JP2023169446A - ホスアプレピタント注射用水溶液剤 - Google Patents
ホスアプレピタント注射用水溶液剤 Download PDFInfo
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- JP2023169446A JP2023169446A JP2020170581A JP2020170581A JP2023169446A JP 2023169446 A JP2023169446 A JP 2023169446A JP 2020170581 A JP2020170581 A JP 2020170581A JP 2020170581 A JP2020170581 A JP 2020170581A JP 2023169446 A JP2023169446 A JP 2023169446A
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- fosaprepitant
- aqueous solution
- injection
- related substances
- acid
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- 229940032329 fosaprepitant injection Drugs 0.000 title claims abstract description 9
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- 229960002891 fosaprepitant Drugs 0.000 claims abstract description 150
- QPCDCPDFJACHGM-UHFFFAOYSA-N N,N-bis{2-[bis(carboxymethyl)amino]ethyl}glycine Chemical compound OC(=O)CN(CC(O)=O)CCN(CC(=O)O)CCN(CC(O)=O)CC(O)=O QPCDCPDFJACHGM-UHFFFAOYSA-N 0.000 claims abstract description 38
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- 238000002347 injection Methods 0.000 claims description 52
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Images
Classifications
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Inorganic Chemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020170581A JP2023169446A (ja) | 2020-10-08 | 2020-10-08 | ホスアプレピタント注射用水溶液剤 |
| PCT/JP2021/037143 WO2022075408A1 (ja) | 2020-10-08 | 2021-10-07 | ホスアプレピタント注射用水溶液剤 |
| TW110137565A TW202228718A (zh) | 2020-10-08 | 2021-10-08 | 福沙吡坦注射用水溶液劑、福沙吡坦注射用水溶液劑中福沙吡坦類似物質的生成抑制劑以及生成抑制方法、二乙三胺五乙酸的用途 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020170581A JP2023169446A (ja) | 2020-10-08 | 2020-10-08 | ホスアプレピタント注射用水溶液剤 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2023169446A true JP2023169446A (ja) | 2023-11-30 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020170581A Pending JP2023169446A (ja) | 2020-10-08 | 2020-10-08 | ホスアプレピタント注射用水溶液剤 |
Country Status (3)
| Country | Link |
|---|---|
| JP (1) | JP2023169446A (zh) |
| TW (1) | TW202228718A (zh) |
| WO (1) | WO2022075408A1 (zh) |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017021880A1 (en) * | 2015-08-03 | 2017-02-09 | Leiutis Pharmaceuticals Pvt Ltd | Liquid formulations of fosaprepitant |
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2020
- 2020-10-08 JP JP2020170581A patent/JP2023169446A/ja active Pending
-
2021
- 2021-10-07 WO PCT/JP2021/037143 patent/WO2022075408A1/ja active Application Filing
- 2021-10-08 TW TW110137565A patent/TW202228718A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2022075408A1 (ja) | 2022-04-14 |
| TW202228718A (zh) | 2022-08-01 |
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