JP2024150466A5 - - Google Patents

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Publication number
JP2024150466A5
JP2024150466A5 JP2024103249A JP2024103249A JP2024150466A5 JP 2024150466 A5 JP2024150466 A5 JP 2024150466A5 JP 2024103249 A JP2024103249 A JP 2024103249A JP 2024103249 A JP2024103249 A JP 2024103249A JP 2024150466 A5 JP2024150466 A5 JP 2024150466A5
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JP
Japan
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invention described
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JP2024103249A
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English (en)
Japanese (ja)
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JP2024150466A (ja
JP7789850B2 (ja
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Priority claimed from PCT/IB2021/054225 external-priority patent/WO2021234544A1/en
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Publication of JP2024150466A publication Critical patent/JP2024150466A/ja
Publication of JP2024150466A5 publication Critical patent/JP2024150466A5/ja
Priority to JP2025244399A priority Critical patent/JP2026048795A/ja
Application granted granted Critical
Publication of JP7789850B2 publication Critical patent/JP7789850B2/ja
Active legal-status Critical Current
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JP2024103249A 2020-05-18 2024-06-26 Lnp023の結晶形態 Active JP7789850B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025244399A JP2026048795A (ja) 2020-05-18 2025-12-10 Lnp023の結晶形態

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US202063026637P 2020-05-18 2020-05-18
US63/026,637 2020-05-18
US202063052699P 2020-07-16 2020-07-16
US63/052,699 2020-07-16
PCT/IB2021/054225 WO2021234544A1 (en) 2020-05-18 2021-05-17 Crystalline form of lnp023
JP2022557633A JP7592743B2 (ja) 2020-05-18 2021-05-17 Lnp023の結晶形態

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2022557633A Division JP7592743B2 (ja) 2020-05-18 2021-05-17 Lnp023の結晶形態

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025244399A Division JP2026048795A (ja) 2020-05-18 2025-12-10 Lnp023の結晶形態

Publications (3)

Publication Number Publication Date
JP2024150466A JP2024150466A (ja) 2024-10-23
JP2024150466A5 true JP2024150466A5 (https=) 2025-04-07
JP7789850B2 JP7789850B2 (ja) 2025-12-22

Family

ID=76076387

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2022557633A Active JP7592743B2 (ja) 2020-05-18 2021-05-17 Lnp023の結晶形態
JP2024103249A Active JP7789850B2 (ja) 2020-05-18 2024-06-26 Lnp023の結晶形態
JP2025244399A Pending JP2026048795A (ja) 2020-05-18 2025-12-10 Lnp023の結晶形態

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2022557633A Active JP7592743B2 (ja) 2020-05-18 2021-05-17 Lnp023の結晶形態

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025244399A Pending JP2026048795A (ja) 2020-05-18 2025-12-10 Lnp023の結晶形態

Country Status (10)

Country Link
US (3) US11603363B2 (https=)
EP (1) EP4153580A1 (https=)
JP (3) JP7592743B2 (https=)
KR (2) KR20230009478A (https=)
CN (4) CN120168469A (https=)
AU (2) AU2021276912B2 (https=)
CA (1) CA3180829A1 (https=)
IL (1) IL297975A (https=)
TW (2) TW202504893A (https=)
WO (1) WO2021234544A1 (https=)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI3675854T1 (sl) 2017-08-31 2025-05-30 Novartis Ag Derivati piperidinil-indola za uporabo v zdravljenju glomerulopatije c3
TW202504893A (zh) * 2020-05-18 2025-02-01 瑞士商諾華公司 Lnp023之結晶形式
US11951101B2 (en) 2020-07-16 2024-04-09 Novartis Ag Methods of using factor B inhibitors
WO2022143940A1 (zh) * 2020-12-30 2022-07-07 南京明德新药研发有限公司 一系列哌啶取代的苯酸类化合物及其应用
EP4333845A1 (en) * 2021-05-07 2024-03-13 Novartis AG Iptacopan for the treatment of atypical hemolytic uremic syndrome
WO2022264101A1 (en) 2021-06-18 2022-12-22 Novartis Ag Method of treating an autoimmune hematological disorder
CA3248808A1 (en) 2022-03-04 2023-09-07 Novartis Ag USE OF IPTACOPAN FOR THE TREATMENT OF LUPUS NEPHROPATHY
JP7849520B2 (ja) * 2022-06-30 2026-04-21 江▲蘇▼恒瑞医▲薬▼股▲フン▼有限公司 含窒素架橋複素環誘導体の薬学的に許容される塩、結晶形及びその調製方法
EP4669321A1 (en) 2023-02-23 2025-12-31 Novartis AG METHODS OF USING FACTOR B INHIBITORS
CN121712505A (zh) 2023-08-25 2026-03-20 诺华股份有限公司 使用因子b抑制剂的方法
WO2025148628A1 (zh) * 2024-01-10 2025-07-17 河北以岭医药研究院有限公司 哌啶基吲哚衍生物及其制备方法和应用
WO2025172910A1 (en) 2024-02-16 2025-08-21 Novartis Ag Factor b inhibitors for treatment of anca-associated vasculitis
WO2026003809A1 (en) * 2024-06-29 2026-01-02 Assia Chemical Industries Ltd. Solid state forms of iptacopan hydrochloride

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0301259D0 (en) 2003-01-20 2003-02-19 Novartis Ag Organic compounds
KR20130086534A (ko) 2010-06-01 2013-08-02 플러스 케미칼스, 에스.에이. 익사베필론의 고체 형태
JO3425B1 (ar) 2013-07-15 2019-10-20 Novartis Ag مشتقات البابيريدينيل-اندول واستخدامها كعامل متمم لمثبطات b
MX2018007392A (es) 2015-12-23 2018-08-15 Greenovation Biotech Gmbh Polipeptidos para inhibir la activacion del complemento.
SI3675854T1 (sl) 2017-08-31 2025-05-30 Novartis Ag Derivati piperidinil-indola za uporabo v zdravljenju glomerulopatije c3
TW202504893A (zh) * 2020-05-18 2025-02-01 瑞士商諾華公司 Lnp023之結晶形式

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