JP4831906B2 - Ｃｘｃｒ３機能を調節するための複素環式化合物および方法 - Google Patents
Ｃｘｃｒ３機能を調節するための複素環式化合物および方法 Download PDFInfo
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- JP4831906B2 JP4831906B2 JP2001519682A JP2001519682A JP4831906B2 JP 4831906 B2 JP4831906 B2 JP 4831906B2 JP 2001519682 A JP2001519682 A JP 2001519682A JP 2001519682 A JP2001519682 A JP 2001519682A JP 4831906 B2 JP4831906 B2 JP 4831906B2
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- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
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- A61P11/06—Antiasthmatics
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- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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| US60/151,212 | 1999-08-27 | ||
| PCT/US2000/023556 WO2001016114A2 (en) | 1999-08-27 | 2000-08-25 | Heterocyclic compounds and methods for modulating cxcr3 function |
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| AU729415B2 (en) | 1996-07-12 | 2001-02-01 | Millennium Pharmaceuticals, Inc. | Chemokine receptor antagonists and methods of use therefor |
| US5919776A (en) | 1996-12-20 | 1999-07-06 | Merck & Co., Inc. | Substituted aminoquinolines as modulators of chemokine receptor activity |
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| EP1091960A1 (en) | 1998-06-29 | 2001-04-18 | The Regents Of The University Of California | Bifunctional antagonists of cytokine-sensitive protein kinase activation cascades and methods for use as anti-inflammatory agents |
| US6617115B1 (en) | 1999-10-27 | 2003-09-09 | Cytokinetics, Inc. | Methods of screening for modulators of cell proliferation |
| US6545004B1 (en) | 1999-10-27 | 2003-04-08 | Cytokinetics, Inc. | Methods and compositions utilizing quinazolinones |
| MXPA02004162A (es) | 1999-10-27 | 2003-08-20 | Cytokinetics Inc | Metodo y composiciones que utilizan quinazolinonas. |
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| US20030119854A1 (en) | 2003-06-26 |
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| AU7080500A (en) | 2001-03-26 |
| ES2272319T3 (es) | 2007-05-01 |
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| US6559160B1 (en) | 2003-05-06 |
| WO2001016114A3 (en) | 2001-08-02 |
| US6992084B2 (en) | 2006-01-31 |
| US20060063763A1 (en) | 2006-03-23 |
| EP1216232B1 (en) | 2006-10-11 |
| DE60031285D1 (de) | 2006-11-23 |
| DE60031285T2 (de) | 2007-08-30 |
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