JP2023116489A5 - - Google Patents

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Publication number
JP2023116489A5
JP2023116489A5 JP2023084119A JP2023084119A JP2023116489A5 JP 2023116489 A5 JP2023116489 A5 JP 2023116489A5 JP 2023084119 A JP2023084119 A JP 2023084119A JP 2023084119 A JP2023084119 A JP 2023084119A JP 2023116489 A5 JP2023116489 A5 JP 2023116489A5
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JP
Japan
Prior art keywords
pharmaceutical composition
composition according
dose
pharmaceutically acceptable
acceptable salt
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JP2023084119A
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English (en)
Japanese (ja)
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JP2023116489A (ja
JP7720354B2 (ja
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Priority claimed from JP2019572820A external-priority patent/JP7285222B2/ja
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Publication of JP2023116489A5 publication Critical patent/JP2023116489A5/ja
Application granted granted Critical
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JP2023084119A 2017-08-14 2023-05-22 副腎皮質刺激ホルモン放出因子受容体拮抗薬 Active JP7720354B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201762545393P 2017-08-14 2017-08-14
US62/545,393 2017-08-14
JP2019572820A JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬
PCT/US2018/046707 WO2019036472A1 (en) 2017-08-14 2018-08-14 CORTICOTROPIN RELEASE FACTOR RECEPTOR ANTAGONISTS

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2019572820A Division JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Publications (3)

Publication Number Publication Date
JP2023116489A JP2023116489A (ja) 2023-08-22
JP2023116489A5 true JP2023116489A5 (https=) 2023-10-26
JP7720354B2 JP7720354B2 (ja) 2025-08-07

Family

ID=65362465

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2019572820A Active JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬
JP2023084119A Active JP7720354B2 (ja) 2017-08-14 2023-05-22 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2019572820A Active JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Country Status (13)

Country Link
US (1) US20210137935A1 (https=)
EP (1) EP3630763A4 (https=)
JP (2) JP7285222B2 (https=)
KR (1) KR102644781B1 (https=)
CN (1) CN110997667A (https=)
AR (1) AR112471A1 (https=)
AU (3) AU2018318990B2 (https=)
BR (1) BR112020002966A2 (https=)
CA (1) CA3064445A1 (https=)
EA (1) EA202090321A1 (https=)
MX (2) MX2019015318A (https=)
TW (2) TWI803504B (https=)
WO (1) WO2019036472A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015112642A1 (en) 2014-01-21 2015-07-30 Neurocrine Biosciences, Inc. Crf1 receptor antagonists for the treatment of congenital adrenal hyperplasia
CN118845788A (zh) 2017-08-14 2024-10-29 云杉生物科学公司 促肾上腺皮质激素释放因子受体拮抗剂
EA202090321A1 (ru) * 2017-08-14 2020-09-24 Спрюс Биосайнсес, Инк. Антагонисты рецептора кортикотропин-рилизинг фактора
EP4438124A3 (en) 2018-04-27 2024-12-18 Spruce Biosciences, Inc. Methods for treating testicular and ovarian adrenal rest tumors
CA3121920A1 (en) 2018-12-07 2020-06-11 Neurocrine Biosciences, Inc. Crf1 receptor antagonist, pharmaceutical formulations and solid forms thereof for the treatment of congenital adrenal hyperplasia
TW202116324A (zh) * 2019-07-19 2021-05-01 美商雲杉生物科技股份有限公司 治療先天性腎上腺增生之方法
JP7623365B2 (ja) 2019-09-27 2025-01-28 ニューロクライン バイオサイエンシーズ,インコーポレイテッド Crf受容体アンタゴニストおよび使用方法
BR112023002497A2 (pt) * 2020-08-12 2023-05-02 Spruce Biosciences Inc Métodos e composições para tratamento da síndrome dos ovários policísticos
JP2023540223A (ja) * 2020-08-26 2023-09-22 ニューロクライン バイオサイエンシーズ,インコーポレイテッド Crf受容体アンタゴニストおよび使用方法
US11708372B2 (en) 2021-11-19 2023-07-25 Spruce Biosciences, Inc. Crystalline composition of tildacerfont and methods of use and preparation thereof
WO2025188842A1 (en) * 2024-03-08 2025-09-12 Spruce Biosciences, Inc. Amorphous solid dispersion of tildacerfont formulations

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3356291B2 (ja) * 1996-02-07 2002-12-16 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Crfレセプター拮抗薬としてのピラゾロピリミジン類
IL137019A (en) * 1998-01-28 2010-11-30 Du Pont Pharm Co 2,7 - dimethyl - 4 - (substituted amino) - 8 - arylpyrazolo [1,5-a] triazine derivatives and pharmaceutical compositions containing them
EP1049699B1 (en) * 1998-01-28 2004-04-21 Bristol-Myers Squibb Pharma Company Pyrazolotriazines as crf antagonists
JP2003516353A (ja) * 1999-12-08 2003-05-13 ファルマシア コーポレイション ヴァルデコキシブ組成物
WO2005079868A2 (en) * 2004-02-13 2005-09-01 Sb Pharmco Puerto Rico Inc Crf receptor antagonists, their preparations, their pharmaceutical composition and their uses
AU2006227300B2 (en) * 2005-03-21 2012-02-02 Eli Lilly And Company Imidazopyridazine compounds
AU2007297481B2 (en) * 2006-09-20 2012-03-08 Eli Lilly And Company Thiophene pyrazolopyrimidine compounds
EP2094709B1 (en) * 2006-09-20 2010-09-15 Eli Lilly And Company Thiazole pyrazolopyrimidines as crf1 receptor antagonists
WO2010039678A1 (en) * 2008-10-02 2010-04-08 Eli Lilly And Company Thiazolyl-pyrazolopyrimidine compounds as synthetic intermediates and related synthetic processes
EA202090321A1 (ru) 2017-08-14 2020-09-24 Спрюс Биосайнсес, Инк. Антагонисты рецептора кортикотропин-рилизинг фактора

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