JP2025165975A5 - - Google Patents

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Publication number
JP2025165975A5
JP2025165975A5 JP2025120662A JP2025120662A JP2025165975A5 JP 2025165975 A5 JP2025165975 A5 JP 2025165975A5 JP 2025120662 A JP2025120662 A JP 2025120662A JP 2025120662 A JP2025120662 A JP 2025120662A JP 2025165975 A5 JP2025165975 A5 JP 2025165975A5
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JP
Japan
Prior art keywords
compound
formula
pharmaceutically acceptable
acceptable salt
cancer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2025120662A
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English (en)
Japanese (ja)
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JP2025165975A (ja
Filing date
Publication date
Priority claimed from JP2021578240A external-priority patent/JP7805170B2/ja
Application filed filed Critical
Publication of JP2025165975A publication Critical patent/JP2025165975A/ja
Publication of JP2025165975A5 publication Critical patent/JP2025165975A5/ja
Pending legal-status Critical Current

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JP2025120662A 2019-07-02 2025-07-17 前立腺特異的膜抗原(psma)リガンド及びその使用 Pending JP2025165975A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP19184015.6 2019-07-02
EP19184015 2019-07-02
JP2021578240A JP7805170B2 (ja) 2019-07-02 2020-06-30 前立腺特異的膜抗原(psma)リガンド及びその使用
PCT/EP2020/068386 WO2021001360A1 (en) 2019-07-02 2020-06-30 Prostate specific membrane antigen (psma) ligands and uses thereof

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2021578240A Division JP7805170B2 (ja) 2019-07-02 2020-06-30 前立腺特異的膜抗原(psma)リガンド及びその使用

Publications (2)

Publication Number Publication Date
JP2025165975A JP2025165975A (ja) 2025-11-05
JP2025165975A5 true JP2025165975A5 (https=) 2026-02-13

Family

ID=67145647

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021578240A Active JP7805170B2 (ja) 2019-07-02 2020-06-30 前立腺特異的膜抗原(psma)リガンド及びその使用
JP2025120662A Pending JP2025165975A (ja) 2019-07-02 2025-07-17 前立腺特異的膜抗原(psma)リガンド及びその使用

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2021578240A Active JP7805170B2 (ja) 2019-07-02 2020-06-30 前立腺特異的膜抗原(psma)リガンド及びその使用

Country Status (16)

Country Link
US (1) US20230226227A1 (https=)
EP (1) EP3993837A1 (https=)
JP (2) JP7805170B2 (https=)
KR (1) KR20220044496A (https=)
CN (3) CN120441497A (https=)
AR (1) AR119331A1 (https=)
AU (3) AU2020299974A1 (https=)
BR (1) BR112021026812A2 (https=)
CA (1) CA3144557A1 (https=)
CL (1) CL2021003525A1 (https=)
CO (1) CO2021017708A2 (https=)
IL (1) IL289039B1 (https=)
MX (1) MX2022000136A (https=)
PH (1) PH12021553284A1 (https=)
TW (1) TW202114742A (https=)
WO (1) WO2021001360A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20230330278A1 (en) * 2020-04-29 2023-10-19 Novartis Ag Methods for radiolabelling psma binding ligands and their kits
KR20260040237A (ko) 2023-07-21 2026-03-24 노파르티스 아게 Psma 표적 방사성 리간드 치료 요법
WO2025125469A1 (en) 2023-12-13 2025-06-19 Swiss Rockets Ag Combination therapy using psma-targeted radiopharmaceuticals and an inhibitor of pi3k, akt, and/or mtor

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2001271026A1 (en) 2000-07-11 2002-01-21 Bml, Inc. Remedies for bone diseases
WO2013022797A1 (en) * 2011-08-05 2013-02-14 Molecular Insight Pharmaceuticals Radiolabeled prostate specific membrane antigen inhibitors
LT4095130T (lt) * 2013-10-18 2024-04-25 Novartis Ag Žymėti prostatos specifinio membranos antigeno (psma) inhibitoriai, jų naudojimas kaip vizualizavimo medžiagų ir farmacinių medžiagų prostatos vėžiui gydyti
HRP20240215T1 (hr) * 2016-03-22 2024-04-26 The Johns Hopkins University Sredstva sa visokim afinitetom za ciljani učinak na membranski antigen specifičan za prostatu za endoradioterapiju raka prostate
WO2018222778A1 (en) * 2017-05-30 2018-12-06 The Johns Hopkins University Prostate-specific membrane antigen targeted high-affinity agents for endoradiotherapy of prostate cancer
KR20250126870A (ko) * 2018-02-06 2025-08-25 더 존스 홉킨스 유니버시티 암 방사선 치료를 위한 psma 표적 방사성 할로겐화 우레아-폴리아미노카복실레이트
WO2020028323A1 (en) * 2018-07-30 2020-02-06 The Johns Hopkins Universtiy Competitive prostate-specific membrane antigen (psma) binding agents for the reduction of non-target organ uptake of radiolabeled psma inhibitors for psma positive tumor imaging and radiopharmaceutical therapy

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