JP5328349B2 - ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤 - Google Patents

ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤 Download PDF

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JP5328349B2
JP5328349B2 JP2008522861A JP2008522861A JP5328349B2 JP 5328349 B2 JP5328349 B2 JP 5328349B2 JP 2008522861 A JP2008522861 A JP 2008522861A JP 2008522861 A JP2008522861 A JP 2008522861A JP 5328349 B2 JP5328349 B2 JP 5328349B2
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JP2009502788A5 (cg-RX-API-DMAC10.html
JP2009502788A (ja
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コッペル，ゲリー，エー．
ミラー，マーヴィン，ジェイ．
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Azevan Pharmaceuticals Inc
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Azevan Pharmaceuticals Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Otolaryngology (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Addiction (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Anesthesiology (AREA)
JP2008522861A 2005-07-19 2006-07-18 ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤 Expired - Fee Related JP5328349B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US70067305P 2005-07-19 2005-07-19
US60/700,673 2005-07-19
PCT/US2006/027703 WO2007011878A2 (en) 2005-07-19 2006-07-18 Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists

Related Child Applications (1)

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JP2013044654A Division JP2013151520A (ja) 2005-07-19 2013-03-06 ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤

Publications (3)

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JP2009502788A JP2009502788A (ja) 2009-01-29
JP2009502788A5 JP2009502788A5 (cg-RX-API-DMAC10.html) 2009-10-08
JP5328349B2 true JP5328349B2 (ja) 2013-10-30

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JP2008522861A Expired - Fee Related JP5328349B2 (ja) 2005-07-19 2006-07-18 ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤
JP2013044654A Pending JP2013151520A (ja) 2005-07-19 2013-03-06 ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤

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US (2) US8048874B2 (cg-RX-API-DMAC10.html)
EP (1) EP1910346B1 (cg-RX-API-DMAC10.html)
JP (2) JP5328349B2 (cg-RX-API-DMAC10.html)
KR (2) KR101521405B1 (cg-RX-API-DMAC10.html)
CN (1) CN101268068B (cg-RX-API-DMAC10.html)
AU (1) AU2006270039B2 (cg-RX-API-DMAC10.html)
BR (1) BRPI0613664B1 (cg-RX-API-DMAC10.html)
CA (1) CA2615813C (cg-RX-API-DMAC10.html)
DK (1) DK1910346T3 (cg-RX-API-DMAC10.html)
ES (1) ES2726942T3 (cg-RX-API-DMAC10.html)
PL (1) PL1910346T3 (cg-RX-API-DMAC10.html)
RU (1) RU2466991C2 (cg-RX-API-DMAC10.html)
SI (1) SI1910346T1 (cg-RX-API-DMAC10.html)
TR (1) TR201907381T4 (cg-RX-API-DMAC10.html)
WO (1) WO2007011878A2 (cg-RX-API-DMAC10.html)

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AU2002342045C1 (en) * 2001-10-12 2009-07-30 Azevan Pharmaceuticals, Inc. Beta-lactamyl vasopressin Vla antagonists
US7601695B2 (en) 2003-03-10 2009-10-13 Optimer Pharmaceuticals, Inc. Antibacterial agents
CN104922117A (zh) 2005-03-22 2015-09-23 阿泽范药品公司 用于治疗月经前病症的β-内酰氨基链烷酸
CA2615813C (en) * 2005-07-19 2015-12-15 Azevan Pharmaceuticals, Inc. Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists
WO2008034032A2 (en) * 2006-09-14 2008-03-20 Azevan Pharmaceuticals, Inc. Beta-lactam cannabinoid receptor modulators
AU2008316830B2 (en) 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
CN107854477A (zh) 2008-10-24 2018-03-30 森普拉制药公司 使用含三唑的大环内酯治疗抗性疾病的方法
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
AU2011272738B2 (en) 2010-07-01 2015-08-20 Azevan Pharmaceuticals, Inc. Methods for treating post traumatic stress disorder
KR20130120458A (ko) 2010-09-10 2013-11-04 셈프라 파마슈티컬스, 인크. 질환을 치료하기 위한 수소결합 형성 플루오로 케토라이드
WO2013148891A1 (en) 2012-03-27 2013-10-03 Cempra Pharmaceuticals, Inc. Parenteral formulations for administering macrolide antibiotics
WO2014152326A1 (en) 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
AU2014233240B2 (en) 2013-03-15 2018-08-09 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents
BR112016022575A2 (pt) 2014-03-28 2017-08-15 Azevan Pharmaceuticals Inc Composições e métodos para o tratamento de doenças neurodegenerativas
KR102790657B1 (ko) * 2017-09-15 2025-04-02 아제반 파마슈티칼스, 인코퍼레이티드 뇌 손상을 치료하기 위한 조성물 및 방법

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US8048874B2 (en) 2011-11-01
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US20120220765A1 (en) 2012-08-30
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