JP2022519375A5 - - Google Patents

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Publication number
JP2022519375A5
JP2022519375A5 JP2021546211A JP2021546211A JP2022519375A5 JP 2022519375 A5 JP2022519375 A5 JP 2022519375A5 JP 2021546211 A JP2021546211 A JP 2021546211A JP 2021546211 A JP2021546211 A JP 2021546211A JP 2022519375 A5 JP2022519375 A5 JP 2022519375A5
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JP
Japan
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JP2021546211A
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Japanese (ja)
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JP2022519375A (ja
JPWO2020165734A5 (https=
JP7493521B2 (ja
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Priority claimed from PCT/IB2020/051031 external-priority patent/WO2020165734A1/en
Publication of JP2022519375A publication Critical patent/JP2022519375A/ja
Publication of JPWO2020165734A5 publication Critical patent/JPWO2020165734A5/ja
Publication of JP2022519375A5 publication Critical patent/JP2022519375A5/ja
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Publication of JP7493521B2 publication Critical patent/JP7493521B2/ja
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JP2021546211A 2019-02-12 2020-02-10 Tno155及びリボシクリブを含む医薬組合せ Active JP7493521B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962804708P 2019-02-12 2019-02-12
US62/804,708 2019-02-12
PCT/IB2020/051031 WO2020165734A1 (en) 2019-02-12 2020-02-10 Pharmaceutical combination comprising tno155 and ribociclib

Publications (4)

Publication Number Publication Date
JP2022519375A JP2022519375A (ja) 2022-03-23
JPWO2020165734A5 JPWO2020165734A5 (https=) 2023-02-17
JP2022519375A5 true JP2022519375A5 (https=) 2023-02-17
JP7493521B2 JP7493521B2 (ja) 2024-05-31

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ID=69724013

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021546211A Active JP7493521B2 (ja) 2019-02-12 2020-02-10 Tno155及びリボシクリブを含む医薬組合せ

Country Status (14)

Country Link
US (1) US12343344B2 (https=)
EP (1) EP3923941B1 (https=)
JP (1) JP7493521B2 (https=)
KR (1) KR20210126653A (https=)
CN (1) CN113382731A (https=)
AU (3) AU2020222296B2 (https=)
BR (1) BR112021015632A2 (https=)
CA (1) CA3127286A1 (https=)
CL (1) CL2021002099A1 (https=)
ES (1) ES3063733T3 (https=)
IL (1) IL284835B2 (https=)
MX (1) MX2021009563A (https=)
TW (1) TWI831916B (https=)
WO (1) WO2020165734A1 (https=)

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JP2022502385A (ja) 2018-09-29 2022-01-11 ノバルティス アーゲー Shp2の活性を阻害するための化合物の製造方法
WO2020072656A1 (en) 2018-10-03 2020-04-09 Gilead Sciences, Inc. Imidozopyrimidine derivatives
MX2021009562A (es) * 2019-02-12 2021-09-08 Novartis Ag Combinacion farmaceutica que comprende tno155 y un inhibidor de pd-1.
IL299131A (en) 2020-06-18 2023-02-01 Revolution Medicines Inc Methods for delaying, preventing and treating acquired resistance to RAS inhibitors
CN115916786B (zh) 2020-07-08 2025-10-17 诺华股份有限公司 用于抑制shp2活性的化合物和组合物的制造
MX2023002248A (es) 2020-09-03 2023-05-16 Revolution Medicines Inc Uso de inhibidores de sos1 para tratar neoplasias malignas con mutaciones de shp2.
MX2023003060A (es) 2020-09-15 2023-04-05 Revolution Medicines Inc Derivados indolicos como inhibidores de ras en el tratamiento del cancer.
AU2022268962A1 (en) 2021-05-05 2023-12-14 Revolution Medicines, Inc. Ras inhibitors for the treatment of cancer
IL308234A (en) * 2021-05-05 2024-01-01 Huyabio Int Llc Monotherapy with an SHP2 inhibitor and its uses
WO2022235866A1 (en) 2021-05-05 2022-11-10 Revolution Medicines, Inc. Covalent ras inhibitors and uses thereof
CA3217393A1 (en) 2021-05-05 2022-11-10 Elena S. Koltun Ras inhibitors
CN117177752A (zh) * 2021-05-05 2023-12-05 诺华股份有限公司 用于治疗mpnst的化合物和组合物
US20240293422A1 (en) * 2021-06-24 2024-09-05 Erasca, Inc. Shp2 and cdk4/6 inhibitors combination therapies for the treatment of cancer
AR127308A1 (es) 2021-10-08 2024-01-10 Revolution Medicines Inc Inhibidores ras
TW202342040A (zh) 2022-02-21 2023-11-01 瑞士商諾華公司 藥物配製物
CN119136806A (zh) 2022-03-08 2024-12-13 锐新医药公司 用于治疗免疫难治性肺癌的方法
WO2023240263A1 (en) 2022-06-10 2023-12-14 Revolution Medicines, Inc. Macrocyclic ras inhibitors
EP4626890A1 (en) 2022-12-01 2025-10-08 KRKA, d.d., Novo mesto Ribociclib salts and formulations thereof
KR20240097396A (ko) 2022-12-20 2024-06-27 재단법인대구경북과학기술원 리보시클립을 유효성분으로 포함하는 신경염증 또는 퇴행성 뇌질환의 예방 또는 치료용 약학적 조성물
EP4687905A1 (en) 2023-03-30 2026-02-11 Revolution Medicines, Inc. Compositions for inducing ras gtp hydrolysis and uses thereof
KR20260005904A (ko) 2023-04-07 2026-01-12 레볼루션 메디슨즈, 인크. 매크로사이클릭 ras 억제제
CN121263418A (zh) 2023-04-07 2026-01-02 锐新医药公司 大环ras抑制剂
AU2024252105A1 (en) 2023-04-14 2025-10-16 Revolution Medicines, Inc. Crystalline forms of ras inhibitors, compositions containing the same, and methods of use thereof
KR20250172857A (ko) 2023-04-14 2025-12-09 레볼루션 메디슨즈, 인크. Ras 억제제의 결정형
AU2024265078A1 (en) 2023-05-04 2025-12-11 Revolution Medicines, Inc. Combination therapy for a ras related disease or disorder
IL326136A (en) 2023-08-07 2026-03-01 Revolution Medicines Inc RMC-6291 for use in the treatment of a disease or disorder associated with the RAS protein
US20250154171A1 (en) 2023-10-12 2025-05-15 Revolution Medicines, Inc. Ras inhibitors
WO2025171296A1 (en) 2024-02-09 2025-08-14 Revolution Medicines, Inc. Ras inhibitors
WO2025240847A1 (en) 2024-05-17 2025-11-20 Revolution Medicines, Inc. Ras inhibitors
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WO2025265060A1 (en) 2024-06-21 2025-12-26 Revolution Medicines, Inc. Therapeutic compositions and methods for managing treatment-related effects
WO2026015796A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
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WO2026015825A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Use of ras inhibitor for treating pancreatic cancer
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WO2026072904A2 (en) 2024-09-26 2026-04-02 Revolution Medicines, Inc. Compositions and methods for treating lung cancer

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MX2021009562A (es) 2019-02-12 2021-09-08 Novartis Ag Combinacion farmaceutica que comprende tno155 y un inhibidor de pd-1.

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