JP2024532845A5 - - Google Patents

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Publication number
JP2024532845A5
JP2024532845A5 JP2024510224A JP2024510224A JP2024532845A5 JP 2024532845 A5 JP2024532845 A5 JP 2024532845A5 JP 2024510224 A JP2024510224 A JP 2024510224A JP 2024510224 A JP2024510224 A JP 2024510224A JP 2024532845 A5 JP2024532845 A5 JP 2024532845A5
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JP
Japan
Prior art keywords
group
optionally substituted
substituted
cancer
alternatively
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024510224A
Other languages
English (en)
Japanese (ja)
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JP2024532845A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/CN2022/112674 external-priority patent/WO2023020457A1/en
Publication of JP2024532845A publication Critical patent/JP2024532845A/ja
Publication of JP2024532845A5 publication Critical patent/JP2024532845A5/ja
Pending legal-status Critical Current

Links

JP2024510224A 2021-08-17 2022-08-16 ピリダジノンまたはピリジノン化合物、その製造方法および用途 Pending JP2024532845A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN2021112906 2021-08-17
CNPCT/CN2021/112906 2021-08-17
PCT/CN2022/112674 WO2023020457A1 (en) 2021-08-17 2022-08-16 Pyridazinone or pyridinone compounds, preparation methods and uses thereof

Publications (2)

Publication Number Publication Date
JP2024532845A JP2024532845A (ja) 2024-09-10
JP2024532845A5 true JP2024532845A5 (https=) 2025-08-13

Family

ID=85240081

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024510224A Pending JP2024532845A (ja) 2021-08-17 2022-08-16 ピリダジノンまたはピリジノン化合物、その製造方法および用途

Country Status (5)

Country Link
US (1) US20240343727A1 (https=)
EP (1) EP4387966A4 (https=)
JP (1) JP2024532845A (https=)
CN (1) CN117897380A (https=)
WO (1) WO2023020457A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2022375782B2 (en) * 2021-10-28 2026-02-26 Gilead Sciences, Inc. Pyridizin-3(2h)-one derivatives
JP2025534359A (ja) * 2022-09-30 2025-10-15 アズカラ セラピューティクス インク ピリダジン-3(2h)-オンおよびピリジン-2(1h)-オンのPARP阻害化合物
GB202217888D0 (en) * 2022-11-29 2023-01-11 Duke Street Bio Ltd Pharmaceutical compound
TW202430518A (zh) * 2023-01-06 2024-08-01 大陸商齊魯製藥有限公司 Parp7抑制劑的製備方法
CN116874496B (zh) * 2023-07-10 2025-07-25 东南大学 三环类化合物及其制备方法、药物组合物和应用
CN117777099A (zh) * 2023-12-26 2024-03-29 诺沃斯达药业(上海)有限公司 Parp7抑制剂及其用途
CN118772063B (zh) * 2024-07-04 2025-06-13 西北师范大学 一种四氢哒嗪类化合物的合成方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19921567A1 (de) * 1999-05-11 2000-11-16 Basf Ag Verwendung von Phthalazine-Derivaten
GB0419072D0 (en) * 2004-08-26 2004-09-29 Kudos Pharm Ltd Phthalazinone derivatives
GB0610680D0 (en) * 2006-05-31 2006-07-12 Istituto Di Ricerche D Biolog Therapeutic compounds
UY31603A1 (es) * 2008-01-23 2009-08-31 Derivados de ftalazinona
CN103130723B (zh) * 2011-11-30 2015-01-14 成都地奥制药集团有限公司 一种多聚(adp-核糖)聚合酶抑制剂
JP7346425B2 (ja) * 2018-01-11 2023-09-19 セントラス セラピューティクス 疾患を治療するためのジヒドロセラミドデサチュラーゼ阻害剤
FI3788040T3 (fi) * 2018-04-30 2023-06-13 Ribon Therapeutics Inc Pyridatsinoneja parp7-inhibiittoreina
CA3113373A1 (en) * 2018-10-12 2020-04-16 InventisBio Co., Ltd. Thyroid hormone receptor agonists
US20240190844A1 (en) * 2019-10-30 2024-06-13 Ribon Therapeutics, Inc. Pyridazinones as parp7 inhibitors

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