JP2025502240A5 - - Google Patents

Info

Publication number
JP2025502240A5
JP2025502240A5 JP2024541916A JP2024541916A JP2025502240A5 JP 2025502240 A5 JP2025502240 A5 JP 2025502240A5 JP 2024541916 A JP2024541916 A JP 2024541916A JP 2024541916 A JP2024541916 A JP 2024541916A JP 2025502240 A5 JP2025502240 A5 JP 2025502240A5
Authority
JP
Japan
Prior art keywords
trifluoromethyl
salt
triazine
amine
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024541916A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025502240A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2023/050208 external-priority patent/WO2023135057A1/en
Publication of JP2025502240A publication Critical patent/JP2025502240A/ja
Publication of JP2025502240A5 publication Critical patent/JP2025502240A5/ja
Pending legal-status Critical Current

Links

JP2024541916A 2022-01-11 2023-01-06 がんの治療のための二環式トリアジン誘導体 Pending JP2025502240A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP22150829 2022-01-11
EP22150829.4 2022-01-11
PCT/EP2023/050208 WO2023135057A1 (en) 2022-01-11 2023-01-06 Bicyclic triazine derivatives for the treatment of cancer

Publications (2)

Publication Number Publication Date
JP2025502240A JP2025502240A (ja) 2025-01-24
JP2025502240A5 true JP2025502240A5 (https=) 2026-01-06

Family

ID=79927598

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024541916A Pending JP2025502240A (ja) 2022-01-11 2023-01-06 がんの治療のための二環式トリアジン誘導体

Country Status (9)

Country Link
US (1) US20250066370A1 (https=)
EP (1) EP4463458A1 (https=)
JP (1) JP2025502240A (https=)
KR (1) KR20240134962A (https=)
CN (1) CN118541372A (https=)
AU (1) AU2023207765A1 (https=)
CA (1) CA3246440A1 (https=)
IL (1) IL313835A (https=)
WO (1) WO2023135057A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021176045A1 (en) * 2020-03-06 2021-09-10 Bayer Aktiengesellschaft Imidazotriazines acting on cancer via inhibition of cdk12

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011529072A (ja) 2008-07-24 2011-12-01 セラヴァンス, インコーポレーテッド 二重作用血圧降下薬
US8791162B2 (en) 2011-02-14 2014-07-29 Merck Sharp & Dohme Corp. Cathepsin cysteine protease inhibitors
MX2019012431A (es) 2017-04-21 2020-08-03 Ikena Oncology Inc Inhibidores del receptor de hidrocarburos de arilo (ahr) de indol y usos de los mismos.
TW202146416A (zh) 2019-12-11 2021-12-16 德商拜耳廠股份有限公司 吡唑并三𠯤
WO2021176045A1 (en) 2020-03-06 2021-09-10 Bayer Aktiengesellschaft Imidazotriazines acting on cancer via inhibition of cdk12
WO2021176049A1 (en) 2020-03-06 2021-09-10 Bayer Aktiengesellschaft Pyrazolopyrazines acting on cancers via inhibition of cdk12

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