JP2022514194A - 自殺のリスクを低減し、うつ病を迅速に軽減するためのガボキサドール - Google Patents

自殺のリスクを低減し、うつ病を迅速に軽減するためのガボキサドール Download PDF

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JP2022514194A
JP2022514194A JP2021529111A JP2021529111A JP2022514194A JP 2022514194 A JP2022514194 A JP 2022514194A JP 2021529111 A JP2021529111 A JP 2021529111A JP 2021529111 A JP2021529111 A JP 2021529111A JP 2022514194 A JP2022514194 A JP 2022514194A
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treatment
gaboxador
suicide
pharmaceutically acceptable
administration
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JP2021529111A
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Japanese (ja)
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JP2022514194A5 (https=
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オステン、パヴェル
ボールドウィン、クリスティン
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Certego Therapeutics Inc
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Certego Therapeutics Inc
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants

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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
JP2021529111A 2018-11-21 2019-11-21 自殺のリスクを低減し、うつ病を迅速に軽減するためのガボキサドール Pending JP2022514194A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862770287P 2018-11-21 2018-11-21
US62/770,287 2018-11-21
PCT/US2019/062554 WO2020106927A1 (en) 2018-11-21 2019-11-21 Gaboxadol for reducing risk of suicide and rapid relief of depression

Publications (2)

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JP2022514194A true JP2022514194A (ja) 2022-02-10
JP2022514194A5 JP2022514194A5 (https=) 2022-11-18

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JP2021529111A Pending JP2022514194A (ja) 2018-11-21 2019-11-21 自殺のリスクを低減し、うつ病を迅速に軽減するためのガボキサドール

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US (3) US20220008398A1 (https=)
EP (1) EP3883566A4 (https=)
JP (1) JP2022514194A (https=)
KR (1) KR20210110585A (https=)
CN (1) CN113395962A (https=)
AU (1) AU2019384157A1 (https=)
BR (1) BR112021009944A2 (https=)
CA (1) CA3120856A1 (https=)
GB (1) GB2594616A (https=)
IL (1) IL283311A (https=)
MX (1) MX2021005992A (https=)
SG (1) SG11202105358RA (https=)
WO (1) WO2020106927A1 (https=)

Cited By (1)

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Publication number Priority date Publication date Assignee Title
JP2024020037A (ja) * 2022-08-01 2024-02-14 学校法人順天堂 痛みと痒みのバイオマーカー

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JOP20200195A1 (ar) 2014-09-08 2017-06-16 Sage Therapeutics Inc سترويدات وتركيبات نشطة عصبياً، واستخداماتها
KR20240157128A (ko) 2016-03-08 2024-10-31 세이지 테라퓨틱스, 인크. 신경활성 스테로이드, 조성물, 및 그의 용도
EP3481387A4 (en) * 2016-08-11 2020-04-08 Ovid Therapeutics Inc METHOD AND COMPOSITIONS FOR TREATING EPILEPTIC DISEASES
US10071083B2 (en) * 2017-02-03 2018-09-11 Ovid Therapeutics Inc Use of gaboxadol in the treatment of tinnitus
ES2907692T3 (es) 2017-12-29 2022-04-26 Celon Pharma Sa Composición de ketamina de polvo seco para su administración por vía pulmonar en la depresión resistente al tratamiento
JP2022514194A (ja) * 2018-11-21 2022-02-10 セルテゴ セラピューティクス インコーポレイテッド 自殺のリスクを低減し、うつ病を迅速に軽減するためのガボキサドール
MX2022014599A (es) 2020-05-20 2022-12-16 Certego Therapeutics Inc Gaboxadol deuterado en anillo y su uso para el tratamiento de trastornos psiquiatricos.

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Cited By (1)

* Cited by examiner, † Cited by third party
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Publication number Publication date
GB202108720D0 (en) 2021-08-04
US20200155522A1 (en) 2020-05-21
KR20210110585A (ko) 2021-09-08
US20220054461A1 (en) 2022-02-24
AU2019384157A1 (en) 2021-06-17
US20220008398A1 (en) 2022-01-13
CA3120856A1 (en) 2020-05-28
CN113395962A (zh) 2021-09-14
EP3883566A1 (en) 2021-09-29
BR112021009944A2 (pt) 2021-08-17
GB2594616A (en) 2021-11-03
WO2020106927A1 (en) 2020-05-28
SG11202105358RA (en) 2021-06-29
IL283311A (en) 2021-07-29
US11123332B2 (en) 2021-09-21
MX2021005992A (es) 2021-09-14
EP3883566A4 (en) 2022-09-07

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