JP2023512729A5 - - Google Patents
Info
- Publication number
- JP2023512729A5 JP2023512729A5 JP2022548400A JP2022548400A JP2023512729A5 JP 2023512729 A5 JP2023512729 A5 JP 2023512729A5 JP 2022548400 A JP2022548400 A JP 2022548400A JP 2022548400 A JP2022548400 A JP 2022548400A JP 2023512729 A5 JP2023512729 A5 JP 2023512729A5
- Authority
- JP
- Japan
- Prior art keywords
- invention described
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202062972484P | 2020-02-10 | 2020-02-10 | |
| US62/972,484 | 2020-02-10 | ||
| PCT/EP2021/053062 WO2021160602A1 (en) | 2020-02-10 | 2021-02-09 | Monoacylglycerol lipase modulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023512729A JP2023512729A (ja) | 2023-03-28 |
| JP2023512729A5 true JP2023512729A5 (https=) | 2024-02-20 |
| JP7795466B2 JP7795466B2 (ja) | 2026-01-07 |
Family
ID=74595268
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022548400A Active JP7795466B2 (ja) | 2020-02-10 | 2021-02-09 | モノアシルグリセロールリパーゼ調節因子 |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US11708359B2 (https=) |
| EP (1) | EP4103557B1 (https=) |
| JP (1) | JP7795466B2 (https=) |
| KR (1) | KR20220140581A (https=) |
| CN (1) | CN115066422B (https=) |
| AR (1) | AR121296A1 (https=) |
| AU (1) | AU2021220539A1 (https=) |
| BR (1) | BR112022015116A2 (https=) |
| CA (1) | CA3169988A1 (https=) |
| CL (1) | CL2022002136A1 (https=) |
| CO (1) | CO2022011275A2 (https=) |
| CR (1) | CR20220376A (https=) |
| DO (1) | DOP2022000162A (https=) |
| EC (1) | ECSP22062460A (https=) |
| IL (1) | IL295447A (https=) |
| JO (1) | JOP20220180A1 (https=) |
| MX (1) | MX2022009804A (https=) |
| PE (1) | PE20221576A1 (https=) |
| PH (1) | PH12022552019A1 (https=) |
| TW (1) | TW202140465A (https=) |
| UY (1) | UY39066A (https=) |
| WO (1) | WO2021160602A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202140465A (zh) * | 2020-02-10 | 2021-11-01 | 比利時商健生藥品公司 | 單醯基甘油脂酶調節劑 |
| CN115362151B (zh) | 2020-03-26 | 2025-02-11 | 詹森药业有限公司 | 作为单酰基甘油脂肪酶调节剂的芳基哌啶 |
| MX2022011903A (es) | 2020-03-26 | 2023-01-11 | Janssen Pharmaceutica Nv | Azaspirociclos como moduladores de monoacilglicerol lipasa. |
| WO2021191391A1 (en) | 2020-03-26 | 2021-09-30 | Janssen Pharmaceutica Nv | Aminocyclobutanes as monoacylglycerol lipase modulators |
| US12115154B2 (en) | 2020-12-16 | 2024-10-15 | Srx Cardio, Llc | Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9) |
| CA3228446A1 (en) | 2021-08-09 | 2023-02-16 | Janssen Pharmaceutica Nv | Monoacylglycerol lipase modulators for use in autism spectrum disorders |
| CA3242372A1 (en) | 2021-12-29 | 2023-07-06 | Psy Therapeutics, Inc. | Inhibiting monoacylglycerol lipase (magl) |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2493637A1 (en) | 2002-07-25 | 2004-02-12 | Manuela Villa | Bicyclo-pyrazoles active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them |
| EP2090576A1 (en) | 2008-02-01 | 2009-08-19 | Merz Pharma GmbH & Co.KGaA | 6-halo-pyrazolo[1,5-a]pyridines, a process for their preparation and their use as metabotropic glutamate receptor (mGluR) modulators |
| KR20140068243A (ko) * | 2011-09-30 | 2014-06-05 | 얀센 파마슈티카 엔.브이. | 대사 질환 및 관련 장애의 치료를 위한 모노아실글리세롤 리파제 억제제 |
| WO2017170830A1 (ja) | 2016-03-31 | 2017-10-05 | 武田薬品工業株式会社 | 複素環化合物 |
| EA036637B1 (ru) | 2016-03-31 | 2020-12-02 | Такеда Фармасьютикал Компани Лимитед | Гетероциклические спиросоединения, ингибирующие моноацилглицерин-липазу |
| GB201613163D0 (en) | 2016-07-29 | 2016-09-14 | Autifony Therapeutics Ltd | Novel compounds |
| MX2020007318A (es) * | 2017-09-29 | 2020-08-24 | Takeda Pharmaceuticals Co | Compuesto heterociclico. |
| CN112272670B (zh) | 2019-04-16 | 2023-12-12 | 上海翰森生物医药科技有限公司 | 含二并环类衍生物抑制剂、其制备方法和应用 |
| TW202140465A (zh) | 2020-02-10 | 2021-11-01 | 比利時商健生藥品公司 | 單醯基甘油脂酶調節劑 |
| CN115362151B (zh) | 2020-03-26 | 2025-02-11 | 詹森药业有限公司 | 作为单酰基甘油脂肪酶调节剂的芳基哌啶 |
| MX2022011903A (es) | 2020-03-26 | 2023-01-11 | Janssen Pharmaceutica Nv | Azaspirociclos como moduladores de monoacilglicerol lipasa. |
| WO2021191391A1 (en) | 2020-03-26 | 2021-09-30 | Janssen Pharmaceutica Nv | Aminocyclobutanes as monoacylglycerol lipase modulators |
-
2021
- 2021-02-09 TW TW110104960A patent/TW202140465A/zh unknown
- 2021-02-09 CA CA3169988A patent/CA3169988A1/en active Pending
- 2021-02-09 KR KR1020227031216A patent/KR20220140581A/ko not_active Withdrawn
- 2021-02-09 PE PE2022001698A patent/PE20221576A1/es unknown
- 2021-02-09 JP JP2022548400A patent/JP7795466B2/ja active Active
- 2021-02-09 CR CR20220376A patent/CR20220376A/es unknown
- 2021-02-09 UY UY0001039066A patent/UY39066A/es unknown
- 2021-02-09 US US17/171,559 patent/US11708359B2/en active Active
- 2021-02-09 MX MX2022009804A patent/MX2022009804A/es unknown
- 2021-02-09 CN CN202180013762.3A patent/CN115066422B/zh active Active
- 2021-02-09 AU AU2021220539A patent/AU2021220539A1/en active Pending
- 2021-02-09 EP EP21705124.2A patent/EP4103557B1/en active Active
- 2021-02-09 IL IL295447A patent/IL295447A/en unknown
- 2021-02-09 PH PH1/2022/552019A patent/PH12022552019A1/en unknown
- 2021-02-09 BR BR112022015116A patent/BR112022015116A2/pt unknown
- 2021-02-09 WO PCT/EP2021/053062 patent/WO2021160602A1/en not_active Ceased
- 2021-02-09 AR ARP210100333A patent/AR121296A1/es not_active Application Discontinuation
-
2022
- 2022-08-08 CL CL2022002136A patent/CL2022002136A1/es unknown
- 2022-08-09 EC ECSENADI202262460A patent/ECSP22062460A/es unknown
- 2022-08-09 JO JOP/2022/0180A patent/JOP20220180A1/ar unknown
- 2022-08-10 CO CONC2022/0011275A patent/CO2022011275A2/es unknown
- 2022-08-10 DO DO2022000162A patent/DOP2022000162A/es unknown
-
2023
- 2023-06-02 US US18/328,242 patent/US20230382902A1/en not_active Abandoned