JP4990155B2 - プロテアソームを阻害するための組成物 - Google Patents

プロテアソームを阻害するための組成物 Download PDF

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JP4990155B2
JP4990155B2 JP2007544636A JP2007544636A JP4990155B2 JP 4990155 B2 JP4990155 B2 JP 4990155B2 JP 2007544636 A JP2007544636 A JP 2007544636A JP 2007544636 A JP2007544636 A JP 2007544636A JP 4990155 B2 JP4990155 B2 JP 4990155B2
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alkyl
hydrogen
absent
aryl
aralkyl
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JP2008522981A5 (OSRAM
JP2008522981A (ja
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エバン アール. ルイス,
マーク グエン ホー,
フェビアナ エヌ. フォンセカ,
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プロテオリックス, インコーポレイテッド
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    • A61K31/336Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having three-membered rings, e.g. oxirane, fumagillin
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JP2007544636A 2004-12-07 2005-12-07 プロテアソームを阻害するための組成物 Expired - Lifetime JP4990155B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US63436604P 2004-12-07 2004-12-07
US60/634,366 2004-12-07
US65593005P 2005-02-23 2005-02-23
US60/655,930 2005-02-23
PCT/US2005/044451 WO2006063154A1 (en) 2004-12-07 2005-12-07 Composition for proteasome inhibition

Publications (3)

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JP2008522981A JP2008522981A (ja) 2008-07-03
JP2008522981A5 JP2008522981A5 (OSRAM) 2008-10-02
JP4990155B2 true JP4990155B2 (ja) 2012-08-01

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JP2007544636A Expired - Lifetime JP4990155B2 (ja) 2004-12-07 2005-12-07 プロテアソームを阻害するための組成物

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US (1) US7737112B2 (OSRAM)
EP (3) EP2260835B1 (OSRAM)
JP (1) JP4990155B2 (OSRAM)
KR (1) KR101299821B1 (OSRAM)
CN (2) CN101180071A (OSRAM)
AT (1) ATE499109T1 (OSRAM)
AU (1) AU2005313975B2 (OSRAM)
CA (1) CA2589921C (OSRAM)
CY (1) CY1111489T1 (OSRAM)
DE (1) DE602005026556D1 (OSRAM)
DK (1) DK1819353T3 (OSRAM)
ES (2) ES2549763T3 (OSRAM)
HU (1) HUE027850T2 (OSRAM)
IL (1) IL183607A (OSRAM)
PL (3) PL2260835T3 (OSRAM)
PT (3) PT2260835E (OSRAM)
WO (1) WO2006063154A1 (OSRAM)

Families Citing this family (53)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8129346B2 (en) 2004-04-15 2012-03-06 Onyx Therapeutics, Inc. Compounds for enzyme inhibition
US8198270B2 (en) * 2004-04-15 2012-06-12 Onyx Therapeutics, Inc. Compounds for proteasome enzyme inhibition
CA2565407A1 (en) * 2004-05-10 2005-11-24 Proteolix, Inc. Compounds for enzyme inhibition
US9034846B2 (en) * 2004-10-10 2015-05-19 Universite De Liege Use of cyclodextrin for treatment and prevention of bronchial inflammatory diseases
KR101434522B1 (ko) * 2005-11-09 2014-08-26 오닉스 세라퓨틱스, 인크. 효소 저해를 위한 화합물
US7691852B2 (en) * 2006-06-19 2010-04-06 Onyx Therapeutics, Inc. Compounds for enzyme inhibition
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