JP2023512823A5 - - Google Patents

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Publication number
JP2023512823A5
JP2023512823A5 JP2022548109A JP2022548109A JP2023512823A5 JP 2023512823 A5 JP2023512823 A5 JP 2023512823A5 JP 2022548109 A JP2022548109 A JP 2022548109A JP 2022548109 A JP2022548109 A JP 2022548109A JP 2023512823 A5 JP2023512823 A5 JP 2023512823A5
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JP
Japan
Prior art keywords
alkyl
group
alkoxy
hydrogen
hydrocarbyl
Prior art date
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Granted
Application number
JP2022548109A
Other languages
English (en)
Japanese (ja)
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JP7678595B2 (ja
JP2023512823A (ja
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Priority claimed from PCT/US2021/016848 external-priority patent/WO2021158936A1/en
Publication of JP2023512823A publication Critical patent/JP2023512823A/ja
Publication of JP2023512823A5 publication Critical patent/JP2023512823A5/ja
Application granted granted Critical
Publication of JP7678595B2 publication Critical patent/JP7678595B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022548109A 2020-02-05 2021-02-05 ピロロ[2,3‐b]ピリジン‐3‐カルボキサミド組成物及び聴力損失を改善するための方法 Active JP7678595B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062970425P 2020-02-05 2020-02-05
US62/970,425 2020-02-05
PCT/US2021/016848 WO2021158936A1 (en) 2020-02-05 2021-02-05 Pyrrolo [2,3-b]pyridine-3-carboxamide compositions and methods for ameliorating hearing loss

Publications (3)

Publication Number Publication Date
JP2023512823A JP2023512823A (ja) 2023-03-29
JP2023512823A5 true JP2023512823A5 (https=) 2025-03-21
JP7678595B2 JP7678595B2 (ja) 2025-05-16

Family

ID=77199407

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022548109A Active JP7678595B2 (ja) 2020-02-05 2021-02-05 ピロロ[2,3‐b]ピリジン‐3‐カルボキサミド組成物及び聴力損失を改善するための方法

Country Status (8)

Country Link
EP (1) EP4100008B1 (https=)
JP (1) JP7678595B2 (https=)
CN (1) CN115515579B (https=)
AU (1) AU2021215925B2 (https=)
CA (1) CA3170121A1 (https=)
ES (1) ES3025983T3 (https=)
MX (1) MX2022009572A (https=)
WO (1) WO2021158936A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023015156A1 (en) * 2021-08-02 2023-02-09 Hudspeth A James Pyrrolopyridine-3- and 4-carboxamide compositions and methods for cellular proliferation
WO2024211621A1 (en) * 2023-04-04 2024-10-10 Children's Hospital Los Angeles Lats kinase inhibitor to treat retinal degeneration

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2888848B1 (fr) * 2005-07-22 2007-09-28 Sanofi Aventis Sa Derives de n-(arylalkyl)-1h-pyrrrolopyridine-2-carboxamides, leur preparation et leur application en therapeutique
WO2007067537A1 (en) * 2005-12-07 2007-06-14 Osi Pharmaceuticals, Inc. Pyrrolopyridine kinase inhibiting compounds
PE20121126A1 (es) * 2006-12-21 2012-08-24 Plexxikon Inc Compuestos pirrolo [2,3-b] piridinas como moduladores de quinasa
TWI667233B (zh) * 2013-12-19 2019-08-01 德商拜耳製藥公司 新穎吲唑羧醯胺,其製備方法、含彼等之醫藥製劑及其製造醫藥之用途
GB201602854D0 (en) * 2016-02-18 2016-04-06 Mission Therapeutics Ltd Novel compounds
JOP20190257A1 (ar) 2017-04-28 2019-10-28 Novartis Ag مركبات أريل غير متجانسة ثنائية الحلقة مندمجة 6-6 واستخدامها كمثبطات lats

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