JP2024503235A5 - - Google Patents

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Publication number
JP2024503235A5
JP2024503235A5 JP2023537491A JP2023537491A JP2024503235A5 JP 2024503235 A5 JP2024503235 A5 JP 2024503235A5 JP 2023537491 A JP2023537491 A JP 2023537491A JP 2023537491 A JP2023537491 A JP 2023537491A JP 2024503235 A5 JP2024503235 A5 JP 2024503235A5
Authority
JP
Japan
Prior art keywords
cancer
ppm
crystal according
values
cukα radiation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023537491A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024503235A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2021/062082 external-priority patent/WO2022137106A1/en
Publication of JP2024503235A publication Critical patent/JP2024503235A/ja
Publication of JP2024503235A5 publication Critical patent/JP2024503235A5/ja
Priority to JP2026067895A priority Critical patent/JP2026123057A/ja
Pending legal-status Critical Current

Links

JP2023537491A 2020-12-24 2021-12-21 Cdk2阻害剤の固体形態 Pending JP2024503235A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2026067895A JP2026123057A (ja) 2020-12-24 2026-04-16 Cdk2阻害剤の固体形態

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063130530P 2020-12-24 2020-12-24
US63/130,530 2020-12-24
PCT/IB2021/062082 WO2022137106A1 (en) 2020-12-24 2021-12-21 Solid forms of a cdk2 inhibitor

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2026067895A Division JP2026123057A (ja) 2020-12-24 2026-04-16 Cdk2阻害剤の固体形態

Publications (2)

Publication Number Publication Date
JP2024503235A JP2024503235A (ja) 2024-01-25
JP2024503235A5 true JP2024503235A5 (enExample) 2024-11-28

Family

ID=79283019

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2023537491A Pending JP2024503235A (ja) 2020-12-24 2021-12-21 Cdk2阻害剤の固体形態
JP2026067895A Pending JP2026123057A (ja) 2020-12-24 2026-04-16 Cdk2阻害剤の固体形態

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2026067895A Pending JP2026123057A (ja) 2020-12-24 2026-04-16 Cdk2阻害剤の固体形態

Country Status (10)

Country Link
US (1) US20240076287A1 (enExample)
EP (1) EP4267563A1 (enExample)
JP (2) JP2024503235A (enExample)
KR (1) KR20230122100A (enExample)
CN (1) CN116723837B (enExample)
AU (1) AU2021404974B2 (enExample)
CA (1) CA3206153A1 (enExample)
MX (1) MX2023007699A (enExample)
TW (1) TWI823213B (enExample)
WO (1) WO2022137106A1 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3217792A1 (en) 2021-05-07 2022-11-10 Kymera Therapeutics, Inc Cdk2 degraders and uses thereof
US20250127759A1 (en) * 2021-12-02 2025-04-24 Pfizer Inc. Methods and dosing regimens comprising a cdk2 inhibitor for the treatment of cancer
CN118679150A (zh) * 2022-01-27 2024-09-20 益方生物科技(上海)股份有限公司 Cdk2抑制剂及其制备方法和用途
WO2024046443A1 (en) * 2022-09-01 2024-03-07 Nutshell Biotech (Shanghai) Co., Ltd. Macrocyclic compounds as selective cdk inhibitors
WO2025191482A1 (en) 2024-03-15 2025-09-18 Pfizer Inc. Synthesis of (1h-pyrazol-5-yl)cyclopentyl carbamate compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9518953D0 (en) 1995-09-15 1995-11-15 Pfizer Ltd Pharmaceutical formulations
WO2000035298A1 (en) 1996-11-27 2000-06-22 Wm. Wrigley Jr. Company Chewing gum containing medicament active agents
CA3128155C (en) * 2019-01-31 2023-09-19 Pfizer Inc. 3-carbonylamino-5-cyclopentyl-1h-pyrazole compounds having inhibitory activity on cdk2

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