JP2024540241A5 - - Google Patents

Info

Publication number
JP2024540241A5
JP2024540241A5 JP2024525932A JP2024525932A JP2024540241A5 JP 2024540241 A5 JP2024540241 A5 JP 2024540241A5 JP 2024525932 A JP2024525932 A JP 2024525932A JP 2024525932 A JP2024525932 A JP 2024525932A JP 2024540241 A5 JP2024540241 A5 JP 2024540241A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
compound
prodrug
solvate
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024525932A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024540241A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/078779 external-priority patent/WO2023076997A1/en
Publication of JP2024540241A publication Critical patent/JP2024540241A/ja
Publication of JP2024540241A5 publication Critical patent/JP2024540241A5/ja
Pending legal-status Critical Current

Links

JP2024525932A 2021-10-28 2022-10-27 治療上の使用のためのアンブロキソールの修飾形態 Pending JP2024540241A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163272743P 2021-10-28 2021-10-28
US63/272,743 2021-10-28
PCT/US2022/078779 WO2023076997A1 (en) 2021-10-28 2022-10-27 Modified forms of ambroxol for therapeutic use

Publications (2)

Publication Number Publication Date
JP2024540241A JP2024540241A (ja) 2024-10-31
JP2024540241A5 true JP2024540241A5 (enExample) 2025-11-04

Family

ID=84364209

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024525932A Pending JP2024540241A (ja) 2021-10-28 2022-10-27 治療上の使用のためのアンブロキソールの修飾形態

Country Status (7)

Country Link
US (1) US20250235413A1 (enExample)
EP (1) EP4423041A1 (enExample)
JP (1) JP2024540241A (enExample)
KR (1) KR20240095271A (enExample)
CN (1) CN118660866A (enExample)
CA (1) CA3235692A1 (enExample)
WO (1) WO2023076997A1 (enExample)

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5073543A (en) 1988-07-21 1991-12-17 G. D. Searle & Co. Controlled release formulations of trophic factors in ganglioside-lipsome vehicle
IT1229203B (it) 1989-03-22 1991-07-25 Bioresearch Spa Impiego di acido 5 metiltetraidrofolico, di acido 5 formiltetraidrofolico e dei loro sali farmaceuticamente accettabili per la preparazione di composizioni farmaceutiche in forma a rilascio controllato attive nella terapia dei disturbi mentali organici e composizioni farmaceutiche relative.
US5120548A (en) 1989-11-07 1992-06-09 Merck & Co., Inc. Swelling modulated polymeric drug delivery device
US5733566A (en) 1990-05-15 1998-03-31 Alkermes Controlled Therapeutics Inc. Ii Controlled release of antiparasitic agents in animals
US5580578A (en) 1992-01-27 1996-12-03 Euro-Celtique, S.A. Controlled release formulations coated with aqueous dispersions of acrylic polymers
US5591767A (en) 1993-01-25 1997-01-07 Pharmetrix Corporation Liquid reservoir transdermal patch for the administration of ketorolac
US5354566A (en) 1993-06-02 1994-10-11 Kraft General Foods, Inc. Preparation of yeast-leavened dough crusts
IT1270594B (it) 1994-07-07 1997-05-07 Recordati Chem Pharm Composizione farmaceutica a rilascio controllato di moguisteina in sospensione liquida
US6440710B1 (en) * 1998-12-10 2002-08-27 The Scripps Research Institute Antibody-catalyzed deuteration, tritiation, dedeuteration or detritiation of carbonyl compounds
DK1104760T3 (da) * 1999-12-03 2003-06-30 Pfizer Prod Inc Sulfamoylheteroarylpyrazolforbindelser som anti-inflammatoriske/analgetiske midler
IL160539A0 (en) 2001-09-04 2004-07-25 Boehringer Ingelheim Int Anti-influenzal agents
TW200413273A (en) * 2002-11-15 2004-08-01 Wako Pure Chem Ind Ltd Heavy hydrogenation method of heterocyclic rings
DE10332487A1 (de) 2003-07-16 2005-02-10 Boehringer Ingelheim Pharma Gmbh & Co. Kg Ambroxol für die Behandlung von chronisch nozizeptiven Schmerzen
US7750168B2 (en) * 2006-02-10 2010-07-06 Sigma-Aldrich Co. Stabilized deuteroborane-tetrahydrofuran complex
CA3055311A1 (en) * 2017-02-07 2018-08-16 Stc.Unm Isotope enhanced ambroxol for long lasting autophagy induction
CN114907221A (zh) * 2021-02-06 2022-08-16 华创合成制药股份有限公司 一种氘代氨溴索衍生物及其制备和用途

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