JP2023063189A5 - - Google Patents

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Publication number
JP2023063189A5
JP2023063189A5 JP2021179359A JP2021179359A JP2023063189A5 JP 2023063189 A5 JP2023063189 A5 JP 2023063189A5 JP 2021179359 A JP2021179359 A JP 2021179359A JP 2021179359 A JP2021179359 A JP 2021179359A JP 2023063189 A5 JP2023063189 A5 JP 2023063189A5
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JP
Japan
Prior art keywords
flt3
cancer
crenolanib
pharmaceutical composition
tyrosine kinase
Prior art date
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Pending
Application number
JP2021179359A
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English (en)
Japanese (ja)
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JP2023063189A (ja
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Publication of JP2023063189A publication Critical patent/JP2023063189A/ja
Publication of JP2023063189A5 publication Critical patent/JP2023063189A5/ja
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JP2021179359A 2021-10-22 2021-11-02 以前の治療に対して再発性/不応性のflt3突然変異増殖性障害を治療するためのクレノラニブ Pending JP2023063189A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US202163270887P 2021-10-22 2021-10-22
US63/270,887 2021-10-22

Publications (2)

Publication Number Publication Date
JP2023063189A JP2023063189A (ja) 2023-05-09
JP2023063189A5 true JP2023063189A5 (enExample) 2024-10-08

Family

ID=86056882

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021179359A Pending JP2023063189A (ja) 2021-10-22 2021-11-02 以前の治療に対して再発性/不応性のflt3突然変異増殖性障害を治療するためのクレノラニブ

Country Status (3)

Country Link
US (3) US11857546B2 (enExample)
JP (1) JP2023063189A (enExample)
WO (1) WO2023069152A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2023063189A (ja) 2021-10-22 2023-05-09 アログ・ファーマシューティカルズ・インコーポレイテッド 以前の治療に対して再発性/不応性のflt3突然変異増殖性障害を治療するためのクレノラニブ
WO2025132479A1 (en) * 2023-12-18 2025-06-26 Institut National de la Santé et de la Recherche Médicale Flt3 inhibitor for modulating macrophages polarization

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2403876A (en) 1943-01-22 1946-07-09 Friedrich F Nord Glycol esters and method of producing same
US5990146A (en) 1997-08-20 1999-11-23 Warner-Lambert Company Benzimidazoles for inhibiting protein tyrosine kinase mediated cellular proliferation
CA2303830A1 (en) 1997-09-26 1999-04-08 Merck & Co., Inc. Novel angiogenesis inhibitors
UA75055C2 (uk) 1999-11-30 2006-03-15 Пфайзер Продактс Інк. Похідні бензоімідазолу, що використовуються як антипроліферативний засіб, фармацевтична композиція на їх основі
PA8580301A1 (es) 2002-08-28 2005-05-24 Pfizer Prod Inc Nuevos derivados de benzoimidazol utiles como agentes antiproliferativos
NZ571898A (en) 2003-06-24 2010-01-29 Pfizer Prod Inc Reaction of 2-chloro-8-benzyloxyquinoline with 2-nitrophenylamine in the presence of 1,2-bis(diphenylphosphino)ethane (dppe), palladium catalyst and a base
BR112015016282A2 (en) * 2013-01-07 2017-07-11 Arog Pharmaceuticals, Inc. crenolanib for treatment of mutated flt3 proliferative disorders
HK1257195A1 (zh) * 2016-11-02 2019-10-18 安罗格制药有限责任公司 用於治疗flt3突变型增殖性疾患相关突变的克莱拉尼
JP2023063189A (ja) 2021-10-22 2023-05-09 アログ・ファーマシューティカルズ・インコーポレイテッド 以前の治療に対して再発性/不応性のflt3突然変異増殖性障害を治療するためのクレノラニブ

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