JP2025509736A5 - - Google Patents
Info
- Publication number
- JP2025509736A5 JP2025509736A5 JP2024555118A JP2024555118A JP2025509736A5 JP 2025509736 A5 JP2025509736 A5 JP 2025509736A5 JP 2024555118 A JP2024555118 A JP 2024555118A JP 2024555118 A JP2024555118 A JP 2024555118A JP 2025509736 A5 JP2025509736 A5 JP 2025509736A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- inhibitors
- linker
- heteroaryl
- alkynyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17/695,259 US20230097887A1 (en) | 2018-04-09 | 2022-03-15 | Bi-functional Molecules to Degrade Circulating Proteins |
| US17/695,259 | 2022-03-15 | ||
| PCT/US2023/064436 WO2023178179A2 (en) | 2022-03-15 | 2023-03-15 | Bi-functional molecules to degrade circulating proteins |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025509736A JP2025509736A (ja) | 2025-04-11 |
| JP2025509736A5 true JP2025509736A5 (https=) | 2026-03-24 |
Family
ID=88024435
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024555118A Pending JP2025509736A (ja) | 2022-03-15 | 2023-03-15 | 循環タンパク質を分解するための二官能性分子 |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP4493220A2 (https=) |
| JP (1) | JP2025509736A (https=) |
| KR (1) | KR20250004953A (https=) |
| CN (1) | CN119212726A (https=) |
| AU (1) | AU2023234543A1 (https=) |
| IL (1) | IL315581A (https=) |
| MX (1) | MX2024011358A (https=) |
| WO (1) | WO2023178179A2 (https=) |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3356415B1 (en) * | 2015-09-29 | 2024-05-01 | Amgen Inc. | Asgr inhibitors for reduzing cholesterol levels |
| WO2019199621A1 (en) * | 2018-04-09 | 2019-10-17 | Yale University | Bi-functional molecules to degrade circulating proteins |
| EP3773727A4 (en) * | 2018-04-09 | 2022-05-04 | Yale University | BIFUNCTIONAL SMALL MOLECULES TO TARGETING THE SELECTIVE DEGRADATION OF CIRCULATING PROTEINS |
| AU2019404061A1 (en) * | 2018-12-19 | 2021-07-22 | The Board Of Trustees Of The Leland Stanford Junior University | Bifunctional molecules for lysosomal targeting and related compositions and methods |
| WO2021155317A1 (en) * | 2020-01-31 | 2021-08-05 | Avilar Therapeutics, Inc. | Asgpr-binding compounds for the degradation of extracellular proteins |
-
2023
- 2023-03-15 KR KR1020247033971A patent/KR20250004953A/ko active Pending
- 2023-03-15 JP JP2024555118A patent/JP2025509736A/ja active Pending
- 2023-03-15 AU AU2023234543A patent/AU2023234543A1/en active Pending
- 2023-03-15 CN CN202380040375.8A patent/CN119212726A/zh active Pending
- 2023-03-15 WO PCT/US2023/064436 patent/WO2023178179A2/en not_active Ceased
- 2023-03-15 EP EP23771634.5A patent/EP4493220A2/en active Pending
- 2023-03-15 IL IL315581A patent/IL315581A/en unknown
-
2024
- 2024-09-13 MX MX2024011358A patent/MX2024011358A/es unknown
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