JP2023516291A5 - - Google Patents
Info
- Publication number
- JP2023516291A5 JP2023516291A5 JP2022551377A JP2022551377A JP2023516291A5 JP 2023516291 A5 JP2023516291 A5 JP 2023516291A5 JP 2022551377 A JP2022551377 A JP 2022551377A JP 2022551377 A JP2022551377 A JP 2022551377A JP 2023516291 A5 JP2023516291 A5 JP 2023516291A5
- Authority
- JP
- Japan
- Prior art keywords
- item
- pharmaceutical composition
- inhibitor
- composition according
- estrogen receptor
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025090731A JP2025131656A (ja) | 2020-03-06 | 2025-05-30 | エストロゲン受容体関連疾患の治療方法 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202062985929P | 2020-03-06 | 2020-03-06 | |
| US62/985,929 | 2020-03-06 | ||
| PCT/US2021/021151 WO2021178846A1 (en) | 2020-03-06 | 2021-03-05 | Methods of treating estrogen receptor-associated diseases |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025090731A Division JP2025131656A (ja) | 2020-03-06 | 2025-05-30 | エストロゲン受容体関連疾患の治療方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023516291A JP2023516291A (ja) | 2023-04-19 |
| JP2023516291A5 true JP2023516291A5 (enExample) | 2024-03-14 |
| JP7708772B2 JP7708772B2 (ja) | 2025-07-15 |
Family
ID=77613854
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022551377A Active JP7708772B2 (ja) | 2020-03-06 | 2021-03-05 | エストロゲン受容体関連疾患の治療方法 |
| JP2025090731A Pending JP2025131656A (ja) | 2020-03-06 | 2025-05-30 | エストロゲン受容体関連疾患の治療方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025090731A Pending JP2025131656A (ja) | 2020-03-06 | 2025-05-30 | エストロゲン受容体関連疾患の治療方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20230129598A1 (enExample) |
| EP (1) | EP4114391B1 (enExample) |
| JP (2) | JP7708772B2 (enExample) |
| KR (1) | KR20220151616A (enExample) |
| CN (1) | CN115175679A (enExample) |
| AU (1) | AU2021230588A1 (enExample) |
| CA (1) | CA3169679A1 (enExample) |
| ES (1) | ES3044433T3 (enExample) |
| MX (1) | MX2022010425A (enExample) |
| WO (1) | WO2021178846A1 (enExample) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2923412T3 (es) | 2018-09-07 | 2022-09-27 | Sanofi Sa | Sales de 6-(2,4-diclorofenil)-5-[4-[(3S)-1-(3-fluoropropil)pirrolidin-3-il]oxifenil]-8,9-dihidro-7H-benzo[7]anuleno-2-carboxilato de metilo y proceso de preparación de las mismas |
| CA3144791A1 (en) * | 2019-07-07 | 2021-01-14 | Olema Pharmaceuticals, Inc. | Regimens of estrogen receptor antagonists |
| JP7680438B2 (ja) | 2019-10-01 | 2025-05-20 | サノフイ | 新規の置換６，７－ジヒドロ－５ｈ－ベンゾ［７］アンヌレン化合物、その製造方法およびその治療的使用 |
| BR112022009705A2 (pt) | 2019-12-09 | 2022-08-09 | Sanofi Sa | Forma cristalina anidra de um derivado de ácido 7h-benzo[7]anuleno-2-carboxílico, seus usos e processos de preparação, forma sólida, medicamento e composição farmacêutica |
| TW202146007A (zh) * | 2020-02-27 | 2021-12-16 | 法商賽諾菲公司 | 包含阿培利司（ａｌｐｅｌｉｓｉｂ）與６－（２，４－二氯苯基）－５－［４－［（３ｓ）－１－（３－氟丙基）吡咯啶－３－基］氧苯基］－８，９－二氫－７ｈ－苯并［７］輪烯－２－羧酸之組合 |
| US12595230B2 (en) | 2020-10-19 | 2026-04-07 | Sanofi | Substituted 6,7-dihydro-5H-benzo[7]annulene compounds and their derivatives, processes for their preparation and therapeutic uses thereof |
| AU2021366223A1 (en) | 2020-10-19 | 2023-06-22 | Sanofi | Substituted 6,7-dihydro-5h-benzo[7]annulene compounds and their derivatives, processes for their preparation and therapeutic uses thereof |
| TWI808648B (zh) * | 2021-02-16 | 2023-07-11 | 美商建南德克公司 | 使用包含gdc-9545及gdc-0077之組合療法治療乳癌 |
| TW202304424A (zh) * | 2021-04-12 | 2023-02-01 | 法商賽諾菲公司 | 包含依維莫司和安森司群的組合 |
| TW202304425A (zh) * | 2021-04-12 | 2023-02-01 | 法商賽諾菲公司 | 包含瑞博西尼和安森司群（ａｍｃｅｎｅｓｔｒａｎｔ）的組合 |
| CN118119620A (zh) * | 2021-11-12 | 2024-05-31 | 南京再明医药有限公司 | 用于治疗肿瘤的药物组合及其应用 |
| KR102743629B1 (ko) * | 2022-02-01 | 2024-12-17 | 일라이 릴리 앤드 캄파니 | 선택적 에스트로겐 수용체 분해제의 제조 방법 |
| WO2023150238A1 (en) * | 2022-02-02 | 2023-08-10 | Intrinsic Innovation Llc | Object placement |
| WO2023221122A1 (en) * | 2022-05-20 | 2023-11-23 | Olema Pharmaceuticals, Inc. | Salts and solid forms of an estrogen receptor antagonist |
| WO2023221123A1 (en) * | 2022-05-20 | 2023-11-23 | Olema Pharmaceuticals, Inc. | Crystalline forms of an estrogen receptor antagonist |
| WO2024015506A1 (en) * | 2022-07-14 | 2024-01-18 | Olema Pharmaceuticals, Inc. | Methods of treating estrogen receptor-mediated disorders |
| CN114933558B (zh) * | 2022-07-26 | 2022-11-22 | 常熟药明康德新药开发有限公司 | 手性硝基化合物催化还原制备手性氨基化合物的方法 |
| EP4598520A1 (en) * | 2022-10-05 | 2025-08-13 | Olema Pharmaceuticals, Inc. | Methods of treating estrogen receptor-mediated disorders |
| WO2024076633A1 (en) * | 2022-10-05 | 2024-04-11 | Olema Pharmaceuticals, Inc. | Methods of treating estrogen receptor-mediated disorders |
| CN115872996B (zh) * | 2023-02-21 | 2023-05-05 | 山东绿叶制药有限公司 | 一种雌激素受体降解剂化合物及其制备方法和应用 |
| WO2025106890A1 (en) * | 2023-11-17 | 2025-05-22 | Olema Pharmaceuticals, Inc. | Salts and solid forms of an estrogen receptor antagonist |
| US12558428B2 (en) | 2024-03-08 | 2026-02-24 | Halda Therapeutics Opco, Inc. | Heterobifunctional compounds and their use in treating disease |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20120157402A1 (en) * | 2009-05-27 | 2012-06-21 | Liangxian Cao | Methods for treating brain tumors |
| US9540361B2 (en) | 2010-12-24 | 2017-01-10 | Merck Sharp & Dohme B.V. | N-substituted azetidine derivatives |
| EP2791128A4 (en) | 2011-12-16 | 2015-04-22 | Olema Pharmaceuticals Inc | NOVEL BENZOPYRAN COMPOUNDS, COMPOSITIONS AND USES THEREOF |
| PE20160874A1 (es) | 2013-05-28 | 2016-09-04 | Astrazeneca Ab | Compuestos quimicos |
| US9855270B2 (en) * | 2014-03-13 | 2018-01-02 | Genentech, Inc. | Methods and compositions for modulating estrogen receptor mutants |
| RS67458B1 (sr) * | 2014-03-28 | 2025-12-31 | Univ Duke | Lečenje kancera dojke pozitivnog na receptor estrogena upotrebom selektivnih modulatora receptora estrogena |
| CN117865872A (zh) | 2014-12-18 | 2024-04-12 | 豪夫迈·罗氏有限公司 | 四氢-吡啶并[3,4-b]吲哚雌激素受体调节剂及其用途 |
| KR102676629B1 (ko) * | 2015-04-29 | 2024-06-18 | 래디어스 파마슈티컬스, 인코포레이티드 | 암을 치료하는 방법 |
| DK3355884T3 (da) * | 2015-10-01 | 2021-08-02 | Olema Pharmaceuticals Inc | Tetrahydro-1h-pyrido[3,4-b]indol-antiøstrogenlægemidler |
| WO2018157000A1 (en) * | 2017-02-23 | 2018-08-30 | Olema Pharmaceuticals, Inc. | Compositions and methods for regulating immune system activity |
| TWI915239B (zh) | 2018-06-21 | 2026-02-11 | 瑞士商赫孚孟拉羅股份公司 | 3-((1r,3r)-1-(2,6-二氟-4-((1-(3-氟丙基)氮雜環丁-3-基)胺基)苯基)-3-甲基-1,3,4,9-四氫-2h-吡啶并[3,4-b]吲哚-2-基)-2,2-二氟丙-1-醇之固體形式及用於製備包含經取代苯基或吡啶基部分之稠合三環化合物之製程，包括其使用方法 |
| TW202430189A (zh) * | 2018-07-23 | 2024-08-01 | 瑞士商赫孚孟拉羅股份公司 | 用pi3k抑制劑gdc-0077治療癌症之方法 |
| MX2021001857A (es) * | 2018-08-17 | 2021-10-13 | Genentech Inc Star | Metodos de diagnostico y terapeuticos para el tratamiento del cancer de mama. |
-
2021
- 2021-03-05 MX MX2022010425A patent/MX2022010425A/es unknown
- 2021-03-05 EP EP21763872.5A patent/EP4114391B1/en active Active
- 2021-03-05 ES ES21763872T patent/ES3044433T3/es active Active
- 2021-03-05 CN CN202180016388.2A patent/CN115175679A/zh active Pending
- 2021-03-05 CA CA3169679A patent/CA3169679A1/en active Pending
- 2021-03-05 AU AU2021230588A patent/AU2021230588A1/en active Pending
- 2021-03-05 KR KR1020227030151A patent/KR20220151616A/ko active Pending
- 2021-03-05 WO PCT/US2021/021151 patent/WO2021178846A1/en not_active Ceased
- 2021-03-05 JP JP2022551377A patent/JP7708772B2/ja active Active
- 2021-03-05 US US17/908,941 patent/US20230129598A1/en active Pending
-
2025
- 2025-05-30 JP JP2025090731A patent/JP2025131656A/ja active Pending
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