JP2025514336A5 - - Google Patents
Info
- Publication number
- JP2025514336A5 JP2025514336A5 JP2024563656A JP2024563656A JP2025514336A5 JP 2025514336 A5 JP2025514336 A5 JP 2025514336A5 JP 2024563656 A JP2024563656 A JP 2024563656A JP 2024563656 A JP2024563656 A JP 2024563656A JP 2025514336 A5 JP2025514336 A5 JP 2025514336A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- compound
- substituted
- cyano
- mmol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202210456939 | 2022-04-27 | ||
| CN202210456939.3 | 2022-04-27 | ||
| PCT/CN2023/091140 WO2023208108A1 (zh) | 2022-04-27 | 2023-04-27 | 可用于降尿酸的化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2025514336A JP2025514336A (ja) | 2025-05-02 |
| JP2025514336A5 true JP2025514336A5 (enExample) | 2025-10-08 |
| JP7792730B2 JP7792730B2 (ja) | 2025-12-26 |
Family
ID=87872273
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024563656A Active JP7792730B2 (ja) | 2022-04-27 | 2023-04-27 | 尿酸を降下させるために使用できる化合物 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20250282753A1 (enExample) |
| EP (1) | EP4516781A4 (enExample) |
| JP (1) | JP7792730B2 (enExample) |
| CN (1) | CN116715633B (enExample) |
| TW (1) | TWI870839B (enExample) |
| WO (1) | WO2023208108A1 (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN119241538A (zh) * | 2024-09-30 | 2025-01-03 | 陕西科技大学 | 一类三唑并吡啶结构的化合物、合成方法及其应用 |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050090529A1 (en) * | 2003-07-31 | 2005-04-28 | Pfizer Inc | 3,5 Disubstituted indazole compounds with nitrogen-bearing 5-membered heterocycles, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation |
| MX2008001778A (es) * | 2005-08-19 | 2008-04-07 | Aventis Pharma Inc | Combinacion de un agente hipnotico y un compuesto de bis arilo y heteroarilo sustituido y aplicacion terapeutica de la misma. |
| CA2623327A1 (en) * | 2005-10-07 | 2007-04-19 | Kissei Pharmaceutical Co., Ltd. | Nitrogenated heterocyclic compound and pharmaceutical composition comprising the same |
| JPWO2010044403A1 (ja) * | 2008-10-15 | 2012-03-15 | キッセイ薬品工業株式会社 | 5員環ヘテロアリール誘導体及びその医薬用途 |
| WO2010044404A1 (ja) * | 2008-10-15 | 2010-04-22 | キッセイ薬品工業株式会社 | 縮合複素環誘導体及びその医薬用途 |
| WO2010093191A2 (en) * | 2009-02-13 | 2010-08-19 | Lg Life Sciences Ltd. | Novel compounds effective as xanthine oxidase inhibitors, method for preparing the same, and pharmaceutical composition containing the same |
| TWI423962B (zh) * | 2009-10-07 | 2014-01-21 | Lg Life Sciences Ltd | 有效作為黃嘌呤氧化酶抑制劑之新穎化合物、其製備方法及含該化合物之醫藥組成物 |
| JP5990106B2 (ja) * | 2011-01-28 | 2016-09-07 | 佐藤製薬株式会社 | 縮環化合物 |
| TWI548630B (zh) * | 2011-04-06 | 2016-09-11 | Lg生命科學有限公司 | 1-(3-氰基-1-異丙基-吲哚-5-基)吡唑-4-羧酸結晶型及其製造方法 |
| KR20150138212A (ko) * | 2013-03-29 | 2015-12-09 | 데이진 화-마 가부시키가이샤 | 피라졸 유도체 |
| CN105439946B (zh) * | 2014-08-13 | 2018-02-02 | 益方生物科技(上海)有限公司 | 羧酸化合物及其制备方法和用途 |
| KR20170105021A (ko) * | 2015-01-28 | 2017-09-18 | 아스테라스 세이야쿠 가부시키가이샤 | 피라진카르복사마이드 화합물의 제조 방법 및 그 합성 중간체 |
| JP6873904B2 (ja) * | 2015-08-28 | 2021-05-19 | Ils株式会社 | キサンチンオキシダーゼ阻害剤 |
| HUE052608T2 (hu) * | 2015-09-02 | 2021-05-28 | Sunshine Lake Pharma Co Ltd | Karboxi-szubsztituált (hetero) aromás gyûrûs származékok, elõállítási eljárásaik és alkalmazásaik |
| EA037280B1 (ru) * | 2015-09-10 | 2021-03-03 | Цзянсу Атом Байосайенс Энд Фармасьютикал Ко., Лтд. | Группа соединений, применяющихся для лечения или предупреждения гиперурикемии или подагры |
| CN107759588B (zh) * | 2016-08-19 | 2020-10-23 | 江苏新元素医药科技有限公司 | 一类苯基-(吡唑并[1,5-a]吡啶-3-基)甲酮衍生物 |
| BR112021001709A2 (pt) * | 2018-08-01 | 2021-05-04 | Araxes Pharma Llc | compostos espiro heterocíclicos e métodos de uso dos mesmos para o tratamento de câncer |
| CN116438175B (zh) * | 2020-11-11 | 2025-07-22 | 南京明德新药研发有限公司 | 苯并脲环衍生物及其制备方法和应用 |
| WO2022233264A1 (zh) * | 2021-05-07 | 2022-11-10 | 江苏新元素医药科技有限公司 | 一类黄嘌呤氧化酶抑制剂 |
-
2023
- 2023-04-27 JP JP2024563656A patent/JP7792730B2/ja active Active
- 2023-04-27 EP EP23795540.6A patent/EP4516781A4/en active Pending
- 2023-04-27 TW TW112115878A patent/TWI870839B/zh active
- 2023-04-27 US US18/860,252 patent/US20250282753A1/en active Pending
- 2023-04-27 CN CN202310469300.3A patent/CN116715633B/zh active Active
- 2023-04-27 WO PCT/CN2023/091140 patent/WO2023208108A1/zh not_active Ceased
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