JP2025131625A5 - - Google Patents
Info
- Publication number
- JP2025131625A5 JP2025131625A5 JP2025083936A JP2025083936A JP2025131625A5 JP 2025131625 A5 JP2025131625 A5 JP 2025131625A5 JP 2025083936 A JP2025083936 A JP 2025083936A JP 2025083936 A JP2025083936 A JP 2025083936A JP 2025131625 A5 JP2025131625 A5 JP 2025131625A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- polymer
- solid dispersion
- amorphous solid
- pharmaceutical composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962832606P | 2019-04-11 | 2019-04-11 | |
| US62/832,606 | 2019-04-11 | ||
| PCT/US2020/027677 WO2020210629A1 (en) | 2019-04-11 | 2020-04-10 | Enhanced performance of amorphous solid and solubilized formulations for achieving therapeutic plasma concentrations |
| JP2021559853A JP2022526656A (ja) | 2019-04-11 | 2020-04-10 | 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021559853A Division JP2022526656A (ja) | 2019-04-11 | 2020-04-10 | 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025131625A JP2025131625A (ja) | 2025-09-09 |
| JP2025131625A5 true JP2025131625A5 (https=) | 2025-11-07 |
Family
ID=70465560
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021559853A Withdrawn JP2022526656A (ja) | 2019-04-11 | 2020-04-10 | 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能 |
| JP2025083936A Pending JP2025131625A (ja) | 2019-04-11 | 2025-05-20 | 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021559853A Withdrawn JP2022526656A (ja) | 2019-04-11 | 2020-04-10 | 治療血漿濃度に達するために増強された非晶質固体および溶解製剤の性能 |
Country Status (18)
| Country | Link |
|---|---|
| US (2) | US12509461B2 (https=) |
| EP (1) | EP3953355A1 (https=) |
| JP (2) | JP2022526656A (https=) |
| KR (1) | KR20210151183A (https=) |
| CN (1) | CN113924300A (https=) |
| AR (1) | AR118650A1 (https=) |
| AU (2) | AU2020271103B2 (https=) |
| BR (1) | BR112021020257A2 (https=) |
| CA (1) | CA3132530A1 (https=) |
| CL (1) | CL2021002627A1 (https=) |
| CO (1) | CO2021015054A2 (https=) |
| EA (1) | EA202192753A1 (https=) |
| IL (1) | IL287103A (https=) |
| MX (2) | MX2021012288A (https=) |
| PE (1) | PE20212367A1 (https=) |
| SG (1) | SG11202111131VA (https=) |
| TW (1) | TW202104228A (https=) |
| WO (1) | WO2020210629A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA3212644A1 (en) | 2021-03-09 | 2022-09-15 | Bayer Aktiengesellschaft | Pharmaceutical dosage forms comprising (4s)-24-chloro-4-ethyl-73-fluoro-35-methoxy-32,5- dioxo-14-(trifluoromethyl)-32h-6-aza-3(4,1)-pyridina-1(1)-[1,2,3]triazola-2(1,2),7(1)- dibenzenaheptaphane-74-carboxamide |
| IL310894A (en) | 2021-09-17 | 2024-04-01 | Bristol Myers Squibb Co | Milovacian for the prevention and treatment of thromboembolic disorders |
| MA71692A (fr) | 2022-08-01 | 2025-05-30 | Bristol-Myers Squibb Company | Utilisation de milvexian pour le traitement ou la prévention d'un accident vasculaire cérébral ischémique |
| KR20250136432A (ko) | 2023-02-06 | 2025-09-16 | 브리스톨-마이어스 스큅 컴퍼니 | 밀벡시안 제약 조성물 |
| WO2025099743A1 (en) * | 2023-11-07 | 2025-05-15 | Dr. Reddy’S Laboratories Limited | Process for preparation of milvexian and solid-state forms thereof |
| WO2025126240A1 (en) * | 2023-12-12 | 2025-06-19 | Dr. Reddy's Laboratories Limited | Pharmaceutical compositions and use thereof |
| WO2025220042A1 (en) * | 2024-04-18 | 2025-10-23 | Dr. Reddy's Laboratories Limited | Pharmaceutical compositions comprising asundexian and use thereof |
| WO2025224678A1 (en) | 2024-04-25 | 2025-10-30 | Assia Chemical Industries Ltd. | Solid state forms of milvexian and process for preparation thereof |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT83812B (en) | 1985-11-27 | 1988-03-15 | Syntex Inc | Process for preparing amorphous benzimidazole derivatives |
| ES2287971T3 (es) | 1997-08-11 | 2007-12-16 | Pfizer Products Inc. | Dispersiones farmaceuticas solidas con biodisponibilidad incrementada. |
| CN1402629A (zh) * | 1999-12-23 | 2003-03-12 | 辉瑞产品公司 | 提供提高的药物浓度的药物组合物 |
| CA2737400C (en) * | 2008-10-07 | 2016-11-22 | Astrazeneca Uk Limited | Pharmaceutical formulation 514 |
| WO2010102245A1 (en) | 2009-03-05 | 2010-09-10 | Upsher-Smith Laboratories, Inc. | Solid dispersion comprising resveratrol |
| MY172424A (en) * | 2009-04-03 | 2019-11-25 | Hoffmann La Roche | Propane- i-sulfonic acid {3- (4-chloro-phenyl)-1h-pyrrolo [2, 3-b] pyridine-3-carconyl] -2, 4-difluoro-phenyl} -amide compositions and uses thereof |
| SG10201908467RA (en) | 2014-01-31 | 2019-10-30 | Bristol Myers Squibb Co | Macrocycles with hetrocyclic p2' groups as factor xia inhibitors |
| PT107568B (pt) | 2014-03-31 | 2018-11-05 | Hovione Farm S A | Processo de secagem por atomização para a produção de pós com propriedades melhoradas. |
| NO2721243T3 (https=) | 2014-10-01 | 2018-10-20 | ||
| US9453018B2 (en) * | 2014-10-01 | 2016-09-27 | Bristol-Myers Squibb Company | Pyrimidinones as factor XIa inhibitors |
| JP6203702B2 (ja) | 2014-11-18 | 2017-09-27 | 信越化学工業株式会社 | ヒプロメロース酢酸エステルコハク酸エステルを用いたスプレードライ用溶液及び固体分散体の製造方法 |
| ES2791319T3 (es) | 2016-04-22 | 2020-11-03 | Astrazeneca Ab | Inhibidores de MCL1 macrocíclicos para tratar el cáncer |
-
2020
- 2020-04-10 BR BR112021020257A patent/BR112021020257A2/pt unknown
- 2020-04-10 TW TW109112257A patent/TW202104228A/zh unknown
- 2020-04-10 WO PCT/US2020/027677 patent/WO2020210629A1/en not_active Ceased
- 2020-04-10 JP JP2021559853A patent/JP2022526656A/ja not_active Withdrawn
- 2020-04-10 SG SG11202111131VA patent/SG11202111131VA/en unknown
- 2020-04-10 CA CA3132530A patent/CA3132530A1/en active Pending
- 2020-04-10 MX MX2021012288A patent/MX2021012288A/es unknown
- 2020-04-10 KR KR1020217036797A patent/KR20210151183A/ko not_active Ceased
- 2020-04-10 AU AU2020271103A patent/AU2020271103B2/en active Active
- 2020-04-10 CN CN202080041944.7A patent/CN113924300A/zh active Pending
- 2020-04-10 EP EP20722195.3A patent/EP3953355A1/en active Pending
- 2020-04-10 US US17/602,025 patent/US12509461B2/en active Active
- 2020-04-10 PE PE2021001691A patent/PE20212367A1/es unknown
- 2020-04-10 EA EA202192753A patent/EA202192753A1/ru unknown
- 2020-04-13 AR ARP200101025A patent/AR118650A1/es unknown
-
2021
- 2021-10-07 IL IL287103A patent/IL287103A/en unknown
- 2021-10-07 MX MX2025011559A patent/MX2025011559A/es unknown
- 2021-10-07 CL CL2021002627A patent/CL2021002627A1/es unknown
- 2021-11-08 CO CONC2021/0015054A patent/CO2021015054A2/es unknown
-
2025
- 2025-05-20 JP JP2025083936A patent/JP2025131625A/ja active Pending
- 2025-07-25 US US19/281,444 patent/US20260042761A1/en active Pending
- 2025-12-11 AU AU2025279715A patent/AU2025279715A1/en active Pending
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