JP5536752B2 - プロスタサイクリン(pgi2)受容体に関連する障害の処置に有用なpgi2受容体の調節因子 - Google Patents
プロスタサイクリン(pgi2)受容体に関連する障害の処置に有用なpgi2受容体の調節因子 Download PDFInfo
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- JP5536752B2 JP5536752B2 JP2011500799A JP2011500799A JP5536752B2 JP 5536752 B2 JP5536752 B2 JP 5536752B2 JP 2011500799 A JP2011500799 A JP 2011500799A JP 2011500799 A JP2011500799 A JP 2011500799A JP 5536752 B2 JP5536752 B2 JP 5536752B2
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- fluorophenyl
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- phenyl
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| KR20220031743A (ko) * | 2008-03-18 | 2022-03-11 | 아레나 파마슈티칼스, 인크. | 프로스타시클린 (pgi2) 수용체와 관련된 장애의 치료에 유용한 상기 수용체의 조절제 |
| BRPI0921369B8 (pt) | 2008-11-26 | 2021-05-25 | Arena Pharm Inc | composto modulador do receptor de prostaciclina (pgi2), sua composição, sua composição farmacêutica, seus usos, bem como processos para a preparação das referidas composições |
| ES2548882T3 (es) | 2008-12-08 | 2015-10-21 | Arena Pharmaceuticals, Inc. | Moduladores del receptor de prostaciclina (PGl2) útiles para el tratamiento de trastornos relacionados con los mismos |
| EP2480526A1 (en) * | 2009-09-23 | 2012-08-01 | Arena Pharmaceuticals, Inc. | Crystalline forms and processes for the preparation of pgi2 receptor agonists |
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| CN106535884A (zh) | 2014-06-06 | 2017-03-22 | 弗雷克萨斯生物科学公司 | 免疫调节剂 |
| US9593061B2 (en) | 2014-10-20 | 2017-03-14 | United Therapeutics Corporation | Synthesis of intermediates for producing prostacyclin derivatives |
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| UY36391A (es) | 2014-11-05 | 2016-06-01 | Flexus Biosciences Inc | Compuestos moduladores de la enzima indolamina 2,3-dioxigenasa (ido1), sus métodos de síntesis y composiciones farmacèuticas que las contienen |
| BR112017008809A2 (pt) | 2014-11-05 | 2017-12-19 | Flexus Biosciences Inc | agentes imunorreguladores |
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| RU2632449C1 (ru) * | 2016-04-26 | 2017-10-04 | Государственное бюджетное образовательное учреждение высшего профессионального образования "Уральский государственный медицинский университет Министерства здравоохранения Российской Федерации" (ГБОУ ВПО УГМУ Минздрава России) | Способ оптимизации лечения мужчин кардиотропной терапией и заместительной гормональной терапией при андрогенодефиците с артериальной гипертензией |
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