JP2022521955A5 - - Google Patents

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Publication number
JP2022521955A5
JP2022521955A5 JP2021549617A JP2021549617A JP2022521955A5 JP 2022521955 A5 JP2022521955 A5 JP 2022521955A5 JP 2021549617 A JP2021549617 A JP 2021549617A JP 2021549617 A JP2021549617 A JP 2021549617A JP 2022521955 A5 JP2022521955 A5 JP 2022521955A5
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JP
Japan
Prior art keywords
group
alkyl
use described
compound
hydrogen
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JP2021549617A
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English (en)
Japanese (ja)
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JP2022521955A (ja
JP7578602B2 (ja
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Priority claimed from PCT/IB2020/000160 external-priority patent/WO2020174283A1/en
Publication of JP2022521955A publication Critical patent/JP2022521955A/ja
Publication of JP2022521955A5 publication Critical patent/JP2022521955A5/ja
Application granted granted Critical
Publication of JP7578602B2 publication Critical patent/JP7578602B2/ja
Active legal-status Critical Current
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JP2021549617A 2019-02-25 2020-02-24 P2x3修飾薬での治療 Active JP7578602B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962810163P 2019-02-25 2019-02-25
US62/810,163 2019-02-25
PCT/IB2020/000160 WO2020174283A1 (en) 2019-02-25 2020-02-24 Treatment with p2x3 modulators

Publications (3)

Publication Number Publication Date
JP2022521955A JP2022521955A (ja) 2022-04-13
JP2022521955A5 true JP2022521955A5 (https=) 2023-02-24
JP7578602B2 JP7578602B2 (ja) 2024-11-06

Family

ID=72239247

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021549617A Active JP7578602B2 (ja) 2019-02-25 2020-02-24 P2x3修飾薬での治療

Country Status (8)

Country Link
US (1) US12485125B2 (https=)
EP (1) EP3930722A4 (https=)
JP (1) JP7578602B2 (https=)
CN (1) CN113727716A (https=)
AU (1) AU2020228760A1 (https=)
CA (1) CA3131312A1 (https=)
IL (1) IL285772A (https=)
WO (1) WO2020174283A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7578602B2 (ja) 2019-02-25 2024-11-06 グラクソスミスクライン、インテレクチュアル、プロパティー、(ナンバー3)、リミテッド P2x3修飾薬での治療
EP4103564A4 (en) * 2020-02-14 2024-05-01 GlaxoSmithKline Intellectual Property (No.3) Limited P2X3 MODULATORS
WO2021244634A1 (zh) * 2020-06-05 2021-12-09 武汉人福创新药物研发中心有限公司 咪唑并吡啶类化合物及其用途
WO2022161462A1 (zh) * 2021-01-29 2022-08-04 上海海雁医药科技有限公司 吗啉衍生物及其药物组合物和用途
CN115043836B (zh) * 2021-08-20 2023-07-18 苏州璞正医药有限公司 一种咪唑并吡啶衍生物的p2x3受体选择性调节剂及其药物用途
GB202212749D0 (en) * 2022-09-01 2022-10-19 Gesynta Pharma Ab New uses

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HRP20250864T1 (hr) * 2018-11-13 2025-09-26 Glaxosmithkline Intellectual Property (No. 3) Limited Kristalni oblici p2x3 modulatora metil (s)‑2‑((2‑(2,6‑difluoro‑4‑(metilkarbamoil)fenil)‑7‑metilimidazo[1,2‑a] piridin‑3‑il)metil)morfolin‑4‑karboksilata
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JP7578602B2 (ja) 2019-02-25 2024-11-06 グラクソスミスクライン、インテレクチュアル、プロパティー、(ナンバー3)、リミテッド P2x3修飾薬での治療
CN115427419B (zh) 2020-02-14 2026-04-21 葛兰素史密斯克莱知识产权(第3号)有限公司 P2x3拮抗剂的制备
EP4103564A4 (en) 2020-02-14 2024-05-01 GlaxoSmithKline Intellectual Property (No.3) Limited P2X3 MODULATORS

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