JP4076114B2 - 4’−c−エチニルプリンヌクレオシド化合物 - Google Patents
4’−c−エチニルプリンヌクレオシド化合物 Download PDFInfo
- Publication number
- JP4076114B2 JP4076114B2 JP2000137982A JP2000137982A JP4076114B2 JP 4076114 B2 JP4076114 B2 JP 4076114B2 JP 2000137982 A JP2000137982 A JP 2000137982A JP 2000137982 A JP2000137982 A JP 2000137982A JP 4076114 B2 JP4076114 B2 JP 4076114B2
- Authority
- JP
- Japan
- Prior art keywords
- compound
- group
- ethynyl
- mmol
- residue
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 0 C[*+][C@@](COCc1ccccc1)(C(C1OC(C)=O)OCc2ccccc2)O[C@]1N(C=CC(N1)=O)C1=O Chemical compound C[*+][C@@](COCc1ccccc1)(C(C1OC(C)=O)OCc2ccccc2)O[C@]1N(C=CC(N1)=O)C1=O 0.000 description 2
- JIBSKFXABQBJBL-OQKBBGGUSA-N C[C@@](COCc1ccccc1)([C@@H]([C@@H]1OC(C)=O)OCc2ccccc2)O[C@H]1[n]1c2nc(N)nc(N)c2nc1 Chemical compound C[C@@](COCc1ccccc1)([C@@H]([C@@H]1OC(C)=O)OCc2ccccc2)O[C@H]1[n]1c2nc(N)nc(N)c2nc1 JIBSKFXABQBJBL-OQKBBGGUSA-N 0.000 description 1
- KNBGNDKDYQTJIB-KUXCXQDQSA-N C[C@@](COCc1ccccc1)([C@@H]1OCc2ccccc2)O[C@@H](CCCCOC(C)=O)[C@H]1OC(C)=O Chemical compound C[C@@](COCc1ccccc1)([C@@H]1OCc2ccccc2)O[C@@H](CCCCOC(C)=O)[C@H]1OC(C)=O KNBGNDKDYQTJIB-KUXCXQDQSA-N 0.000 description 1
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- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2000137982A JP4076114B2 (ja) | 1999-05-12 | 2000-05-11 | 4’−c−エチニルプリンヌクレオシド化合物 |
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP13153999 | 1999-05-12 | ||
| JP17492099 | 1999-06-22 | ||
| JP31824699 | 1999-11-09 | ||
| JP11-174920 | 2000-03-23 | ||
| JP11-318246 | 2000-03-23 | ||
| JP11-131539 | 2000-03-23 | ||
| JP2000081117 | 2000-03-23 | ||
| JP2000-81117 | 2000-03-23 | ||
| JP2000137982A JP4076114B2 (ja) | 1999-05-12 | 2000-05-11 | 4’−c−エチニルプリンヌクレオシド化合物 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007314092A Division JP2008110983A (ja) | 1999-05-12 | 2007-12-05 | 4’−c−エチニルヌクレオシド化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2001335592A JP2001335592A (ja) | 2001-12-04 |
| JP2001335592A5 JP2001335592A5 (enExample) | 2007-08-30 |
| JP4076114B2 true JP4076114B2 (ja) | 2008-04-16 |
Family
ID=27527275
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000137982A Expired - Lifetime JP4076114B2 (ja) | 1999-05-12 | 2000-05-11 | 4’−c−エチニルプリンヌクレオシド化合物 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JP4076114B2 (enExample) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2502109C (en) * | 2004-03-24 | 2010-02-23 | Yamasa Corporation | 4'-c-substituted-2-haloadenosine derivative |
| JP2008069182A (ja) * | 2004-03-24 | 2008-03-27 | Yamasa Shoyu Co Ltd | 4’−c−置換−2−ハロアデノシン誘導体 |
| MX356509B (es) | 2011-12-22 | 2018-05-30 | Alios Biopharma Inc | Nucleósidos sustituidos, nucleótidos y análogos de los mismos. |
| SG11201405351RA (en) * | 2012-03-21 | 2014-10-30 | Alios Biopharma Inc | Substituted nucleosides, nucleotides and analogs thereof |
| USRE48171E1 (en) | 2012-03-21 | 2020-08-25 | Janssen Biopharma, Inc. | Substituted nucleosides, nucleotides and analogs thereof |
| US9441007B2 (en) | 2012-03-21 | 2016-09-13 | Alios Biopharma, Inc. | Substituted nucleosides, nucleotides and analogs thereof |
| JP6191989B2 (ja) * | 2014-02-12 | 2017-09-06 | 学校法人東京理科大学 | アデニン誘導体又はその薬理学的に許容しうる塩、その製造方法、及びその用途 |
| EP3543238B1 (en) | 2016-11-16 | 2021-05-19 | National Center for Global Health and Medicine | Nucleoside derivatives having anti-viral activity |
| KR102686384B1 (ko) * | 2019-04-05 | 2024-07-17 | 가부시기가이샤 닛뽕쇼꾸바이 | 가교형 인공 뉴클레오시드의 제조 |
-
2000
- 2000-05-11 JP JP2000137982A patent/JP4076114B2/ja not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| JP2001335592A (ja) | 2001-12-04 |
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