JP2023528280A5 - - Google Patents
Info
- Publication number
- JP2023528280A5 JP2023528280A5 JP2022570530A JP2022570530A JP2023528280A5 JP 2023528280 A5 JP2023528280 A5 JP 2023528280A5 JP 2022570530 A JP2022570530 A JP 2022570530A JP 2022570530 A JP2022570530 A JP 2022570530A JP 2023528280 A5 JP2023528280 A5 JP 2023528280A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- pyrazole
- imidazole
- dihydro
- ethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025139598A JP2025168429A (ja) | 2020-05-22 | 2025-08-25 | 例えば、うつ病を治療するための、gpr139拮抗薬としての1-((1h-ピラゾール-4-イル)メチル)-3-(フェニル)-1,3-ジヒドロ-2h-イミダゾール-2-オン誘導体および関連化合物 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020090110 | 2020-05-22 | ||
| JP2020090110A JP2021183586A (ja) | 2020-05-22 | 2020-05-22 | 複素環化合物 |
| PCT/IB2021/000336 WO2021234450A1 (en) | 2020-05-22 | 2021-05-20 | 1-((1h-pyrazol-4-yl)methyl)-3-(phenyl)-1,3-dihydro-2h-imidazol-2-one derivatives and related compounds as gpr139 antagonists for the treatment of e.g. depression |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025139598A Division JP2025168429A (ja) | 2020-05-22 | 2025-08-25 | 例えば、うつ病を治療するための、gpr139拮抗薬としての1-((1h-ピラゾール-4-イル)メチル)-3-(フェニル)-1,3-ジヒドロ-2h-イミダゾール-2-オン誘導体および関連化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023528280A JP2023528280A (ja) | 2023-07-04 |
| JP2023528280A5 true JP2023528280A5 (https=) | 2024-05-23 |
| JP7734152B2 JP7734152B2 (ja) | 2025-09-04 |
Family
ID=76797025
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020090110A Pending JP2021183586A (ja) | 2020-05-22 | 2020-05-22 | 複素環化合物 |
| JP2022570530A Active JP7734152B2 (ja) | 2020-05-22 | 2021-05-20 | 例えば、うつ病を治療するための、gpr139拮抗薬としての1-((1h-ピラゾール-4-イル)メチル)-3-(フェニル)-1,3-ジヒドロ-2h-イミダゾール-2-オン誘導体および関連化合物 |
| JP2025139598A Pending JP2025168429A (ja) | 2020-05-22 | 2025-08-25 | 例えば、うつ病を治療するための、gpr139拮抗薬としての1-((1h-ピラゾール-4-イル)メチル)-3-(フェニル)-1,3-ジヒドロ-2h-イミダゾール-2-オン誘導体および関連化合物 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020090110A Pending JP2021183586A (ja) | 2020-05-22 | 2020-05-22 | 複素環化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025139598A Pending JP2025168429A (ja) | 2020-05-22 | 2025-08-25 | 例えば、うつ病を治療するための、gpr139拮抗薬としての1-((1h-ピラゾール-4-イル)メチル)-3-(フェニル)-1,3-ジヒドロ-2h-イミダゾール-2-オン誘導体および関連化合物 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20230348435A1 (https=) |
| EP (1) | EP4153583B1 (https=) |
| JP (3) | JP2021183586A (https=) |
| AR (1) | AR122142A1 (https=) |
| ES (1) | ES3001126T3 (https=) |
| TW (1) | TW202208349A (https=) |
| WO (1) | WO2021234450A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2021183587A (ja) | 2020-05-22 | 2021-12-02 | 武田薬品工業株式会社 | 複素環化合物 |
| TW202400588A (zh) * | 2022-02-28 | 2024-01-01 | 香港商維泰瑞隆(香港)生物科技有限公司 | Rip1調製劑、其製備及用途 |
| CN121159462A (zh) * | 2025-11-19 | 2025-12-19 | 杭州市第七人民医院(杭州市心理危机研究与干预中心) | 喹唑啉酮类化合物及其在制备神经系统疾病药物中的应用 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2374610A1 (en) | 1999-06-28 | 2001-01-04 | Jordan J. N. Tang | Catalytically active recombinant memapsin and methods of use thereof |
| AR052342A1 (es) * | 2004-12-21 | 2007-03-14 | Janssen Pharmaceutica Nv | Derivados sustituidos de triazolona,tetrazolona e imidazolona con actividad selectiva antagonista de alfa2c-adenoreceptores |
| US8148367B2 (en) | 2007-01-12 | 2012-04-03 | Takeda Pharmaceutical Company Limited | Renin inhibitors |
| WO2008094556A2 (en) | 2007-01-30 | 2008-08-07 | Biogen Idec Ma Inc. | Imidazolone compounds as tgf-beta family type i receptors, alk5 and/or alk4 antagonists |
| WO2011145735A1 (ja) * | 2010-05-21 | 2011-11-24 | 武田薬品工業株式会社 | チアゾール誘導体 |
| AR103990A1 (es) * | 2015-01-09 | 2017-06-21 | Bristol Myers Squibb Co | Ureas cíclicas como inhibidoras de rock |
| WO2020097609A1 (en) * | 2018-11-09 | 2020-05-14 | Blackthorn Therapeutics, Inc. | Gpr139 receptor modulators |
| JP7199940B2 (ja) | 2018-12-03 | 2023-01-06 | 川崎重工業株式会社 | 複合材料製航空機用部品およびその製造方法 |
-
2020
- 2020-05-22 JP JP2020090110A patent/JP2021183586A/ja active Pending
-
2021
- 2021-05-20 ES ES21737768T patent/ES3001126T3/es active Active
- 2021-05-20 WO PCT/IB2021/000336 patent/WO2021234450A1/en not_active Ceased
- 2021-05-20 TW TW110118331A patent/TW202208349A/zh unknown
- 2021-05-20 EP EP21737768.8A patent/EP4153583B1/en active Active
- 2021-05-20 US US17/999,505 patent/US20230348435A1/en active Pending
- 2021-05-20 AR ARP210101386A patent/AR122142A1/es unknown
- 2021-05-20 JP JP2022570530A patent/JP7734152B2/ja active Active
-
2025
- 2025-08-25 JP JP2025139598A patent/JP2025168429A/ja active Pending
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