JP2024120882A5 - - Google Patents
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- Publication number
- JP2024120882A5 JP2024120882A5 JP2024025063A JP2024025063A JP2024120882A5 JP 2024120882 A5 JP2024120882 A5 JP 2024120882A5 JP 2024025063 A JP2024025063 A JP 2024025063A JP 2024025063 A JP2024025063 A JP 2024025063A JP 2024120882 A5 JP2024120882 A5 JP 2024120882A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- pharma
- acceptable salt
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025143871A JP2025176085A (ja) | 2023-02-24 | 2025-08-29 | 置換ピラゾロピリミジン化合物及びその医薬用途 |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023027432 | 2023-02-24 | ||
| JP2023027432 | 2023-02-24 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025143871A Division JP2025176085A (ja) | 2023-02-24 | 2025-08-29 | 置換ピラゾロピリミジン化合物及びその医薬用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2024120882A JP2024120882A (ja) | 2024-09-05 |
| JP2024120882A5 true JP2024120882A5 (https=) | 2025-05-26 |
| JP7737490B2 JP7737490B2 (ja) | 2025-09-10 |
Family
ID=92501386
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024025063A Active JP7737490B2 (ja) | 2023-02-24 | 2024-02-22 | 置換ピラゾロピリミジン化合物及びその医薬用途 |
| JP2025143871A Pending JP2025176085A (ja) | 2023-02-24 | 2025-08-29 | 置換ピラゾロピリミジン化合物及びその医薬用途 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025143871A Pending JP2025176085A (ja) | 2023-02-24 | 2025-08-29 | 置換ピラゾロピリミジン化合物及びその医薬用途 |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP4671247A1 (https=) |
| JP (2) | JP7737490B2 (https=) |
| KR (1) | KR20250151389A (https=) |
| CN (1) | CN120752239A (https=) |
| AR (1) | AR131919A1 (https=) |
| AU (1) | AU2024226032A1 (https=) |
| CL (1) | CL2025002505A1 (https=) |
| CO (1) | CO2025011311A2 (https=) |
| IL (1) | IL322520A (https=) |
| MX (1) | MX2025009965A (https=) |
| PE (1) | PE20252572A1 (https=) |
| TW (1) | TW202448887A (https=) |
| WO (1) | WO2024177127A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN120230110A (zh) * | 2023-12-31 | 2025-07-01 | 杭州百新生物医药科技有限公司 | 吡唑并嘧啶类化合物及其医药用途 |
| WO2025153532A1 (en) | 2024-01-16 | 2025-07-24 | NodThera Limited | Nlrp3 inhibitors and glp-1 agonists combination therapies |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10005781B2 (en) * | 2013-10-30 | 2018-06-26 | Shanghai Hengrui Pharmaceutical Co., Ltd. | Pyrazolopyrimidone or pyrrolotriazone derivatives, method of preparing same, and pharmaceutical applications thereof |
| WO2017205766A1 (en) * | 2016-05-27 | 2017-11-30 | Pharmacyclics Llc | Inhibitors of interleukin-1 receptor-associated kinase |
| ES2930151T3 (es) * | 2019-01-14 | 2022-12-07 | Innate Tumor Immunity Inc | Moduladores heterocíclicos de NLRP3, para su uso en el tratamiento del cáncer |
| EP3911641A1 (en) * | 2019-01-14 | 2021-11-24 | Innate Tumor Immunity, Inc. | Nlrp3 modulators |
| US20230399319A1 (en) * | 2019-12-27 | 2023-12-14 | Japan Tobacco Inc. | Acylsulfamide Compound and Pharmaceutical Use Therefor |
| US20240382488A1 (en) * | 2021-03-29 | 2024-11-21 | Halia Therapeutics, Inc. | Nek7 inhibitors |
| JP2024513227A (ja) * | 2021-04-05 | 2024-03-22 | ハリア・セラピューティクス・インコーポレイテッド | Nek7阻害剤 |
| WO2023032987A1 (ja) * | 2021-08-31 | 2023-03-09 | 日本たばこ産業株式会社 | 6-アミノピラゾロピリミジン化合物及びその医薬用途 |
| AR130318A1 (es) * | 2022-08-29 | 2024-11-27 | Japan Tobacco Inc | Compuestos de pirazolopirimidina y su uso médico |
| EP4694980A1 (en) * | 2023-04-14 | 2026-02-18 | Takeda Pharmaceutical Company Limited | Pyrazolopyrimidine derivatives as inhibitors of nlrp3 |
-
2024
- 2024-02-22 WO PCT/JP2024/006433 patent/WO2024177127A1/ja not_active Ceased
- 2024-02-22 EP EP24760425.9A patent/EP4671247A1/en active Pending
- 2024-02-22 KR KR1020257027024A patent/KR20250151389A/ko active Pending
- 2024-02-22 CN CN202480014319.1A patent/CN120752239A/zh active Pending
- 2024-02-22 AU AU2024226032A patent/AU2024226032A1/en active Pending
- 2024-02-22 TW TW113106397A patent/TW202448887A/zh unknown
- 2024-02-22 JP JP2024025063A patent/JP7737490B2/ja active Active
- 2024-02-22 PE PE2025001836A patent/PE20252572A1/es unknown
- 2024-02-22 IL IL322520A patent/IL322520A/en unknown
- 2024-02-22 AR ARP240100407A patent/AR131919A1/es unknown
-
2025
- 2025-08-20 CL CL2025002505A patent/CL2025002505A1/es unknown
- 2025-08-21 CO CONC2025/0011311A patent/CO2025011311A2/es unknown
- 2025-08-22 MX MX2025009965A patent/MX2025009965A/es unknown
- 2025-08-29 JP JP2025143871A patent/JP2025176085A/ja active Pending
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