JP2024529307A5 - - Google Patents

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Publication number
JP2024529307A5
JP2024529307A5 JP2024500469A JP2024500469A JP2024529307A5 JP 2024529307 A5 JP2024529307 A5 JP 2024529307A5 JP 2024500469 A JP2024500469 A JP 2024500469A JP 2024500469 A JP2024500469 A JP 2024500469A JP 2024529307 A5 JP2024529307 A5 JP 2024529307A5
Authority
JP
Japan
Prior art keywords
cancer
acid
conjugate according
alkyl
sifa
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024500469A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024529307A (ja
Filing date
Publication date
Priority claimed from GBGB2109922.1A external-priority patent/GB202109922D0/en
Application filed filed Critical
Publication of JP2024529307A publication Critical patent/JP2024529307A/ja
Publication of JP2024529307A5 publication Critical patent/JP2024529307A5/ja
Pending legal-status Critical Current

Links

JP2024500469A 2021-07-09 2022-07-08 線維芽細胞活性化タンパク質(fap)に結合する放射性トレーサーおよび治療薬 Pending JP2024529307A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB2109922.1 2021-07-09
GBGB2109922.1A GB202109922D0 (en) 2021-07-09 2021-07-09 Radiotracers and therapeutics binding to fibroblast activation protein (fap)
PCT/US2022/073544 WO2023283627A1 (en) 2021-07-09 2022-07-08 Radiotracers and therapeutics binding to fibroblast activation protein (fap)

Publications (2)

Publication Number Publication Date
JP2024529307A JP2024529307A (ja) 2024-08-06
JP2024529307A5 true JP2024529307A5 (enExample) 2025-06-11

Family

ID=77353994

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024500469A Pending JP2024529307A (ja) 2021-07-09 2022-07-08 線維芽細胞活性化タンパク質(fap)に結合する放射性トレーサーおよび治療薬

Country Status (7)

Country Link
US (1) US20240399001A1 (enExample)
EP (1) EP4366786A1 (enExample)
JP (1) JP2024529307A (enExample)
KR (1) KR20240035488A (enExample)
CN (1) CN117836013A (enExample)
GB (1) GB202109922D0 (enExample)
WO (1) WO2023283627A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2024152775A1 (zh) * 2023-01-17 2024-07-25 云合智药(苏州)生物科技有限公司 缀合物、配体单元及其用途
WO2024227137A1 (en) * 2023-04-28 2024-10-31 The Board Of Regents Of The University Of Texas System Structurally-reinforced stable theranostic copper radiopharmaceuticals targeting fibroblast activation protein for cancer diagnosis and therapy
WO2025106926A1 (en) * 2023-11-16 2025-05-22 Praxis Biotech LLC Conjugates targeting fibroblast activation protein and uses thereof
WO2026041109A1 (zh) * 2024-08-23 2026-02-26 苏州博锐创合医药有限公司 成纤维细胞活化蛋白抑制剂及其用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116474108A (zh) 2016-12-14 2023-07-25 普渡研究基金会 成纤维细胞活化蛋白(fap)-靶向成像和治疗
HUE070098T2 (hu) 2017-07-28 2025-05-28 Univ Muenchen Tech Kettõs módusú radioaktív jelzõ és terapeutikumok
EA202090776A1 (ru) 2017-10-23 2020-07-27 Дзе Джонс Хопкинс Юниверсити Визуализирующие и радиотерапевтические агенты, нацеленные на фибробласт-активирующий белок-альфа (fapalpha)
EP3749663A1 (en) 2018-02-06 2020-12-16 Universität Heidelberg Fap inhibitor
CA3128406A1 (en) 2019-01-30 2020-08-06 Technische Universitat Munchen Cancer diagnostic imaging agents
EA202191691A1 (ru) 2019-01-30 2021-11-01 Технише Универзитет Мюнхен Радиоактивная метка, связывающая psma двумя способами, и терапевтическое средство
JP7801207B2 (ja) 2019-07-08 2026-01-16 3ベー ファーマシューティカルズ ゲーエムベーハー 線維芽細胞活性化タンパク質リガンドを含む化合物およびその使用
FI3997103T3 (fi) 2019-07-08 2025-02-03 3B Pharmaceuticals Gmbh Fibroblastien aktivaatioproteiinin ligandia käsittäviä yhdisteitä ja niiden käyttö

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