JP5448844B2 - ネビボロールを含む固体の医薬組成物 - Google Patents
ネビボロールを含む固体の医薬組成物 Download PDFInfo
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- JP5448844B2 JP5448844B2 JP2009546620A JP2009546620A JP5448844B2 JP 5448844 B2 JP5448844 B2 JP 5448844B2 JP 2009546620 A JP2009546620 A JP 2009546620A JP 2009546620 A JP2009546620 A JP 2009546620A JP 5448844 B2 JP5448844 B2 JP 5448844B2
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- nebivolol
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- active ingredient
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- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Molecular Biology (AREA)
- Inorganic Chemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biochemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Biophysics (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CA2575527 | 2007-01-22 | ||
| CA2,575,527 | 2007-01-22 | ||
| PCT/CA2008/000119 WO2008089549A1 (en) | 2007-01-22 | 2008-01-22 | Pharmaceutical compositions comprising nebivolol or a nebivolol analogue |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010516712A JP2010516712A (ja) | 2010-05-20 |
| JP2010516712A5 JP2010516712A5 (enExample) | 2010-12-16 |
| JP5448844B2 true JP5448844B2 (ja) | 2014-03-19 |
Family
ID=39644046
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009546620A Expired - Fee Related JP5448844B2 (ja) | 2007-01-22 | 2008-01-22 | ネビボロールを含む固体の医薬組成物 |
Country Status (6)
| Country | Link |
|---|---|
| US (2) | US20100137424A1 (enExample) |
| EP (1) | EP2124931A4 (enExample) |
| JP (1) | JP5448844B2 (enExample) |
| AU (1) | AU2008209264B2 (enExample) |
| CA (1) | CA2675538C (enExample) |
| WO (1) | WO2008089549A1 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2019183470A2 (en) | 2018-03-22 | 2019-09-26 | Incarda Therapeutics, Inc. | A novel method to slow ventricular rate |
| US20220016025A1 (en) * | 2020-07-08 | 2022-01-20 | Vinayak Dinesh DENDUKURI | Formulations of nebivolol |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1337429C (en) | 1983-12-05 | 1995-10-24 | Guy Rosalia Eugene Van Lommen | Derivatives of 2,2'-iminobisethanol |
| CA1337432C (en) | 1988-03-23 | 1995-10-24 | Raymond M. Xhonneux | Method of lowering the blood pressure |
| US5338732A (en) * | 1991-06-18 | 1994-08-16 | Bristol-Myers Squibb Company | Megestrol acetate formulation |
| TW355683B (en) * | 1994-02-17 | 1999-04-11 | Janssen Pharmaceutica Nv | Composition containing micronized nebivolol |
| JPH098913A (ja) | 1995-06-22 | 1997-01-10 | Hitachi Maxell Ltd | 情報通信システム |
| UA74141C2 (uk) * | 1998-12-09 | 2005-11-15 | Дж.Д. Сірл Енд Ко. | Фармацевтична композиція на основі тонкоподрібненого еплеренону (варіанти), спосіб її одержання та спосіб лікування розладів, опосередкованих альдостероном (варіанти) |
| FR2809731B1 (fr) * | 2000-05-31 | 2002-07-19 | Sanofi Synthelabo | Derives de 1,4-diazabicyclo-[3.2.2] nonane-pheylisoxazole, leur preparation et leur application en therapeutique |
| WO2005099699A1 (en) | 2004-04-07 | 2005-10-27 | Sepracor Inc. | Combination of (s)-amlodipine and a beta-blocker, and methods for reducing hypertension |
| WO2005117899A1 (en) * | 2004-06-02 | 2005-12-15 | Cipla Limited | Pharmaceutical composition comprising tibolone and process for procuding the same |
| EP1737847B1 (en) * | 2004-07-30 | 2008-06-04 | Torrent Pharmaceuticals Ltd | Nebivolol and its pharmaceutically acceptable salts, process for preparation and pharmaceutical compositions of nebivolol |
| EP1850842A1 (de) | 2005-02-11 | 2007-11-07 | Stada Arzneimittel Ag | Pharmazeutische zusammensetzungen nebivolo und ein hydrophiles polymer |
| CA2610694A1 (en) * | 2005-05-31 | 2006-12-07 | Mylan Laboratories, Inc. | Compositions comrising nebivolol |
| EP1839658A1 (en) * | 2006-03-30 | 2007-10-03 | Hexal A/S | Pharmaceutical composition comprising micronized nebivolol |
-
2008
- 2008-01-22 US US12/523,686 patent/US20100137424A1/en not_active Abandoned
- 2008-01-22 AU AU2008209264A patent/AU2008209264B2/en not_active Ceased
- 2008-01-22 EP EP08706266.7A patent/EP2124931A4/en not_active Withdrawn
- 2008-01-22 CA CA2675538A patent/CA2675538C/en active Active
- 2008-01-22 WO PCT/CA2008/000119 patent/WO2008089549A1/en not_active Ceased
- 2008-01-22 JP JP2009546620A patent/JP5448844B2/ja not_active Expired - Fee Related
-
2015
- 2015-05-05 US US14/704,375 patent/US10117939B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| AU2008209264B2 (en) | 2014-11-27 |
| EP2124931A4 (en) | 2013-08-28 |
| JP2010516712A (ja) | 2010-05-20 |
| WO2008089549A1 (en) | 2008-07-31 |
| CA2675538A1 (en) | 2008-07-31 |
| EP2124931A1 (en) | 2009-12-02 |
| US10117939B2 (en) | 2018-11-06 |
| CA2675538C (en) | 2017-02-28 |
| AU2008209264A1 (en) | 2008-07-31 |
| US20100137424A1 (en) | 2010-06-03 |
| US20150231261A1 (en) | 2015-08-20 |
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