JP2024052694A5 - - Google Patents
Info
- Publication number
- JP2024052694A5 JP2024052694A5 JP2024011686A JP2024011686A JP2024052694A5 JP 2024052694 A5 JP2024052694 A5 JP 2024052694A5 JP 2024011686 A JP2024011686 A JP 2024011686A JP 2024011686 A JP2024011686 A JP 2024011686A JP 2024052694 A5 JP2024052694 A5 JP 2024052694A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- ester
- peptide
- solvent
- amino acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021214900 | 2021-12-28 | ||
| JP2021214900 | 2021-12-28 | ||
| JP2022168608 | 2022-10-20 | ||
| JP2022168608 | 2022-10-20 | ||
| JP2023568520A JP7430297B2 (ja) | 2021-12-28 | 2022-12-27 | Ｎ－アルキルアミノ酸、およびｎ－アルキルアミノ酸を含むペプチドの製造方法 |
| PCT/JP2022/048135 WO2023127869A1 (ja) | 2021-12-28 | 2022-12-27 | Ｎ－アルキルアミノ酸、およびｎ－アルキルアミノ酸を含むペプチドの製造方法 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023568520A Division JP7430297B2 (ja) | 2021-12-28 | 2022-12-27 | Ｎ－アルキルアミノ酸、およびｎ－アルキルアミノ酸を含むペプチドの製造方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024052694A JP2024052694A (ja) | 2024-04-11 |
| JP2024052694A5 true JP2024052694A5 (https=) | 2026-01-09 |
Family
ID=86999039
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023568520A Active JP7430297B2 (ja) | 2021-12-28 | 2022-12-27 | Ｎ－アルキルアミノ酸、およびｎ－アルキルアミノ酸を含むペプチドの製造方法 |
| JP2024011686A Pending JP2024052694A (ja) | 2021-12-28 | 2024-01-30 | Ｎ－アルキルアミノ酸、およびｎ－アルキルアミノ酸を含むペプチドの製造方法 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023568520A Active JP7430297B2 (ja) | 2021-12-28 | 2022-12-27 | Ｎ－アルキルアミノ酸、およびｎ－アルキルアミノ酸を含むペプチドの製造方法 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20250197450A1 (https=) |
| EP (1) | EP4414374A4 (https=) |
| JP (2) | JP7430297B2 (https=) |
| KR (1) | KR102844018B1 (https=) |
| AR (1) | AR128119A1 (https=) |
| AU (1) | AU2022428318A1 (https=) |
| CA (1) | CA3237911A1 (https=) |
| IL (1) | IL312468A (https=) |
| MX (1) | MX2024008002A (https=) |
| TW (1) | TW202342495A (https=) |
| WO (1) | WO2023127869A1 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202446781A (zh) | 2011-12-28 | 2024-12-01 | 日商中外製藥股份有限公司 | 胜肽化合物之製造方法 |
| KR20250007021A (ko) | 2017-06-09 | 2025-01-13 | 추가이 세이야쿠 가부시키가이샤 | N-치환 아미노산을 포함하는 펩타이드의 합성 방법 |
| EP3878836B1 (en) | 2018-11-07 | 2025-07-23 | Chugai Seiyaku Kabushiki Kaisha | O-substituted serine derivative production method |
| BR112022007535A2 (pt) | 2019-11-07 | 2022-07-12 | Chugai Pharmaceutical Co Ltd | Composto peptídico cíclico tendo ação inibitória de kras |
| US12312379B2 (en) | 2021-05-07 | 2025-05-27 | Chugai Seiyaku Kabushiki Kaisha | Methods for producing cyclic compounds comprising N-substituted amino acid residues |
| JP7823181B2 (ja) | 2022-05-06 | 2026-03-03 | 中外製薬株式会社 | Ｈｒａｓおよびｎｒａｓに対して選択的なｋｒａｓ阻害作用を有する環状化合物 |
| JPWO2024096023A1 (https=) | 2022-11-01 | 2024-05-10 | ||
| WO2024143514A1 (ja) | 2022-12-28 | 2024-07-04 | 中外製薬株式会社 | 環状ペプチドの精製法及び製造法 |
| TW202523345A (zh) | 2023-09-28 | 2025-06-16 | 日商中外製藥股份有限公司 | 使用混合酸酐法的胜肽化合物的製造方法 |
| TW202535901A (zh) | 2023-12-27 | 2025-09-16 | 日商中外製藥股份有限公司 | 使用獨立型縮合劑的胜肽化合物的製造方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL1010063C2 (nl) | 1998-09-10 | 2000-03-13 | Holland Sweetener Co | Werkwijze voor de bereiding van neotaam. |
| CN110869544B (zh) | 2017-06-09 | 2024-03-08 | 中外制药株式会社 | 膜透过性高的环状肽化合物及包含其的文库 |
| KR20250007021A (ko) * | 2017-06-09 | 2025-01-13 | 추가이 세이야쿠 가부시키가이샤 | N-치환 아미노산을 포함하는 펩타이드의 합성 방법 |
| WO2020111238A1 (ja) * | 2018-11-30 | 2020-06-04 | 中外製薬株式会社 | ペプチド化合物、またはアミド化合物の脱保護法および固相反応における脱樹脂方法、並びにペプチド化合物の製造方法 |
| WO2020122182A1 (ja) | 2018-12-12 | 2020-06-18 | 中外製薬株式会社 | 分子内水素結合可能な官能基を有するアミノ酸とそれらのアミノ酸を含むペプチド化合物、およびそれらの製造方法 |
| EP3939962A4 (en) | 2019-03-15 | 2022-12-28 | Chugai Seiyaku Kabushiki Kaisha | PROCESS FOR PREPARING AN AROMATIC AMINO ACID DERIVATIVE |
| BR112022007535A2 (pt) * | 2019-11-07 | 2022-07-12 | Chugai Pharmaceutical Co Ltd | Composto peptídico cíclico tendo ação inibitória de kras |
-
2022
- 2022-12-27 TW TW111150100A patent/TW202342495A/zh unknown
- 2022-12-27 CA CA3237911A patent/CA3237911A1/en active Pending
- 2022-12-27 JP JP2023568520A patent/JP7430297B2/ja active Active
- 2022-12-27 MX MX2024008002A patent/MX2024008002A/es unknown
- 2022-12-27 AU AU2022428318A patent/AU2022428318A1/en active Pending
- 2022-12-27 IL IL312468A patent/IL312468A/en unknown
- 2022-12-27 KR KR1020247023000A patent/KR102844018B1/ko active Active
- 2022-12-27 US US18/723,993 patent/US20250197450A1/en active Pending
- 2022-12-27 WO PCT/JP2022/048135 patent/WO2023127869A1/ja not_active Ceased
- 2022-12-27 EP EP22916092.4A patent/EP4414374A4/en active Pending
- 2022-12-27 AR ARP220103601A patent/AR128119A1/es unknown
-
2024
- 2024-01-30 JP JP2024011686A patent/JP2024052694A/ja active Pending
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