JP2022533747A5 - - Google Patents

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Publication number
JP2022533747A5
JP2022533747A5 JP2021569238A JP2021569238A JP2022533747A5 JP 2022533747 A5 JP2022533747 A5 JP 2022533747A5 JP 2021569238 A JP2021569238 A JP 2021569238A JP 2021569238 A JP2021569238 A JP 2021569238A JP 2022533747 A5 JP2022533747 A5 JP 2022533747A5
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JP
Japan
Prior art keywords
formula
compound
process according
reaction
salt
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JP2021569238A
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English (en)
Japanese (ja)
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JP7658916B2 (ja
JP2022533747A (ja
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Priority claimed from PCT/EP2020/064123 external-priority patent/WO2020234381A1/en
Publication of JP2022533747A publication Critical patent/JP2022533747A/ja
Publication of JP2022533747A5 publication Critical patent/JP2022533747A5/ja
Application granted granted Critical
Publication of JP7658916B2 publication Critical patent/JP7658916B2/ja
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JP2021569238A 2019-05-21 2020-05-20 Btk阻害剤を調製するためのプロセス及び中間体 Active JP7658916B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CNPCT/CN2019/087823 2019-05-21
CN2019087823 2019-05-21
PCT/EP2020/064123 WO2020234381A1 (en) 2019-05-21 2020-05-20 Processes and intermediates for preparing a btk inhibitor

Publications (3)

Publication Number Publication Date
JP2022533747A JP2022533747A (ja) 2022-07-25
JP2022533747A5 true JP2022533747A5 (cg-RX-API-DMAC10.html) 2024-12-09
JP7658916B2 JP7658916B2 (ja) 2025-04-08

Family

ID=70857160

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021569238A Active JP7658916B2 (ja) 2019-05-21 2020-05-20 Btk阻害剤を調製するためのプロセス及び中間体

Country Status (11)

Country Link
US (1) US12215110B2 (cg-RX-API-DMAC10.html)
EP (1) EP3972977A1 (cg-RX-API-DMAC10.html)
JP (1) JP7658916B2 (cg-RX-API-DMAC10.html)
KR (1) KR20220011668A (cg-RX-API-DMAC10.html)
CN (1) CN113874378A (cg-RX-API-DMAC10.html)
AU (1) AU2020278162A1 (cg-RX-API-DMAC10.html)
BR (1) BR112021022347A2 (cg-RX-API-DMAC10.html)
CA (1) CA3135240A1 (cg-RX-API-DMAC10.html)
IL (1) IL288154A (cg-RX-API-DMAC10.html)
MX (1) MX2021014246A (cg-RX-API-DMAC10.html)
WO (1) WO2020234381A1 (cg-RX-API-DMAC10.html)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12450495B2 (en) 2022-06-13 2025-10-21 International Business Machines Corporation Neural capacitance: neural network selection via edge dynamics

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2529621B1 (en) * 2006-09-22 2016-10-05 Pharmacyclics LLC Inhibitors of bruton's tyrosine kinase
UY32531A (es) 2009-03-31 2010-10-29 Boehringer Ingelheim Int Nuevos compuestos para el tratamiento de trastornos del snc
CN103121999A (zh) * 2012-08-29 2013-05-29 苏州迪飞医药科技有限公司 一种酪氨酸激酶抑制剂pci-32765的合成方法
EP2970291B1 (en) * 2013-03-15 2022-05-11 Janssen Pharmaceutica, N.V. Processes and intermediates for preparing a medicament
US9156847B2 (en) 2013-03-15 2015-10-13 Janssen Pharmaceutica Nv Processes and intermediates for preparing a medicament
MX365614B (es) 2013-10-17 2019-06-07 Blueprint Medicines Corp Composiciones utiles para tratar trastornos relacionados con kit.
MA41350A (fr) 2015-01-14 2017-11-21 Janssen Pharmaceutica Nv Synthèse d'un inhibiteur de la tyrosine kinase de bruton
RU2712440C2 (ru) 2015-02-12 2020-01-29 Шанхай Дьюд Медикал Сайенс Энд Текнолоджи Ко., Лтд Способ получения ибрутиниба

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