AU2005313975B2 - Composition for proteasome inhibition - Google Patents
Composition for proteasome inhibition Download PDFInfo
- Publication number
- AU2005313975B2 AU2005313975B2 AU2005313975A AU2005313975A AU2005313975B2 AU 2005313975 B2 AU2005313975 B2 AU 2005313975B2 AU 2005313975 A AU2005313975 A AU 2005313975A AU 2005313975 A AU2005313975 A AU 2005313975A AU 2005313975 B2 AU2005313975 B2 AU 2005313975B2
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- Prior art keywords
- alkyl
- hydrogen
- aryl
- absent
- salkyl
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- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/336—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having three-membered rings, e.g. oxirane, fumagillin
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
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- Health & Medical Sciences (AREA)
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2012261655A AU2012261655C1 (en) | 2004-12-07 | 2012-12-06 | Composition for proteasome inhibition |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US63436604P | 2004-12-07 | 2004-12-07 | |
| US60/634,366 | 2004-12-07 | ||
| US65593005P | 2005-02-23 | 2005-02-23 | |
| US60/655,930 | 2005-02-23 | ||
| PCT/US2005/044451 WO2006063154A1 (en) | 2004-12-07 | 2005-12-07 | Composition for proteasome inhibition |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2012261655A Division AU2012261655C1 (en) | 2004-12-07 | 2012-12-06 | Composition for proteasome inhibition |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2005313975A1 AU2005313975A1 (en) | 2006-06-15 |
| AU2005313975B2 true AU2005313975B2 (en) | 2012-09-06 |
Family
ID=36143200
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2005313975A Active 2030-12-07 AU2005313975B2 (en) | 2004-12-07 | 2005-12-07 | Composition for proteasome inhibition |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US7737112B2 (OSRAM) |
| EP (3) | EP2260835B1 (OSRAM) |
| JP (1) | JP4990155B2 (OSRAM) |
| KR (1) | KR101299821B1 (OSRAM) |
| CN (2) | CN101180071A (OSRAM) |
| AT (1) | ATE499109T1 (OSRAM) |
| AU (1) | AU2005313975B2 (OSRAM) |
| CA (1) | CA2589921C (OSRAM) |
| CY (1) | CY1111489T1 (OSRAM) |
| DE (1) | DE602005026556D1 (OSRAM) |
| DK (1) | DK1819353T3 (OSRAM) |
| ES (2) | ES2549763T3 (OSRAM) |
| HU (1) | HUE027850T2 (OSRAM) |
| IL (1) | IL183607A (OSRAM) |
| PL (3) | PL2260835T3 (OSRAM) |
| PT (3) | PT2260835E (OSRAM) |
| WO (1) | WO2006063154A1 (OSRAM) |
Families Citing this family (53)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8129346B2 (en) | 2004-04-15 | 2012-03-06 | Onyx Therapeutics, Inc. | Compounds for enzyme inhibition |
| US8198270B2 (en) * | 2004-04-15 | 2012-06-12 | Onyx Therapeutics, Inc. | Compounds for proteasome enzyme inhibition |
| CA2565407A1 (en) * | 2004-05-10 | 2005-11-24 | Proteolix, Inc. | Compounds for enzyme inhibition |
| US9034846B2 (en) * | 2004-10-10 | 2015-05-19 | Universite De Liege | Use of cyclodextrin for treatment and prevention of bronchial inflammatory diseases |
| KR101434522B1 (ko) * | 2005-11-09 | 2014-08-26 | 오닉스 세라퓨틱스, 인크. | 효소 저해를 위한 화합물 |
| US7691852B2 (en) * | 2006-06-19 | 2010-04-06 | Onyx Therapeutics, Inc. | Compounds for enzyme inhibition |
| RS54847B2 (sr) | 2007-10-04 | 2019-09-30 | Onyx Therapeutics Inc | Inhibitori kristalne peptid epoksi keton proteaze i sinteza aminokiselinskih keto-epoksida |
| US7635773B2 (en) | 2008-04-28 | 2009-12-22 | Cydex Pharmaceuticals, Inc. | Sulfoalkyl ether cyclodextrin compositions |
| WO2010039762A2 (en) * | 2008-10-01 | 2010-04-08 | Dr. Reddy's Laboratories Ltd. | Pharmaceutical compositions comprising boronic acid compounds |
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