JP4334229B2 - プロポフォール及びスルホアルキルエーテルシクロデキストリン含有製剤 - Google Patents

プロポフォール及びスルホアルキルエーテルシクロデキストリン含有製剤 Download PDF

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JP4334229B2
JP4334229B2 JP2002572914A JP2002572914A JP4334229B2 JP 4334229 B2 JP4334229 B2 JP 4334229B2 JP 2002572914 A JP2002572914 A JP 2002572914A JP 2002572914 A JP2002572914 A JP 2002572914A JP 4334229 B2 JP4334229 B2 JP 4334229B2
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propofol
formulation
sae
liquid
cyclodextrin
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Japanese (ja)
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JP2004526730A (ja
JP2004526730A5 (enExample
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ジェロルド・エル・モーシャー
ダイアン・オー・トムプソン
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サイデックス・ファーマシューティカルズ・インコーポレイテッド
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    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B82—NANOTECHNOLOGY
    • B82Y—SPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00—Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/05—Phenols
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/716—Glucans
    • A61K31/724—Cyclodextrins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A61P23/02—Local anaesthetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Anesthesiology (AREA)
  • Molecular Biology (AREA)
  • Nanotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Biophysics (AREA)
  • Biotechnology (AREA)
  • General Engineering & Computer Science (AREA)
  • Medical Informatics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
JP2002572914A 2001-03-20 2002-03-19 プロポフォール及びスルホアルキルエーテルシクロデキストリン含有製剤 Expired - Fee Related JP4334229B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27730501P 2001-03-20 2001-03-20
PCT/US2002/008596 WO2002074200A1 (en) 2001-03-20 2002-03-19 Formulations containing propofol and a sulfoalkyl ether cyclodextrin

Publications (3)

Publication Number Publication Date
JP2004526730A JP2004526730A (ja) 2004-09-02
JP2004526730A5 JP2004526730A5 (enExample) 2005-12-22
JP4334229B2 true JP4334229B2 (ja) 2009-09-30

Family

ID=23060281

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002572914A Expired - Fee Related JP4334229B2 (ja) 2001-03-20 2002-03-19 プロポフォール及びスルホアルキルエーテルシクロデキストリン含有製剤

Country Status (6)

Country Link
US (1) US20030055023A1 (enExample)
EP (1) EP1383445A4 (enExample)
JP (1) JP4334229B2 (enExample)
AU (1) AU2002254309B2 (enExample)
CA (1) CA2441744C (enExample)
WO (1) WO2002074200A1 (enExample)

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US7550155B2 (en) 2002-07-29 2009-06-23 Transform Pharmaceuticals Inc. Aqueous pharmaceutical compositions of 2,6-diisopropylphenol (propofol) and their uses
US7089927B2 (en) * 2002-10-23 2006-08-15 New York University System and method for guidance of anesthesia, analgesia and amnesia
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WO2004108113A1 (en) * 2003-06-10 2004-12-16 Dinesh Shantilal Patel Improved novel, clear, painless preparation of propofol
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KR20070058608A (ko) * 2004-09-13 2007-06-08 바라트 쎄럼스 앤드 백신스 리미티드 항미생물 방부 효능을 갖는 정맥 내 투여를 위한 안정한에멀젼 조성물
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US20100204178A1 (en) 2006-10-02 2010-08-12 James Cloyd Novel parenteral carbamazepine formulation
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JP5537033B2 (ja) * 2005-12-19 2014-07-02 ザ ユニヴァーシティー オブ リヴァプール 無痛覚
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Also Published As

Publication number Publication date
EP1383445A1 (en) 2004-01-28
JP2004526730A (ja) 2004-09-02
CA2441744C (en) 2011-07-12
AU2002254309B2 (en) 2006-02-02
WO2002074200B1 (en) 2003-03-06
WO2002074200A1 (en) 2002-09-26
US20030055023A1 (en) 2003-03-20
EP1383445A4 (en) 2005-04-13
CA2441744A1 (en) 2002-09-26

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