JP2022500402A5 - - Google Patents
Info
- Publication number
- JP2022500402A5 JP2022500402A5 JP2021513827A JP2021513827A JP2022500402A5 JP 2022500402 A5 JP2022500402 A5 JP 2022500402A5 JP 2021513827 A JP2021513827 A JP 2021513827A JP 2021513827 A JP2021513827 A JP 2021513827A JP 2022500402 A5 JP2022500402 A5 JP 2022500402A5
- Authority
- JP
- Japan
- Prior art keywords
- triazolo
- pyrimidine
- methyl
- alkyl
- amino
- Prior art date
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024096058A JP2024123079A (ja) | 2018-09-12 | 2024-06-13 | トリアゾロ－ピリミジン化合物およびそれらの使用 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2018/105220 | 2018-09-12 | ||
| CN2018105220 | 2018-09-12 | ||
| PCT/CN2019/105591 WO2020052631A1 (en) | 2018-09-12 | 2019-09-12 | Triazolo-pyrimidine compounds and uses thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024096058A Division JP2024123079A (ja) | 2018-09-12 | 2024-06-13 | トリアゾロ－ピリミジン化合物およびそれらの使用 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2022500402A JP2022500402A (ja) | 2022-01-04 |
| JP2022500402A5 true JP2022500402A5 (https=) | 2022-09-05 |
| JPWO2020052631A5 JPWO2020052631A5 (https=) | 2022-09-05 |
| JP7572353B2 JP7572353B2 (ja) | 2024-10-23 |
Family
ID=69778192
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021513827A Active JP7572353B2 (ja) | 2018-09-12 | 2019-09-12 | トリアゾロ－ピリミジン化合物およびそれらの使用 |
| JP2024096058A Pending JP2024123079A (ja) | 2018-09-12 | 2024-06-13 | トリアゾロ－ピリミジン化合物およびそれらの使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024096058A Pending JP2024123079A (ja) | 2018-09-12 | 2024-06-13 | トリアゾロ－ピリミジン化合物およびそれらの使用 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US10858365B2 (https=) |
| EP (1) | EP3849983A4 (https=) |
| JP (2) | JP7572353B2 (https=) |
| KR (1) | KR102841843B1 (https=) |
| CN (3) | CN111635408B (https=) |
| AR (1) | AR116315A1 (https=) |
| AU (1) | AU2019340767B9 (https=) |
| BR (1) | BR112021004774A2 (https=) |
| CA (1) | CA3111869A1 (https=) |
| MX (1) | MX2021002998A (https=) |
| TW (1) | TWI820209B (https=) |
| WO (1) | WO2020052631A1 (https=) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11066410B2 (en) * | 2017-03-24 | 2021-07-20 | 3100 Central Expressway Llc | Fused triazolo-pyrimidine compounds having useful pharmaceutical application |
| WO2019018584A1 (en) | 2017-07-18 | 2019-01-24 | GiraFpharma LLC | HETEROCYCLIC COMPOUNDS AS ADENOSINE ANTAGONISTS |
| BR122023024273A2 (pt) | 2018-02-27 | 2024-02-20 | Incyte Corporation | Compostos imidazopirimidinas e triazolopirimidinas, seus usos, método para inibir uma atividade de um receptor de adenosina e composição farmacêutica dos mesmos |
| US11220510B2 (en) | 2018-04-09 | 2022-01-11 | Incyte Corporation | Pyrrole tricyclic compounds as A2A / A2B inhibitors |
| WO2019222677A1 (en) | 2018-05-18 | 2019-11-21 | Incyte Corporation | Fused pyrimidine derivatives as a2a / a2b inhibitors |
| GEP20237548B (en) | 2018-07-05 | 2023-10-10 | Incyte Corp | Fused pyrazine derivatives as a2a /a2b inhibitors |
| AR116315A1 (es) * | 2018-09-12 | 2021-04-21 | Dizal Jiangsu Pharmaceutical Co Ltd | Compuestos de triazolo-pirimidina y usos de los mismos |
| EP3911324A4 (en) | 2019-01-18 | 2022-08-17 | Nuvation Bio Inc. | 1,8-NAPHTHYRIDINONE COMPOUNDS AND THEIR USES |
| EP3911323A4 (en) | 2019-01-18 | 2022-11-16 | Nuvation Bio Inc. | HETEROCYCLIC COMPOUNDS AS ADENOSINE ANTAGONISTS |
| TWI829857B (zh) | 2019-01-29 | 2024-01-21 | 美商英塞特公司 | 作為a2a / a2b抑制劑之吡唑并吡啶及三唑并吡啶 |
| US20210061809A1 (en) * | 2019-08-26 | 2021-03-04 | Incyte Corporation | Triazolopyrimidines as a2a / a2b inhibitors |
| WO2021156439A1 (en) | 2020-02-06 | 2021-08-12 | Astrazeneca Ab | Triazole compounds as adenosine receptor antagonists |
| CN120022278A (zh) * | 2023-11-22 | 2025-05-23 | 英诺湖医药(杭州)有限公司 | 用于治疗癌症的化合物 |
| CN117865963B (zh) * | 2023-12-15 | 2026-02-24 | 上海凌凯科技股份有限公司 | 一种嘧啶酮衍生物的合成方法及嘧啶酮衍生物 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4195729B2 (ja) * | 1997-03-24 | 2008-12-10 | 協和醗酵工業株式会社 | ［１，２，４］トリアゾロ［１，５−ｃ］ピリミジン誘導体 |
| JPWO2002079204A1 (ja) | 2001-03-28 | 2004-07-22 | 協和醗酵工業株式会社 | ８−チアゾリル［１，２，４］トリアゾロ［１，５−ｃ］ピリミジン誘導体 |
| PE20030739A1 (es) | 2001-11-30 | 2003-08-28 | Schering Corp | Antagonistas del receptor de adenosina a2a |
| EP1544200A1 (en) | 2002-09-24 | 2005-06-22 | Kyowa Hakko Kogyo Co., Ltd. | 1,2,4 -TRIAZOLO 1,5-c PYRIMIDINE DERIVATIVE |
| CN110214012B (zh) * | 2017-01-20 | 2023-05-09 | 艾库斯生物科学有限公司 | 用于治疗癌症相关疾病的唑嘧啶 |
| CN109963854B (zh) * | 2017-03-16 | 2022-04-12 | 江苏恒瑞医药股份有限公司 | 杂芳基并[4,3-c]嘧啶-5-胺类衍生物、其制备方法及其在医药上的应用 |
| PL3611174T3 (pl) * | 2017-04-07 | 2022-08-08 | Medshine Discovery Inc. | Pochodne [1,2,4]triazolo[1,5-c]pirymidyny jako inhibitor receptora a2a |
| CN109535161B (zh) * | 2017-09-22 | 2021-09-03 | 江苏恒瑞医药股份有限公司 | 三唑并嘧啶类衍生物、其制备方法及其在医药上的应用 |
| BR122023024273A2 (pt) * | 2018-02-27 | 2024-02-20 | Incyte Corporation | Compostos imidazopirimidinas e triazolopirimidinas, seus usos, método para inibir uma atividade de um receptor de adenosina e composição farmacêutica dos mesmos |
| CN112105617B (zh) * | 2018-04-28 | 2022-04-05 | 南京明德新药研发有限公司 | 一种三唑并嘧啶类化合物的晶型、盐型及其制备方法 |
| AR116315A1 (es) * | 2018-09-12 | 2021-04-21 | Dizal Jiangsu Pharmaceutical Co Ltd | Compuestos de triazolo-pirimidina y usos de los mismos |
-
2019
- 2019-09-11 AR ARP190102589A patent/AR116315A1/es unknown
- 2019-09-11 TW TW108132759A patent/TWI820209B/zh active
- 2019-09-12 JP JP2021513827A patent/JP7572353B2/ja active Active
- 2019-09-12 CA CA3111869A patent/CA3111869A1/en active Pending
- 2019-09-12 CN CN202010656938.4A patent/CN111635408B/zh active Active
- 2019-09-12 CN CN202010657655.1A patent/CN112279852B/zh active Active
- 2019-09-12 WO PCT/CN2019/105591 patent/WO2020052631A1/en not_active Ceased
- 2019-09-12 BR BR112021004774-3A patent/BR112021004774A2/pt unknown
- 2019-09-12 AU AU2019340767A patent/AU2019340767B9/en active Active
- 2019-09-12 KR KR1020217010809A patent/KR102841843B1/ko active Active
- 2019-09-12 CN CN201980006436.2A patent/CN111601809A/zh active Pending
- 2019-09-12 EP EP19859380.8A patent/EP3849983A4/en active Pending
- 2019-09-12 MX MX2021002998A patent/MX2021002998A/es unknown
-
2020
- 2020-06-24 US US16/910,334 patent/US10858365B2/en active Active
- 2020-09-22 US US17/027,740 patent/US11629147B2/en active Active
-
2024
- 2024-06-13 JP JP2024096058A patent/JP2024123079A/ja active Pending
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