JP2022521859A5 - - Google Patents

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Publication number
JP2022521859A5
JP2022521859A5 JP2021571055A JP2021571055A JP2022521859A5 JP 2022521859 A5 JP2022521859 A5 JP 2022521859A5 JP 2021571055 A JP2021571055 A JP 2021571055A JP 2021571055 A JP2021571055 A JP 2021571055A JP 2022521859 A5 JP2022521859 A5 JP 2022521859A5
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JP
Japan
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alkyl
compound
cycloalkyl
alkoxy
heteroalkyl
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JP2021571055A
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English (en)
Japanese (ja)
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JP2022521859A (ja
JP7615056B2 (ja
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Priority claimed from PCT/CN2020/074696 external-priority patent/WO2020168939A1/zh
Publication of JP2022521859A publication Critical patent/JP2022521859A/ja
Publication of JP2022521859A5 publication Critical patent/JP2022521859A5/ja
Priority to JP2024231551A priority Critical patent/JP7821259B2/ja
Application granted granted Critical
Publication of JP7615056B2 publication Critical patent/JP7615056B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021571055A 2019-02-19 2020-02-11 複素環化合物、これを含む薬物組成物、その製造方法および使用 Active JP7615056B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024231551A JP7821259B2 (ja) 2019-02-19 2024-12-27 複素環化合物、これを含む薬物組成物、その製造方法および使用

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
CN201910124584.6 2019-02-19
CN201910124584 2019-02-19
CN201910437878 2019-05-24
CN201910437878.4 2019-05-24
CN201910932095.3 2019-09-29
CN201910932095 2019-09-29
PCT/CN2020/074696 WO2020168939A1 (zh) 2019-02-19 2020-02-11 杂环化合物、包含其的药物组合物及其制备方法和用途

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024231551A Division JP7821259B2 (ja) 2019-02-19 2024-12-27 複素環化合物、これを含む薬物組成物、その製造方法および使用

Publications (3)

Publication Number Publication Date
JP2022521859A JP2022521859A (ja) 2022-04-12
JP2022521859A5 true JP2022521859A5 (https=) 2023-08-29
JP7615056B2 JP7615056B2 (ja) 2025-01-16

Family

ID=72143544

Family Applications (2)

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JP2021571055A Active JP7615056B2 (ja) 2019-02-19 2020-02-11 複素環化合物、これを含む薬物組成物、その製造方法および使用
JP2024231551A Active JP7821259B2 (ja) 2019-02-19 2024-12-27 複素環化合物、これを含む薬物組成物、その製造方法および使用

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JP2024231551A Active JP7821259B2 (ja) 2019-02-19 2024-12-27 複素環化合物、これを含む薬物組成物、その製造方法および使用

Country Status (16)

Country Link
US (1) US20220144847A1 (https=)
EP (1) EP3929198A4 (https=)
JP (2) JP7615056B2 (https=)
KR (1) KR20210131314A (https=)
CN (3) CN117263945A (https=)
AU (1) AU2020226422C1 (https=)
BR (1) BR112021016299A2 (https=)
CA (1) CA3130245A1 (https=)
CL (1) CL2021002205A1 (https=)
CO (1) CO2021011023A2 (https=)
IL (1) IL285378B2 (https=)
MX (1) MX2021009971A (https=)
PH (1) PH12021552004A1 (https=)
SA (1) SA521430084B1 (https=)
SG (1) SG11202107848TA (https=)
WO (1) WO2020168939A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022022398A1 (zh) * 2020-07-28 2022-02-03 四川科伦博泰生物医药股份有限公司 一种嘧啶类化合物的盐和晶型及其制备方法
KR20230159367A (ko) * 2021-03-24 2023-11-21 쓰촨 케룬-바이오테크 바이오파마수티컬 컴퍼니 리미티드 키나아제 약물 내성 돌연변이와 관련된 질병의 치료에있어서의 헤테로사이클릭 화합물의 용도 및 그 방법
CN114235976B (zh) * 2021-11-09 2023-11-03 暨南大学 一种含氮杂环有机化合物中间产物的合成和分析方法
CN120897743A (zh) 2023-05-19 2025-11-04 四川科伦博泰生物医药股份有限公司 杂环化合物治疗与ret基因改变相关疾病的用途和方法
WO2025256440A1 (zh) * 2024-06-14 2025-12-18 四川科伦博泰生物医药股份有限公司 含杂环化合物富马酸盐的制备方法
WO2026017002A1 (zh) * 2024-07-16 2026-01-22 四川科伦博泰生物医药股份有限公司 以杂环化合物为活性成分的药物组合物、其制备方法及用途
GB202410599D0 (en) 2024-07-19 2024-09-04 Ellipses Pharma Ltd Therapeutics useful synergistic combinations

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA200707227B (en) * 2005-02-28 2009-08-26 Japan Tobacco Inc Novel aminopyridine compound with syk inhibitory activity
BRPI0607062A2 (pt) 2005-02-28 2009-08-04 Japan Tobacco Inc composto de aminopiridina com atividade inibidora de syk, composição farmacêutica e agente terapêutico compreendendo os mesmos
WO2008013622A2 (en) * 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
US20080234267A1 (en) * 2007-03-20 2008-09-25 Karen Elizabeth Lackey Compounds and Methods of Treatment
JP2010208945A (ja) * 2007-06-01 2010-09-24 Mitsubishi Tanabe Pharma Corp 複素環化合物
ES2539170T3 (es) 2010-01-12 2015-06-26 Ab Science Inhibidores de quinasas de oxazol
JP2013107824A (ja) 2010-03-17 2013-06-06 Dainippon Sumitomo Pharma Co Ltd 新規単環ピリミジン誘導体
EP2634176A4 (en) * 2010-10-28 2014-04-16 Nippon Shinyaku Co Ltd PYRIDINE DERIVATIVE AND MEDICINAL AGENT
US9145391B2 (en) * 2011-05-10 2015-09-29 Merck Sharp & Dohme Corp. Bipyridylaminopyridines as Syk inhibitors
WO2016127074A1 (en) 2015-02-06 2016-08-11 Blueprint Medicines Corporation 2-(pyridin-3-yl)-pyrimidine derivatives as ret inhibitors
SI3371171T1 (sl) 2015-11-02 2024-03-29 Blueprint Medicines Corporation Inhibitorji ret
TWI704148B (zh) 2016-10-10 2020-09-11 美商亞雷生物製藥股份有限公司 作為ret激酶抑制劑之經取代吡唑并[1,5-a]吡啶化合物
WO2018136661A1 (en) 2017-01-18 2018-07-26 Andrews Steven W SUBSTITUTED PYRAZOLO[1,5-a]PYRAZINE COMPOUNDS AS RET KINASE INHIBITORS

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