JP2023116489A5 - - Google Patents

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Publication number
JP2023116489A5
JP2023116489A5 JP2023084119A JP2023084119A JP2023116489A5 JP 2023116489 A5 JP2023116489 A5 JP 2023116489A5 JP 2023084119 A JP2023084119 A JP 2023084119A JP 2023084119 A JP2023084119 A JP 2023084119A JP 2023116489 A5 JP2023116489 A5 JP 2023116489A5
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JP
Japan
Prior art keywords
pharmaceutical composition
composition according
dose
pharmaceutically acceptable
acceptable salt
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Application number
JP2023084119A
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English (en)
Japanese (ja)
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JP2023116489A (ja
JP7720354B2 (ja
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Priority claimed from PCT/US2018/046707 external-priority patent/WO2019036472A1/en
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Publication of JP2023116489A publication Critical patent/JP2023116489A/ja
Publication of JP2023116489A5 publication Critical patent/JP2023116489A5/ja
Application granted granted Critical
Publication of JP7720354B2 publication Critical patent/JP7720354B2/ja
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JP2023084119A 2017-08-14 2023-05-22 副腎皮質刺激ホルモン放出因子受容体拮抗薬 Active JP7720354B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201762545393P 2017-08-14 2017-08-14
US62/545,393 2017-08-14
PCT/US2018/046707 WO2019036472A1 (en) 2017-08-14 2018-08-14 CORTICOTROPIN RELEASE FACTOR RECEPTOR ANTAGONISTS
JP2019572820A JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2019572820A Division JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Publications (3)

Publication Number Publication Date
JP2023116489A JP2023116489A (ja) 2023-08-22
JP2023116489A5 true JP2023116489A5 (https=) 2023-10-26
JP7720354B2 JP7720354B2 (ja) 2025-08-07

Family

ID=65362465

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2019572820A Active JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬
JP2023084119A Active JP7720354B2 (ja) 2017-08-14 2023-05-22 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2019572820A Active JP7285222B2 (ja) 2017-08-14 2018-08-14 副腎皮質刺激ホルモン放出因子受容体拮抗薬

Country Status (13)

Country Link
US (1) US20210137935A1 (https=)
EP (1) EP3630763A4 (https=)
JP (2) JP7285222B2 (https=)
KR (1) KR102644781B1 (https=)
CN (1) CN110997667A (https=)
AR (1) AR112471A1 (https=)
AU (3) AU2018318990B2 (https=)
BR (1) BR112020002966A2 (https=)
CA (1) CA3064445A1 (https=)
EA (1) EA202090321A1 (https=)
MX (2) MX2019015318A (https=)
TW (2) TW202400179A (https=)
WO (1) WO2019036472A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RS65839B1 (sr) 2014-01-21 2024-09-30 Neurocrine Biosciences Inc Crf1 receptor antagonisti za tretman kongenitalne adrenalne hiperplazije
JP7285222B2 (ja) * 2017-08-14 2023-06-01 スプルース バイオサイエンシズ インコーポレイテッド 副腎皮質刺激ホルモン放出因子受容体拮抗薬
WO2019036503A1 (en) 2017-08-14 2019-02-21 Spruce Biosciences, Inc. CORTICOTROPIN RELEASE FACTOR RECEPTOR ANTAGONISTS
EP4643950A3 (en) * 2018-04-27 2026-01-14 Spruce Biosciences, Inc. Methods for treating testicular and ovarian adrenal rest tumors
US20220023266A1 (en) 2018-12-07 2022-01-27 Neurocrine Biosciences, Inc. Crf1 receptor antagonist, pharmaceutical formulations and solid forms thereof for the treatment of congenital adrenal hyperplasia
JP2022541550A (ja) * 2019-07-19 2022-09-26 スプルース バイオサイエンシーズ,インク. 先天性副腎過形成を処置する方法
JP7623365B2 (ja) 2019-09-27 2025-01-28 ニューロクライン バイオサイエンシーズ,インコーポレイテッド Crf受容体アンタゴニストおよび使用方法
KR20240023691A (ko) 2020-08-12 2024-02-22 스프루스 바이오사이언시스 인코포레이티드 다낭성 난소 증후군을 치료하기 위한 방법 및 조성물
US20240024330A1 (en) * 2020-08-26 2024-01-25 Neurocrine Biosciences, Inc. Crf receptor antagonists and methods of use
US11708372B2 (en) 2021-11-19 2023-07-25 Spruce Biosciences, Inc. Crystalline composition of tildacerfont and methods of use and preparation thereof
WO2025188842A1 (en) * 2024-03-08 2025-09-12 Spruce Biosciences, Inc. Amorphous solid dispersion of tildacerfont formulations

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU713673B2 (en) 1996-02-07 1999-12-09 Neurocrine Biosciences Inc. Pyrazolopyrimidines as crf receptor antagonists
ATE301657T1 (de) 1998-01-28 2005-08-15 Bristol Myers Squibb Pharma Co Azolo-pyrimidine
IL137019A (en) * 1998-01-28 2010-11-30 Du Pont Pharm Co 2,7 - dimethyl - 4 - (substituted amino) - 8 - arylpyrazolo [1,5-a] triazine derivatives and pharmaceutical compositions containing them
PL351069A1 (en) * 1999-12-08 2003-03-10 Pharmacia Corp Valdecoxib compositions
EP1722826A2 (en) * 2004-02-13 2006-11-22 SB Pharmco Puerto Rico Inc. Crf receptor antagonists, their preparations, their pharmaceutical composition and their uses
EP1869049B1 (en) * 2005-03-21 2009-03-04 Eli Lilly And Company Imidazopyridazine compounds
HRP20100516T1 (hr) * 2006-09-20 2010-10-31 Eli Lilly And Company Tiazolpirazolopirimidini kao antagonisti receptora crf1
JP5184536B2 (ja) * 2006-09-20 2013-04-17 イーライ リリー アンド カンパニー チオフェンピラゾロピリミジン化合物
DK2350079T3 (da) * 2008-10-02 2012-12-17 Lilly Co Eli Thiazolylpyrazolopyrimidinforbindelser som syntetiske mellemprodukter og dertil relaterede syntetiske fremgangsmåder
JP7285222B2 (ja) 2017-08-14 2023-06-01 スプルース バイオサイエンシズ インコーポレイテッド 副腎皮質刺激ホルモン放出因子受容体拮抗薬

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