012502061A (ja) 2012-01-26
JP2012502061A5 JP2012502061A5 (enExample) 2012-09-20
JP5608653B2 true JP5608653B2 (ja) 2014-10-15

Family

ID=41219093

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011526247A Expired - Fee Related JP5608653B2 (ja) 2008-09-04 2009-09-04 チュアブルな徐放性製剤

Country Status (8)

Country Link
US (1) US10668012B2 (enExample)
EP (1) EP2331076B1 (enExample)
JP (1) JP5608653B2 (enExample)
CN (1) CN102202654B (enExample)
AU (1) AU2009289464B2 (enExample)
CA (1) CA2736119C (enExample)
ES (1) ES2536736T3 (enExample)
WO (1) WO2010028290A1 (enExample)

Families Citing this family (16)

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IT1400578B1 (it) * 2010-06-18 2013-06-14 Alpex Pharma Sa Processo per la preparazione di compresse a rilascio controllato.
CA2854054C (en) * 2011-12-02 2020-05-12 Pegasus Laboratories, Inc. Amphipathic lipid-based sustained release compositions
US10722458B2 (en) * 2011-12-02 2020-07-28 Pegasus Laboratories, Inc. Amphipathic lipid-based sustained release compositions
CN104427977B (zh) 2012-05-10 2018-02-02 佩因拉佛姆有限公司 局部麻醉剂的储库制剂及其制备方法
CN103686676A (zh) * 2012-08-31 2014-03-26 中兴通讯股份有限公司 设备到设备通信系统的通信方法、装置及系统
US20140080908A1 (en) * 2012-09-19 2014-03-20 Phyto Tech Corp. Compositions and methods for improving or preventing depression-like symptoms
CN111803465B (zh) 2013-03-15 2023-05-09 阿根塔创新有限公司 可咀嚼配制物
MX392606B (es) 2016-03-17 2025-03-24 Thiogenesis Therapeutics Inc Composiciones para la liberacion controlada de cisteamina y el tratamiento sistemico de trastornos sensibles a la cisteamina.
JP6800596B2 (ja) * 2016-03-29 2020-12-16 小林製薬株式会社 錠剤
EP3519812B1 (en) 2016-09-27 2026-05-06 Zolentroff, William C. Ala and salt formulation
CN110996920A (zh) * 2017-07-26 2020-04-10 太杰先软嚼有限责任公司 用于兽医应用的无淀粉软咀嚼物
CN109420163B (zh) * 2017-08-23 2022-06-21 中山市力恩普制药有限公司 治疗呼吸道感染的药物组合物及其制备方法和用途
WO2019060634A1 (en) 2017-09-20 2019-03-28 Thiogenesis Therapeutics, Inc. METHODS OF TREATING CYSTEAMINE SENSITIVE DISORDERS
CN113260351A (zh) * 2018-12-29 2021-08-13 3M创新有限公司 口腔制品及使用方法
US12390488B2 (en) * 2018-12-29 2025-08-19 Solventum Intellectual Properties Company Oral articles and methods of use
CN111744018A (zh) * 2019-03-26 2020-10-09 北京福元医药股份有限公司 一种盐酸氨基葡萄糖药物制剂

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US5032406A (en) * 1989-02-21 1991-07-16 Norwich Eaton Pharmaceuticals, Inc. Dual-action tablet
GB8913889D0 (en) 1989-06-16 1989-08-02 May & Baker Ltd New compositions of matter
US5182130A (en) * 1989-11-06 1993-01-26 Opta Food Ingredients, Inc. Method for producing an edible prolamine coating from an aqueous latex
US5077053A (en) * 1990-02-12 1991-12-31 Warner-Lambert Company Zein as a moisture barrier for sugarless edible compositions and method for preparing same
US5599556A (en) * 1991-12-31 1997-02-04 Abbott Laboratories Prolamine coatings for taste masking
US6210714B1 (en) * 1993-11-23 2001-04-03 Euro-Celtique S.A. Immediate release tablet cores of acetaminophen having sustained-release coating
US5965161A (en) * 1994-11-04 1999-10-12 Euro-Celtique, S.A. Extruded multi-particulates
DE19630035A1 (de) 1996-07-25 1998-01-29 Asta Medica Ag Tramadol Multiple Unit Formulierungen
JP3877083B2 (ja) * 1996-08-03 2007-02-07 昭和産業株式会社 第4胃以降消化・吸収性反芻動物用飼料製剤並びにそれを含有する反芻動物用飼料
FR2752732B1 (fr) 1996-08-28 1998-11-20 Pf Medicament Forme galenique a liberation prolongee de milnacipran
US5904937A (en) * 1997-10-03 1999-05-18 Fmc Corporation Taste masked pharmaceutical compositions
WO1999048372A1 (en) * 1998-03-23 1999-09-30 General Mills, Inc. Encapsulation of components into edible products
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PL2486942T3 (pl) * 2004-11-24 2019-05-31 Meda Pharmaceuticals Inc Kompozycje zawierające azelastynę oraz sposoby ich stosowania
WO2006082824A1 (ja) * 2005-02-03 2006-08-10 Nrl Pharma, Inc. マトリックス型腸溶性・徐放性組成物
JP4602949B2 (ja) * 2006-08-02 2010-12-22 和光堂株式会社 被覆粒子含有組成物及びその製造方法

Also Published As

Publication number Publication date
ES2536736T3 (es) 2015-05-28
EP2331076B1 (en) 2015-03-04
CN102202654B (zh) 2014-07-30
CA2736119C (en) 2016-08-23
AU2009289464A1 (en) 2010-03-11
US20100062988A1 (en) 2010-03-11
EP2331076A1 (en) 2011-06-15
AU2009289464B2 (en) 2015-12-10
CN102202654A (zh) 2011-09-28
JP2012502061A (ja) 2012-01-26
WO2010028290A1 (en) 2010-03-11
CA2736119A1 (en) 2010-03-11
US10668012B2 (en) 2020-06-02

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