JP2023520333A5 - - Google Patents

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Publication number
JP2023520333A5
JP2023520333A5 JP2022557856A JP2022557856A JP2023520333A5 JP 2023520333 A5 JP2023520333 A5 JP 2023520333A5 JP 2022557856 A JP2022557856 A JP 2022557856A JP 2022557856 A JP2022557856 A JP 2022557856A JP 2023520333 A5 JP2023520333 A5 JP 2023520333A5
Authority
JP
Japan
Prior art keywords
cancer
alkyl
inhibitor
pharmaceutical product
product according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022557856A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023520333A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/023752 external-priority patent/WO2021195128A1/en
Publication of JP2023520333A publication Critical patent/JP2023520333A/ja
Publication of JP2023520333A5 publication Critical patent/JP2023520333A5/ja
Pending legal-status Critical Current

Links

JP2022557856A 2020-03-24 2021-03-23 Eif4a阻害剤組み合わせ Pending JP2023520333A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062993889P 2020-03-24 2020-03-24
US62/993,889 2020-03-24
PCT/US2021/023752 WO2021195128A1 (en) 2020-03-24 2021-03-23 Eif4a inhibitor combinations

Publications (2)

Publication Number Publication Date
JP2023520333A JP2023520333A (ja) 2023-05-17
JP2023520333A5 true JP2023520333A5 (https=) 2024-04-03

Family

ID=77855108

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022557856A Pending JP2023520333A (ja) 2020-03-24 2021-03-23 Eif4a阻害剤組み合わせ

Country Status (8)

Country Link
US (1) US20210299111A1 (https=)
EP (1) EP4125884A4 (https=)
JP (1) JP2023520333A (https=)
KR (1) KR20230005175A (https=)
CN (1) CN115996716A (https=)
AU (1) AU2021244462A1 (https=)
CA (1) CA3176264A1 (https=)
WO (1) WO2021195128A1 (https=)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4395775A1 (en) 2021-09-01 2024-07-10 KHR Biotec GmbH Cyclopenta[4,5]furo[3,2-c]pyridine derivatives as ras inhibitors for use in the treatment of hyperproliferative diseases or genetic disorders
TW202508595A (zh) 2023-05-04 2025-03-01 美商銳新醫藥公司 用於ras相關疾病或病症之組合療法
WO2024254195A1 (en) * 2023-06-06 2024-12-12 Baylor University Methods for treating pancreatic cancer with a combination of des-methyl pateamine a and a class 1 hdac inhibitor
US20250049810A1 (en) 2023-08-07 2025-02-13 Revolution Medicines, Inc. Methods of treating a ras protein-related disease or disorder
AU2024360465A1 (en) 2023-10-12 2026-04-09 Revolution Medicines, Inc. Macrocyclic ras inhibitors
WO2025171296A1 (en) 2024-02-09 2025-08-14 Revolution Medicines, Inc. Ras inhibitors
TW202547461A (zh) 2024-05-17 2025-12-16 美商銳新醫藥公司 Ras抑制劑
WO2025255438A1 (en) 2024-06-07 2025-12-11 Revolution Medicines, Inc. Methods of treating a ras protein-related disease or disorder
WO2025265060A1 (en) 2024-06-21 2025-12-26 Revolution Medicines, Inc. Therapeutic compositions and methods for managing treatment-related effects
WO2026006747A1 (en) 2024-06-28 2026-01-02 Revolution Medicines, Inc. Ras inhibitors
WO2026015801A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2026015790A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2026015796A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2026015825A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Use of ras inhibitor for treating pancreatic cancer
WO2026050446A1 (en) 2024-08-29 2026-03-05 Revolution Medicines, Inc. Ras inhibitors
WO2026072904A2 (en) 2024-09-26 2026-04-02 Revolution Medicines, Inc. Compositions and methods for treating lung cancer
CN119351519B (zh) * 2024-10-21 2025-08-01 吉林大学 一种靶向隐孢子虫解旋酶的抗隐孢子虫小分子先导化合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102011111400A1 (de) * 2011-08-23 2013-02-28 Merck Patent Gmbh Bicyclische heteroaromatische Verbindungen
EP3191098A4 (en) * 2014-09-12 2018-04-25 G1 Therapeutics, Inc. Combinations and dosing regimes to treat rb-positive tumors
DK3888658T3 (da) * 2015-11-25 2024-03-18 Effector Therapeutics Inc Eif4-a-inhiberende forbindelser og fremgangsmåder relateret dertil
CA3063563A1 (en) * 2017-05-24 2018-11-29 Effector Therapeutics, Inc. Compositions and methods for an improved antitumor immune response

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