JP2023528859A5 - - Google Patents

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Publication number
JP2023528859A5
JP2023528859A5 JP2022574270A JP2022574270A JP2023528859A5 JP 2023528859 A5 JP2023528859 A5 JP 2023528859A5 JP 2022574270 A JP2022574270 A JP 2022574270A JP 2022574270 A JP2022574270 A JP 2022574270A JP 2023528859 A5 JP2023528859 A5 JP 2023528859A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
solvate
isomer
hydrate
modulating
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022574270A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023528859A (ja
JP7777544B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2021/097583 external-priority patent/WO2021244505A1/zh
Publication of JP2023528859A publication Critical patent/JP2023528859A/ja
Publication of JP2023528859A5 publication Critical patent/JP2023528859A5/ja
Application granted granted Critical
Publication of JP7777544B2 publication Critical patent/JP7777544B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022574270A 2020-06-01 2021-06-01 新規ピラジン化合物 Active JP7777544B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
CN202010486394.1 2020-06-01
CN202010486394 2020-06-01
CN202010947590 2020-09-10
CN202010947590.4 2020-09-10
CN202110587528.3 2021-05-27
CN202110587528 2021-05-27
PCT/CN2021/097583 WO2021244505A1 (zh) 2020-06-01 2021-06-01 新型吡嗪化合物

Publications (3)

Publication Number Publication Date
JP2023528859A JP2023528859A (ja) 2023-07-06
JP2023528859A5 true JP2023528859A5 (enExample) 2024-05-31
JP7777544B2 JP7777544B2 (ja) 2025-11-28

Family

ID=78830119

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022574270A Active JP7777544B2 (ja) 2020-06-01 2021-06-01 新規ピラジン化合物

Country Status (11)

Country Link
US (1) US12600714B2 (enExample)
EP (1) EP4159731A4 (enExample)
JP (1) JP7777544B2 (enExample)
KR (1) KR20230019444A (enExample)
CN (1) CN115698000B (enExample)
AU (1) AU2021284676A1 (enExample)
BR (1) BR112022022220A2 (enExample)
CA (1) CA3179395A1 (enExample)
MX (1) MX2022013397A (enExample)
TW (1) TWI845843B (enExample)
WO (1) WO2021244505A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4373817B1 (en) * 2021-07-20 2025-05-21 Astrazeneca AB Substituted pyrazine-2-carboxamides as hpk1 inhibitors for the treatment of cancer

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU5108000A (en) 1999-06-10 2001-01-02 Yamanouchi Pharmaceutical Co., Ltd. Novel nitrogen-contaiing heterocyclic derivatives or salts thereof
WO2003045924A1 (en) * 2001-11-21 2003-06-05 Pharmacia & Upjohn Company Substituted aryl 1,4-pyrazine derivatives
JP5364159B2 (ja) * 2009-05-08 2013-12-11 アステラス製薬株式会社 ジアミノへテロ環カルボキサミド化合物
WO2013108754A1 (ja) 2012-01-17 2013-07-25 アステラス製薬株式会社 ピラジンカルボキサミド化合物
CA2975072A1 (en) * 2015-01-28 2016-08-04 Astellas Pharma Inc. Method for producing pyrazinecarboxamide compound and synthetic intermediate thereof
MA42623A (fr) 2015-06-02 2018-06-20 Pharmacyclics Llc Inhibiteurs de la tyrosine kinase de bruton
WO2018103663A1 (zh) * 2016-12-09 2018-06-14 深圳市塔吉瑞生物医药有限公司 一种取代的吡嗪甲酰胺类化合物及包含该化合物的组合物及其用途
EP3656769B1 (en) 2017-07-19 2023-01-25 Chia Tai Tianqing Pharmaceutical Group Co., Ltd. Aryl-phosphorus-oxygen compound as egfr kinase inhibitor

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