JP2023513679A - 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体 - Google Patents

中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体 Download PDF

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JP2023513679A
JP2023513679A JP2022548056A JP2022548056A JP2023513679A JP 2023513679 A JP2023513679 A JP 2023513679A JP 2022548056 A JP2022548056 A JP 2022548056A JP 2022548056 A JP2022548056 A JP 2022548056A JP 2023513679 A JP2023513679 A JP 2023513679A
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JPWO2021155468A5 (https=
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スラッシ、アブデルマリク
アラウホ、ジョーセフ
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マインドセット ファーマ インコーポレイテッド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/572—Five-membered rings
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    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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JP2022548056A 2020-02-04 2021-02-04 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体 Pending JP2023513679A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025172009A JP2026010068A (ja) 2020-02-04 2025-10-10 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体

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US202062969934P 2020-02-04 2020-02-04
US62/969,934 2020-02-04
PCT/CA2021/050123 WO2021155468A1 (en) 2020-02-04 2021-02-04 Psilocin derivatives as serotonergic psychedelic agents for the treatment of cns disorders

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JP2025172009A Division JP2026010068A (ja) 2020-02-04 2025-10-10 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体

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JP2023513679A true JP2023513679A (ja) 2023-04-03
JPWO2021155468A5 JPWO2021155468A5 (https=) 2024-02-07
JP2023513679A5 JP2023513679A5 (https=) 2024-02-07

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JP2022548056A Pending JP2023513679A (ja) 2020-02-04 2021-02-04 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体
JP2022548057A Pending JP2023513680A (ja) 2020-02-04 2021-02-04 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体
JP2024015076A Pending JP2024054193A (ja) 2020-02-04 2024-02-02 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体
JP2025172009A Pending JP2026010068A (ja) 2020-02-04 2025-10-10 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体
JP2025243928A Pending JP2026053405A (ja) 2020-02-04 2025-12-09 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体

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JP2022548057A Pending JP2023513680A (ja) 2020-02-04 2021-02-04 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体
JP2024015076A Pending JP2024054193A (ja) 2020-02-04 2024-02-02 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体
JP2025172009A Pending JP2026010068A (ja) 2020-02-04 2025-10-10 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体
JP2025243928A Pending JP2026053405A (ja) 2020-02-04 2025-12-09 中枢神経系障害の治療のためのセロトニン作動性幻覚薬としてのシロシン誘導体

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US (9) US20220024956A1 (https=)
EP (2) EP4100390A4 (https=)
JP (5) JP2023513679A (https=)
KR (3) KR20240023678A (https=)
CN (3) CN115974757A (https=)
AU (2) AU2021217424A1 (https=)
BR (2) BR112022015375A2 (https=)
CA (2) CA3166936A1 (https=)
IL (2) IL295371B1 (https=)
MX (2) MX2022009526A (https=)
PH (1) PH12022551981A1 (https=)
WO (2) WO2021155468A1 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2024508922A (ja) * 2021-03-02 2024-02-28 マインドセット ファーマ インコーポレイテッド セロトニン作動性薬に関係する障害の治療に有用なセロトニン作動性薬としてのインドール誘導体

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