JP2024521791A5 - - Google Patents

Info

Publication number
JP2024521791A5
JP2024521791A5 JP2023572825A JP2023572825A JP2024521791A5 JP 2024521791 A5 JP2024521791 A5 JP 2024521791A5 JP 2023572825 A JP2023572825 A JP 2023572825A JP 2023572825 A JP2023572825 A JP 2023572825A JP 2024521791 A5 JP2024521791 A5 JP 2024521791A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
egfr
cancer
composition according
mediated cancer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023572825A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024521791A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/031193 external-priority patent/WO2022251539A2/en
Publication of JP2024521791A publication Critical patent/JP2024521791A/ja
Publication of JP2024521791A5 publication Critical patent/JP2024521791A5/ja
Pending legal-status Critical Current

Links

JP2023572825A 2021-05-26 2022-05-26 脳又はcnsへの癌転移を治療するためのegfrデグレーダー Pending JP2024521791A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163193574P 2021-05-26 2021-05-26
US63/193,574 2021-05-26
US202163270488P 2021-10-21 2021-10-21
US63/270,488 2021-10-21
PCT/US2022/031193 WO2022251539A2 (en) 2021-05-26 2022-05-26 Egfr degraders to treat cancer metastasis to the brain or cns

Publications (2)

Publication Number Publication Date
JP2024521791A JP2024521791A (ja) 2024-06-04
JP2024521791A5 true JP2024521791A5 (https=) 2025-06-03

Family

ID=84230313

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023572825A Pending JP2024521791A (ja) 2021-05-26 2022-05-26 脳又はcnsへの癌転移を治療するためのegfrデグレーダー

Country Status (11)

Country Link
US (1) US20240158418A1 (https=)
EP (1) EP4347044A4 (https=)
JP (1) JP2024521791A (https=)
KR (1) KR20240019099A (https=)
AU (1) AU2022280070A1 (https=)
BR (1) BR112023024507A2 (https=)
CA (1) CA3174207A1 (https=)
IL (1) IL308182A (https=)
MX (1) MX2023014061A (https=)
TW (1) TW202313025A (https=)
WO (1) WO2022251539A2 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110769822A (zh) 2017-06-20 2020-02-07 C4医药公司 用于蛋白降解的n/o-连接的降解决定子和降解决定子体
EP4735452A2 (en) 2023-06-30 2026-05-06 Merck Patent GmbH Heterobifunctional compounds for the degradation of kras protein
EP4735438A2 (en) 2023-06-30 2026-05-06 Merck Patent GmbH Heterobifunctional compounds for the degradation of kras
CN117503737B (zh) * 2024-01-05 2024-04-16 成都金瑞基业生物科技有限公司 和厚朴酚在制备治疗脂肪肉瘤药物中的用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017164887A1 (en) * 2016-03-25 2017-09-28 OSI Pharmaceuticals, LLC Pulse dosing regimen and methods for treatment
PE20211388A1 (es) * 2018-06-29 2021-07-27 Hoffmann La Roche Compuestos
IL288522B2 (en) * 2019-06-21 2025-02-01 Hoffmann La Roche EGFR inhibitor for cancer treatment
KR20220119415A (ko) * 2019-12-20 2022-08-29 씨4 테라퓨틱스, 인코포레이티드 Egfr 분해를 위한 이소인돌리논 및 인다졸 화합물

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