JP2023503852A5 - - Google Patents
Info
- Publication number
- JP2023503852A5 JP2023503852A5 JP2022527989A JP2022527989A JP2023503852A5 JP 2023503852 A5 JP2023503852 A5 JP 2023503852A5 JP 2022527989 A JP2022527989 A JP 2022527989A JP 2022527989 A JP2022527989 A JP 2022527989A JP 2023503852 A5 JP2023503852 A5 JP 2023503852A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- pyridine
- oxy
- piperidine
- dichlorophenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962934407P | 2019-11-12 | 2019-11-12 | |
| US62/934,407 | 2019-11-12 | ||
| PCT/US2020/060108 WO2021097009A1 (en) | 2019-11-12 | 2020-11-12 | Small molecule furin inhibitors for treating infectious diseases |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2023503852A JP2023503852A (ja) | 2023-02-01 |
| JP2023503852A5 true JP2023503852A5 (enExample) | 2023-11-20 |
Family
ID=73793799
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022527989A Pending JP2023503852A (ja) | 2019-11-12 | 2020-11-12 | 感染症を処置するための低分子フーリン阻害剤 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20230011571A1 (enExample) |
| EP (1) | EP4058021A1 (enExample) |
| JP (1) | JP2023503852A (enExample) |
| KR (1) | KR20220104744A (enExample) |
| CN (1) | CN114929220A (enExample) |
| AU (1) | AU2020382819A1 (enExample) |
| CA (1) | CA3157892A1 (enExample) |
| WO (1) | WO2021097009A1 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112384509B (zh) | 2018-05-11 | 2024-04-30 | 葛兰素史密斯克莱知识产权发展有限公司 | 弗林蛋白酶抑制剂 |
| DE102023126563A1 (de) * | 2023-09-28 | 2025-04-03 | Philipps-Universität Marburg, Körperschaft des öffentlichen Rechts | Hemmstoffe der Proproteinkonvertase Furin, Verfahren zu deren Herstellung und Verwendung |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003037346A1 (en) * | 2001-10-31 | 2003-05-08 | Cell Therapeutics, Inc. | 6-phenyl-n-phenyl-(1,3,5) -triazine-2,4-diamine derivatives and related compounds with lysophphosphatidic acid acyltransferase beta (lpaat-beta) inhibitory activity for use in the treatment of cancer |
| CA2687024A1 (en) | 2007-05-09 | 2009-02-19 | Burnham Institute For Medical Research | Targeting host proteinases as a therapeutic strategy against viral and bacterial pathogens |
| WO2013138666A1 (en) | 2012-03-16 | 2013-09-19 | Sanford-Burnham Medical Research Institute | Inhibitors of furin and other pro-protein convertases |
| WO2014152716A1 (en) * | 2013-03-15 | 2014-09-25 | President And Fellows Of Harvard College | Substituted heterocyclic compounds for treating or preventing viral infections |
| CN107441094B (zh) * | 2017-08-08 | 2020-05-22 | 南方医科大学 | 尼罗替尼作为治疗登革病毒感染的药物及其制药用途 |
| CN112384509B (zh) * | 2018-05-11 | 2024-04-30 | 葛兰素史密斯克莱知识产权发展有限公司 | 弗林蛋白酶抑制剂 |
-
2020
- 2020-11-12 CA CA3157892A patent/CA3157892A1/en active Pending
- 2020-11-12 CN CN202080092431.9A patent/CN114929220A/zh active Pending
- 2020-11-12 US US17/776,067 patent/US20230011571A1/en not_active Abandoned
- 2020-11-12 WO PCT/US2020/060108 patent/WO2021097009A1/en not_active Ceased
- 2020-11-12 KR KR1020227019647A patent/KR20220104744A/ko not_active Ceased
- 2020-11-12 EP EP20823987.1A patent/EP4058021A1/en active Pending
- 2020-11-12 JP JP2022527989A patent/JP2023503852A/ja active Pending
- 2020-11-12 AU AU2020382819A patent/AU2020382819A1/en active Pending
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