JP2022539256A5 - - Google Patents

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Publication number
JP2022539256A5
JP2022539256A5 JP2022500099A JP2022500099A JP2022539256A5 JP 2022539256 A5 JP2022539256 A5 JP 2022539256A5 JP 2022500099 A JP2022500099 A JP 2022500099A JP 2022500099 A JP2022500099 A JP 2022500099A JP 2022539256 A5 JP2022539256 A5 JP 2022539256A5
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JP
Japan
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JP2022500099A
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Japanese (ja)
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JPWO2021003157A5 (https=
JP7595055B2 (ja
JP2022539256A (ja
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Priority claimed from PCT/US2020/040299 external-priority patent/WO2021003157A1/en
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Publication of JPWO2021003157A5 publication Critical patent/JPWO2021003157A5/ja
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JP2022500099A 2019-07-02 2020-06-30 eIF4E阻害4-オキソ-3,4-ジヒドロピリド[3,4-D]ピリミジン化合物 Active JP7595055B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962869662P 2019-07-02 2019-07-02
US62/869,662 2019-07-02
PCT/US2020/040299 WO2021003157A1 (en) 2019-07-02 2020-06-30 Eif4e-inhibiting 4-oxo-3,4-dihydropyrido[3,4-d]pyrimidine compounds

Publications (4)

Publication Number Publication Date
JP2022539256A JP2022539256A (ja) 2022-09-07
JP2022539256A5 true JP2022539256A5 (https=) 2023-06-16
JPWO2021003157A5 JPWO2021003157A5 (https=) 2023-06-16
JP7595055B2 JP7595055B2 (ja) 2024-12-05

Family

ID=71614984

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022500099A Active JP7595055B2 (ja) 2019-07-02 2020-06-30 eIF4E阻害4-オキソ-3,4-ジヒドロピリド[3,4-D]ピリミジン化合物

Country Status (15)

Country Link
US (2) US11286268B1 (https=)
EP (1) EP3994139A1 (https=)
JP (1) JP7595055B2 (https=)
KR (1) KR20220061945A (https=)
CN (1) CN114269756B (https=)
AR (1) AR119339A1 (https=)
AU (1) AU2020299362B2 (https=)
BR (1) BR112021026682A2 (https=)
CA (2) CA3085255A1 (https=)
CL (1) CL2021003573A1 (https=)
IL (1) IL289456A (https=)
PY (1) PY2031844A (https=)
TW (1) TWI748541B (https=)
UY (1) UY38773A (https=)
WO (1) WO2021003157A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20220378821A1 (en) * 2019-07-02 2022-12-01 Effector Therapeutics, Inc. Methods of treating braf-mutated cancer cells
EP4076438A4 (en) * 2019-12-18 2023-11-29 Merck Sharp & Dohme LLC BICYCLIC HETEROCYCLIC COMPOUNDS AND THEIR USE FOR THE TREATMENT OF HERPES VIRUSES
WO2021240337A1 (en) * 2020-05-27 2021-12-02 Effector Therapeutics, Inc. Covalent modifiers of eif4e inhibiting compounds
JP2023554521A (ja) 2020-12-22 2023-12-27 ファイザー・インク Eif4e阻害剤の固体形態
JP2025539263A (ja) * 2022-11-10 2025-12-04 リボメトリックス,インコーポレイティド eIF4E阻害剤としての化合物及び組成物、ならびにそれらの使用
TW202428278A (zh) * 2022-12-23 2024-07-16 大陸商南京聖和藥業股份有限公司 作為eIF4E抑制劑的化合物及其應用
IL326137A (en) 2023-07-28 2026-03-01 Cogent Biosciences Inc PI3K inhibitors
WO2025101516A1 (en) * 2023-11-06 2025-05-15 Ribometrix, Inc. Methods of using eif4e inhibitors for treating cancer
WO2025120599A1 (en) * 2023-12-08 2025-06-12 Ribometrix, Inc. METHODS OF USING eIF4E INHIBITORS FOR TREATING CANCER

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080255161A1 (en) * 2007-04-11 2008-10-16 Dmitry Koltun 3-HYDROQUINAZOLIN-4-ONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS
US20110065671A1 (en) * 2008-05-19 2011-03-17 Harris Joel M Bicyclic heterocycle derivatives and use thereof as gpr119 modulators
TW201412740A (zh) 2012-09-20 2014-04-01 Bayer Pharma AG 經取代之吡咯并嘧啶胺基苯并噻唑酮
WO2014179237A1 (en) 2013-04-29 2014-11-06 Vanderbilt University Substituted 3-benzylquinoxalin-4(3h)-one analogs as positive allosteric modulators of muscarinic acetycholine receptor m1
WO2015120350A2 (en) 2014-02-07 2015-08-13 Effector Therapeutics, Inc. Compositions and methods for treating fibrotic disease
TWI713455B (zh) 2014-06-25 2020-12-21 美商伊凡克特治療公司 MnK抑制劑及其相關方法

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