JP2025165975A5 - - Google Patents

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Publication number
JP2025165975A5
JP2025165975A5 JP2025120662A JP2025120662A JP2025165975A5 JP 2025165975 A5 JP2025165975 A5 JP 2025165975A5 JP 2025120662 A JP2025120662 A JP 2025120662A JP 2025120662 A JP2025120662 A JP 2025120662A JP 2025165975 A5 JP2025165975 A5 JP 2025165975A5
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JP
Japan
Prior art keywords
compound
formula
pharmaceutically acceptable
acceptable salt
cancer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2025120662A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025165975A (ja
Filing date
Publication date
Priority claimed from JP2021578240A external-priority patent/JP7805170B2/ja
Application filed filed Critical
Publication of JP2025165975A publication Critical patent/JP2025165975A/ja
Publication of JP2025165975A5 publication Critical patent/JP2025165975A5/ja
Pending legal-status Critical Current

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JP2025120662A 2019-07-02 2025-07-17 前立腺特異的膜抗原(psma)リガンド及びその使用 Pending JP2025165975A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP19184015 2019-07-02
EP19184015.6 2019-07-02
JP2021578240A JP7805170B2 (ja) 2019-07-02 2020-06-30 前立腺特異的膜抗原(psma)リガンド及びその使用
PCT/EP2020/068386 WO2021001360A1 (en) 2019-07-02 2020-06-30 Prostate specific membrane antigen (psma) ligands and uses thereof

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2021578240A Division JP7805170B2 (ja) 2019-07-02 2020-06-30 前立腺特異的膜抗原(psma)リガンド及びその使用

Publications (2)

Publication Number Publication Date
JP2025165975A JP2025165975A (ja) 2025-11-05
JP2025165975A5 true JP2025165975A5 (https=) 2026-02-13

Family

ID=67145647

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021578240A Active JP7805170B2 (ja) 2019-07-02 2020-06-30 前立腺特異的膜抗原(psma)リガンド及びその使用
JP2025120662A Pending JP2025165975A (ja) 2019-07-02 2025-07-17 前立腺特異的膜抗原(psma)リガンド及びその使用

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2021578240A Active JP7805170B2 (ja) 2019-07-02 2020-06-30 前立腺特異的膜抗原(psma)リガンド及びその使用

Country Status (16)

Country Link
US (1) US20230226227A1 (https=)
EP (1) EP3993837A1 (https=)
JP (2) JP7805170B2 (https=)
KR (1) KR20220044496A (https=)
CN (3) CN114341118A (https=)
AR (1) AR119331A1 (https=)
AU (3) AU2020299974A1 (https=)
BR (1) BR112021026812A2 (https=)
CA (1) CA3144557A1 (https=)
CL (1) CL2021003525A1 (https=)
CO (1) CO2021017708A2 (https=)
IL (1) IL289039B1 (https=)
MX (1) MX2022000136A (https=)
PH (1) PH12021553284A1 (https=)
TW (1) TW202114742A (https=)
WO (1) WO2021001360A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL297323A (en) * 2020-04-29 2022-12-01 Novartis Ag Methods for radiological labeling of psma-binding ligands and their kits
WO2022108992A1 (en) * 2020-11-17 2022-05-27 The Johns Hopkins University Prostate-specific membrane antigen (psma)-targeted prodrug for selective killing of cells expressing psma
CN121604981A (zh) 2023-07-21 2026-03-03 诺华公司 靶向psma的放射性配体治疗方案
WO2025125469A1 (en) 2023-12-13 2025-06-19 Swiss Rockets Ag Combination therapy using psma-targeted radiopharmaceuticals and an inhibitor of pi3k, akt, and/or mtor

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2415709A1 (en) 2000-07-11 2003-01-10 Bml, Inc. Remedies for bone diseases
AU2012294639B2 (en) * 2011-08-05 2017-10-26 Molecular Insight Pharmaceuticals, Inc. Radiolabeled prostate specific membrane antigen inhibitors
EP3456700A1 (en) * 2013-10-18 2019-03-20 Deutsches Krebsforschungszentrum Labeled inhibitors of prostate specific membrane antigen (psma), their use as imaging agents and pharmaceutical agents for the treatment of prostate cancer
RS65188B1 (sr) * 2016-03-22 2024-03-29 Univ Johns Hopkins Sredstva sa visokim afinitetom za ciljano dejstvo na membranski antigen specifičan za prostatu za endoradioterapiju kancera prostate
CN111032632B (zh) * 2017-05-30 2024-04-12 约翰霍普金斯大学 用于前列腺癌的腔内放射疗法的前列腺特异性膜抗原靶向的高亲和力剂
US11813340B2 (en) * 2018-02-06 2023-11-14 The Johns Hopkins University PSMA targeted radiohalogenated urea-polyaminocarboxylates for cancer radiotherapy
US20210338846A1 (en) * 2018-07-30 2021-11-04 The Johns Hopkins University Competitive prostate-specific membrane antigen (psma) binding agents for reduction of non-target organ uptake of radiolabeled psma inhibitors for psma positive tumor imaging and radiopharmaceutical therapy

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