JP5057780B2 - スタウロスポリン誘導体の新規医薬的使用 - Google Patents
スタウロスポリン誘導体の新規医薬的使用 Download PDFInfo
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- JP5057780B2 JP5057780B2 JP2006515982A JP2006515982A JP5057780B2 JP 5057780 B2 JP5057780 B2 JP 5057780B2 JP 2006515982 A JP2006515982 A JP 2006515982A JP 2006515982 A JP2006515982 A JP 2006515982A JP 5057780 B2 JP5057780 B2 JP 5057780B2
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Classifications
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
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Landscapes
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US47957503P | 2003-06-18 | 2003-06-18 | |
| US60/479,575 | 2003-06-18 | ||
| PCT/EP2004/006562 WO2004112794A2 (en) | 2003-06-18 | 2004-06-17 | New pharmaceutical uses of staurosporine derivatives |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2012101493A Division JP2012144572A (ja) | 2003-06-18 | 2012-04-26 | スタウロスポリン誘導体の新規医薬的使用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2006527727A JP2006527727A (ja) | 2006-12-07 |
| JP2006527727A5 JP2006527727A5 (es) | 2007-07-26 |
| JP5057780B2 true JP5057780B2 (ja) | 2012-10-24 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2006515982A Expired - Lifetime JP5057780B2 (ja) | 2003-06-18 | 2004-06-17 | スタウロスポリン誘導体の新規医薬的使用 |
| JP2012101493A Pending JP2012144572A (ja) | 2003-06-18 | 2012-04-26 | スタウロスポリン誘導体の新規医薬的使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012101493A Pending JP2012144572A (ja) | 2003-06-18 | 2012-04-26 | スタウロスポリン誘導体の新規医薬的使用 |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US8575146B2 (es) |
| EP (1) | EP1638574B1 (es) |
| JP (2) | JP5057780B2 (es) |
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| BE (1) | BE2017C067I2 (es) |
| BR (1) | BRPI0411563B8 (es) |
| CA (2) | CA2785950A1 (es) |
| CY (2) | CY1110179T1 (es) |
| DE (1) | DE602004026578D1 (es) |
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| FR (1) | FR17C1063I2 (es) |
| HK (1) | HK1095519A1 (es) |
| HU (1) | HUS000503I2 (es) |
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| MX (1) | MXPA05013722A (es) |
| NL (1) | NL300917I2 (es) |
| PL (1) | PL1638574T3 (es) |
| PT (1) | PT1638574E (es) |
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| TW (1) | TWI324604B (es) |
| WO (1) | WO2004112794A2 (es) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012144572A (ja) * | 2003-06-18 | 2012-08-02 | Novartis Ag | スタウロスポリン誘導体の新規医薬的使用 |
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|---|---|---|---|---|
| US20060014165A1 (en) * | 2003-07-14 | 2006-01-19 | Decode Genetics Ehf. | Methods of diagnosis and treatment for asthma and other respiratory diseases based on haplotype association |
| DE602004020654D1 (de) | 2003-11-18 | 2009-05-28 | Novartis Ag | Hemmer der mutanten form von kit |
| WO2005115385A1 (en) * | 2004-05-24 | 2005-12-08 | Ab Science | Use of c-kit inhibitors for treating acne |
| AU2005274852B2 (en) * | 2004-07-19 | 2011-12-08 | The Johns Hopkins University | FLT3 inhibitors for immune suppression |
| MX2007001155A (es) * | 2004-07-29 | 2007-08-14 | Creabilis Therapeutics Spa | Uso de inhibidores de k-252a y de quinasa para la prevencion o el tratamiento de patologias asociadas con hmgb1. |
| GB0419159D0 (en) * | 2004-08-27 | 2004-09-29 | Novartis Ag | Organic compounds |
| CA2606716C (en) * | 2005-05-02 | 2013-07-23 | Novartis Ag | Use of pyrimidylaminobenzamide derivatives for the treatment of systematic mastocytosis |
| AU2006271652B2 (en) * | 2005-07-20 | 2010-04-29 | Peter Valent | Compositions for treatment of systemic mastocytosis |
| RU2443421C2 (ru) * | 2005-11-14 | 2012-02-27 | Университэт Цюрих | Производные стауроспорина для применения при лечении альвеолярной рабдомиосаркомы |
| WO2009092442A1 (en) * | 2008-01-23 | 2009-07-30 | Universidad De Barcelona | Treatment of portal hypertension and related conditions by combined inhibition of the vegf and pdgf signalling pathways |
| WO2012064981A2 (en) | 2010-11-10 | 2012-05-18 | National Jewish Health | Methods to test allergic conditions |
| BR112021008516A2 (pt) | 2018-11-01 | 2021-09-14 | Syros Pharmaceuticals, Inc. | Inibidores de quinase 7 dependente de ciclina (cdk 7) |
| US11325978B2 (en) * | 2018-11-06 | 2022-05-10 | The United States Of America, As Represented By The Secretary Of The Department Of Health And Human Services | Compositions and methods for treating beta-globinopathies |
| US11839619B2 (en) * | 2019-09-16 | 2023-12-12 | The Regents Of The University Of California | Methods for treatment of pediatric systemic mastocytosis |
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| US4639455A (en) * | 1984-10-02 | 1987-01-27 | Key Pharmaceuticals, Inc. | Means of aiding in the prevention of sudden infant death syndrome |
| JPH0826037B2 (ja) | 1987-01-22 | 1996-03-13 | 協和醗酵工業株式会社 | 生理活性物質ｋ−２５２の誘導体 |
| US5093330A (en) * | 1987-06-15 | 1992-03-03 | Ciba-Geigy Corporation | Staurosporine derivatives substituted at methylamino nitrogen |
| CA2046801C (en) | 1990-08-07 | 2002-02-26 | Peter D. Davis | Substituted pyrroles |
| EP0518468B1 (en) * | 1991-05-09 | 1999-06-30 | Neurim Pharmaceuticals (1991) Limited | Melatonin containing compositions |
| AR004480A1 (es) * | 1995-04-06 | 1998-12-16 | Amico Derin C D | Compuestos de ascomicina que poseen actividad antiinflamatoria, pro cedimiento para prepararlos, uso de dichos compuestos para preparar agentesfarmaceuticos y composiciones farmaceuticas que los incluyen |
| US6184217B1 (en) * | 1996-06-25 | 2001-02-06 | Cephalon, Inc. | Use of K-252a derivative |
| US6093740A (en) * | 1997-04-30 | 2000-07-25 | Eli Lilly And Company | Therapeutic treatment for skin disorders |
| WO1999062537A1 (en) * | 1998-06-04 | 1999-12-09 | The Rockefeller University | Methods and agents for modulating the immune response and inflammation involving monocyte and dendritic cell membrane proteins |
| GB9903547D0 (en) * | 1999-02-16 | 1999-04-07 | Novartis Ag | Organic compounds |
| MXPA03005139A (es) * | 2000-12-08 | 2004-01-29 | Ortho Mcneil Pharm Inc | Compuestos macroheterociclicos utiles como inhibidores de cinasa. |
| GB0108606D0 (en) * | 2001-04-05 | 2001-05-23 | Novartis Ag | Organic compounds |
| US20030091974A1 (en) * | 2001-06-29 | 2003-05-15 | Alain Moussy | Method for screening compounds capable of depleting mast cells |
| US20050176687A1 (en) * | 2001-06-29 | 2005-08-11 | Alain Moussy | Use of tyrosine kinase inhibitors for treating autoimmune diseases |
| WO2003037347A1 (en) | 2001-10-30 | 2003-05-08 | Novartis Ag | Staurosporine derivatives as inhibitors of flt3 receptor tyrosine kinase activity |
| US6998391B2 (en) | 2002-02-07 | 2006-02-14 | Supergen.Inc. | Method for treating diseases associated with abnormal kinase activity |
| JPWO2004091663A1 (ja) | 2003-04-18 | 2006-07-06 | 協和醗酵工業株式会社 | 神経再生薬 |
| WO2004093910A1 (ja) * | 2003-04-22 | 2004-11-04 | Astellas Pharma Inc. | ＰＰＡＲδアゴニストによる脳神経変性疾患治療剤 |
| TWI324604B (en) * | 2003-06-18 | 2010-05-11 | Novartis Ag | New use of staurosporine derivatives |
| DE602004020654D1 (de) | 2003-11-18 | 2009-05-28 | Novartis Ag | Hemmer der mutanten form von kit |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012144572A (ja) * | 2003-06-18 | 2012-08-02 | Novartis Ag | スタウロスポリン誘導体の新規医薬的使用 |
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