JP2023518161A5 - - Google Patents
Info
- Publication number
- JP2023518161A5 JP2023518161A5 JP2022549375A JP2022549375A JP2023518161A5 JP 2023518161 A5 JP2023518161 A5 JP 2023518161A5 JP 2022549375 A JP2022549375 A JP 2022549375A JP 2022549375 A JP2022549375 A JP 2022549375A JP 2023518161 A5 JP2023518161 A5 JP 2023518161A5
- Authority
- JP
- Japan
- Prior art keywords
- atoms
- group
- conjugate
- pharmaceutically acceptable
- polymorph
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP20162699.1 | 2020-03-12 | ||
| EP20162699 | 2020-03-12 | ||
| PCT/EP2021/056424 WO2021180969A1 (en) | 2020-03-12 | 2021-03-12 | Cyclic peptides and their conjugates for addressing alpha-v-beta-6 integrin in vivo |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023518161A JP2023518161A (ja) | 2023-04-28 |
| JP2023518161A5 true JP2023518161A5 (https=) | 2023-10-30 |
| JP7787083B2 JP7787083B2 (ja) | 2025-12-16 |
Family
ID=69810651
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022549375A Active JP7787083B2 (ja) | 2020-03-12 | 2021-03-12 | アルファ－ｖ－ベータ－６－インテグリンをインビボでアドレッシングするための環状ペプチド及びそれらのコンジュゲート |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20230173113A1 (https=) |
| EP (1) | EP4117736A1 (https=) |
| JP (1) | JP7787083B2 (https=) |
| KR (1) | KR20220152322A (https=) |
| CN (1) | CN115297893B (https=) |
| AU (1) | AU2021233176A1 (https=) |
| BR (1) | BR112022016986A2 (https=) |
| CA (1) | CA3175061A1 (https=) |
| IL (1) | IL296081A (https=) |
| MX (1) | MX2022011287A (https=) |
| WO (1) | WO2021180969A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2021226432A2 (en) * | 2020-05-08 | 2021-11-11 | The Regents Of The University Of California | Methods of detecting and treating lung damage in respiratory-related viral infections |
| WO2025218677A1 (zh) * | 2024-04-16 | 2025-10-23 | 中山医诺维申新药研发有限公司 | 双重靶向成纤维细胞激活蛋白和整合素亚型的化合物及其制备和应用 |
| WO2026027771A1 (en) | 2024-08-02 | 2026-02-05 | Trimt Gmbh | Alpha v beta 6-integrin binding cyclopeptides with non-natural amino acids, and conjugates thereof |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19933173A1 (de) | 1999-07-15 | 2001-01-18 | Merck Patent Gmbh | Cyclische Peptidderivate als Inhibitoren des Integrins alpha¶v¶beta¶6¶ |
| DK2265283T3 (da) | 2008-03-18 | 2014-10-20 | Seattle Genetics Inc | Auristatin-lægemiddel-linker-konjugater |
| CA2937753A1 (en) | 2014-02-17 | 2015-08-20 | Seattle Genetics, Inc. | Hydrophilic antibody-drug conjugates |
| SI3350222T1 (sl) | 2015-09-18 | 2022-01-31 | Technische Universitaet Muenchen | Ligandi za integrin avbeta6, sinteza in uporaba le-teh |
| EP3468984A4 (en) * | 2016-06-13 | 2020-03-11 | The Regents of the University of California | ALPHA (V) BETA (6) BINDING PEPTIDES AND METHODS OF USE THEREOF |
| CA3090196A1 (en) | 2018-02-06 | 2019-08-15 | Klinikum Rechts Der Isar Der Technischen Universitat Munchen | Compound for intraoperative molecular bioimaging, method of making the same, use thereof in intraoperative molecular bioimaging and surgical method comprising intraoperative molecular bioimaging |
-
2021
- 2021-03-12 WO PCT/EP2021/056424 patent/WO2021180969A1/en not_active Ceased
- 2021-03-12 EP EP21710520.4A patent/EP4117736A1/en active Pending
- 2021-03-12 BR BR112022016986A patent/BR112022016986A2/pt unknown
- 2021-03-12 JP JP2022549375A patent/JP7787083B2/ja active Active
- 2021-03-12 CA CA3175061A patent/CA3175061A1/en active Pending
- 2021-03-12 KR KR1020227035503A patent/KR20220152322A/ko active Pending
- 2021-03-12 MX MX2022011287A patent/MX2022011287A/es unknown
- 2021-03-12 US US17/910,728 patent/US20230173113A1/en active Pending
- 2021-03-12 CN CN202180020982.9A patent/CN115297893B/zh active Active
- 2021-03-12 AU AU2021233176A patent/AU2021233176A1/en active Pending
- 2021-03-12 IL IL296081A patent/IL296081A/en unknown
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