JP2024523506A5 - - Google Patents

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Publication number
JP2024523506A5
JP2024523506A5 JP2023579154A JP2023579154A JP2024523506A5 JP 2024523506 A5 JP2024523506 A5 JP 2024523506A5 JP 2023579154 A JP2023579154 A JP 2023579154A JP 2023579154 A JP2023579154 A JP 2023579154A JP 2024523506 A5 JP2024523506 A5 JP 2024523506A5
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JP
Japan
Prior art keywords
compound
diffraction pattern
ray powder
powder diffraction
crystalline
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023579154A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024523506A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/034550 external-priority patent/WO2022271846A1/en
Publication of JP2024523506A publication Critical patent/JP2024523506A/ja
Publication of JP2024523506A5 publication Critical patent/JP2024523506A5/ja
Pending legal-status Critical Current

Links

JP2023579154A 2021-06-23 2022-06-22 上皮成長因子受容体阻害剤の塩及び結晶形態 Pending JP2024523506A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163214089P 2021-06-23 2021-06-23
US63/214,089 2021-06-23
PCT/US2022/034550 WO2022271846A1 (en) 2021-06-23 2022-06-22 Salt and crystal forms of an epidermal growth factor receptor inhibitor

Publications (2)

Publication Number Publication Date
JP2024523506A JP2024523506A (ja) 2024-06-28
JP2024523506A5 true JP2024523506A5 (enExample) 2025-06-30

Family

ID=82608408

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023579154A Pending JP2024523506A (ja) 2021-06-23 2022-06-22 上皮成長因子受容体阻害剤の塩及び結晶形態

Country Status (9)

Country Link
US (1) US20240293404A1 (enExample)
EP (1) EP4359400B1 (enExample)
JP (1) JP2024523506A (enExample)
CN (1) CN117836287A (enExample)
CA (1) CA3223859A1 (enExample)
ES (1) ES3042447T3 (enExample)
IL (1) IL309469A (enExample)
TW (1) TW202317543A (enExample)
WO (1) WO2022271846A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3213079A1 (en) 2021-04-13 2022-10-20 Kristin Lynne ANDREWS Amino-substituted heterocycles for treating cancers with egfr mutations
IL309447A (en) * 2021-06-23 2024-02-01 Blueprint Medicines Corp Pharmaceutical preparations of epidermal growth factor receptor inhibitor
CN116554150B (zh) * 2022-12-30 2025-12-19 苏州浦合医药科技有限公司 第四代egfr抑制剂

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI726968B (zh) * 2016-01-07 2021-05-11 開曼群島商Cs醫藥技術公司 Egfr酪胺酸激酶之臨床重要突變體之選擇性抑制劑
JP7752617B2 (ja) * 2019-12-23 2025-10-10 ブループリント メディシンズ コーポレイション Egfrの変異型の阻害剤
US20240058340A1 (en) * 2020-09-21 2024-02-22 The Regents Of The University Of California Compositions and methods for treating cancer
IL309447A (en) * 2021-06-23 2024-02-01 Blueprint Medicines Corp Pharmaceutical preparations of epidermal growth factor receptor inhibitor
CN117881670A (zh) * 2021-06-23 2024-04-12 缆图药品公司 制备egfr抑制剂的方法

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